AR021500A2 - Compuesto intermediario para preparar compuestos herbicidas 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona y 3-(1,2-benzisotiazol)-e isoxazol-5-il)-4(3h)pirimidinona o tiona - Google Patents
Compuesto intermediario para preparar compuestos herbicidas 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona y 3-(1,2-benzisotiazol)-e isoxazol-5-il)-4(3h)pirimidinona o tionaInfo
- Publication number
- AR021500A2 AR021500A2 ARP990105577A ARP990105577A AR021500A2 AR 021500 A2 AR021500 A2 AR 021500A2 AR P990105577 A ARP990105577 A AR P990105577A AR P990105577 A ARP990105577 A AR P990105577A AR 021500 A2 AR021500 A2 AR 021500A2
- Authority
- AR
- Argentina
- Prior art keywords
- groups
- halogen
- alkyl
- isoxazol
- group
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 5
- AXLOCHLTNQDFFS-BESJYZOMSA-N azastene Chemical compound C([C@H]1[C@@H]2CC[C@@]([C@]2(CC[C@@H]1[C@@]1(C)C2)C)(O)C)C=C1C(C)(C)C1=C2C=NO1 AXLOCHLTNQDFFS-BESJYZOMSA-N 0.000 title 1
- 230000002363 herbicidal effect Effects 0.000 title 1
- 239000004009 herbicide Substances 0.000 title 1
- 229910052736 halogen Inorganic materials 0.000 abstract 5
- 150000002367 halogens Chemical group 0.000 abstract 5
- 229910052739 hydrogen Inorganic materials 0.000 abstract 5
- 239000001257 hydrogen Substances 0.000 abstract 5
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 5
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 4
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 3
- 229910052760 oxygen Inorganic materials 0.000 abstract 3
- 229910052717 sulfur Inorganic materials 0.000 abstract 3
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 2
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000000304 alkynyl group Chemical group 0.000 abstract 2
- 125000004429 atom Chemical group 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- PXBRQCKWGAHEHS-UHFFFAOYSA-N dichlorodifluoromethane Chemical group FC(F)(Cl)Cl PXBRQCKWGAHEHS-UHFFFAOYSA-N 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 abstract 1
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 abstract 1
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- 101150020251 NR13 gene Proteins 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 241001061127 Thione Species 0.000 abstract 1
- 125000004183 alkoxy alkyl group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000000051 benzyloxy group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])O* 0.000 abstract 1
- 125000002619 bicyclic group Chemical group 0.000 abstract 1
- RLDQYSHDFVSAPL-UHFFFAOYSA-L calcium;dithiocyanate Chemical group [Ca+2].[S-]C#N.[S-]C#N RLDQYSHDFVSAPL-UHFFFAOYSA-L 0.000 abstract 1
- 125000000392 cycloalkenyl group Chemical group 0.000 abstract 1
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 1
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000002950 monocyclic group Chemical group 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004043 oxo group Chemical group O=* 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 239000011593 sulfur Substances 0.000 abstract 1
- 125000000464 thioxo group Chemical group S=* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
- C07F9/6539—Five-membered rings
- C07F9/6541—Five-membered rings condensed with carbocyclic rings or carbocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Environmental Sciences (AREA)
- Plant Pathology (AREA)
- Agronomy & Crop Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Pest Control & Pesticides (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Un compuesto intermediario para preparar compuestos de 3-(1,2-benzisotiazol-e isoxazol-5-il)-2,4(1H,3H)-pirimidindiona o tiona de la formula (1) ycompuestos de 3-(1,2-benzisotiazol-e isoxazol-5-il)-4(3H)-pirimidinona o tiona de la formula (2) donde R1 y R2 son cada uno independientemente hidrogeno,halogeno, alquilo de C1-6, cicloalquilo de C3-7, haloalquilo de C1-6, alquenilo de C3-6, haloalquenilo de C3-6, alquinilo de C3-6, OR7, S(O)nR8 o NR9R10 ycuando R1 Y R2 tomados junto con los átomos a los que están unidos, representan un anillo de cuatro a siete miembros saturado o no saturado opcionalmenteinterrumpido por oxígeno, azufre o nitrogeno, y opcionalmente sustituido con uno o tres grupos metilo o uno o más átomos de halogeno; X es hidrogeno, halogenoo alquilo de C1-4; X1 es hidrogeno, halogeno, alquilo de C1-4, haloalquilo de C1-4, alcoxi de C1-4 o haloalcoxi de C1-4; Z es O o S(O)m; Y es halogeno, ciano,R12, X2R12, X3R12, X2X3R12 o X3X2R12; X2 es O, S(O)p o NR13; X3 es -C(=A3)-, -C(=NOR14)-o-C(=N-NR13R50); R4, R5, R6, R7, R8, R9, R10 y R14 son cada unoindependientemente hidrogeno, alquilo de C1-6, cicloalquilo de C3-7, alcoxialquilo de C2-8, alquenilo de C2-6, alquinilo o bencilo de C2-6;R12 es hidrogeno, ungrupo alquilo deC1-8, cicloalquilo de C3-7, alquenilo de C2-8, cicloalquenilo de C5-6 o alquinilo de C2-8, donde cada grupo está opcionalmente sustituido conuna combinacion de uno o seis átomos de halogeno, uno a tres grupos de alcoxi de C1-6, benciloxi o alquiltiode C1-6, uno o dos grupos haloalcoxi de C1-10,uno o dos grupos NR15R16, uno a tres grupos S(O)qR17, uno o dos grupos ciano, uno o dos grupos cicloalquilo de C3-7, un grupo tiociano, un grupo O(SO2)R17, ungrupo O(NO2), uno o dos grupos C(O)R18, uno odos grupos CO2R19, uno o dos C(O)SR19, uno o dos C(O)NR20R21, uno a tres grupos X4R22, uno o dos grupos P(O)(OR23)2, uno o dos Si(R24)3, un anillo de 4 a 10 miembros heterocíclico, monocíclico o bicíclico fusionado opcionalmente sustituido con cualquier combinacionde uno a dos grupos oxo, uno o dos grupos tioxo, uno a tres átomos de halogeno, uno a tres grupos de alquilo de C1-4, uno a tres grupos de haloalquilo C1-4
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US93145197A | 1997-09-17 | 1997-09-17 | |
| US12883198A | 1998-08-04 | 1998-08-04 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR021500A2 true AR021500A2 (es) | 2002-07-24 |
Family
ID=26826981
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP980104611A AR015168A1 (es) | 1997-09-17 | 1998-09-16 | Compuesto herbicida 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona o 3-(1,2-benzisotiazol)-e isoxazol-5-il)-4(3h)-pirimidinona o tiona, y procedimiento para preparar el compuesto 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona |
| ARP990105577A AR021500A2 (es) | 1997-09-17 | 1999-11-04 | Compuesto intermediario para preparar compuestos herbicidas 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona y 3-(1,2-benzisotiazol)-e isoxazol-5-il)-4(3h)pirimidinona o tiona |
| ARP990105578A AR021081A2 (es) | 1997-09-17 | 1999-11-04 | Un proceso para la preparacion de un compuesto intermediario para preparar compuestos herbicidas 3-(1,2-benzisotiazol) -e isoxazol-5-il) -2,4-(1h,3h)-pirimidindiona o tiona y 3-(1,2-benzisotiazol) -e isoxazol-5-il)-4(eh)- pirimidinona o tiona |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP980104611A AR015168A1 (es) | 1997-09-17 | 1998-09-16 | Compuesto herbicida 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona o 3-(1,2-benzisotiazol)-e isoxazol-5-il)-4(3h)-pirimidinona o tiona, y procedimiento para preparar el compuesto 3-(1,2-benzisotiazol)-e isoxazol-5-il)-2,4-(1h,3h)-pirimidindiona o tiona |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP990105578A AR021081A2 (es) | 1997-09-17 | 1999-11-04 | Un proceso para la preparacion de un compuesto intermediario para preparar compuestos herbicidas 3-(1,2-benzisotiazol) -e isoxazol-5-il) -2,4-(1h,3h)-pirimidindiona o tiona y 3-(1,2-benzisotiazol) -e isoxazol-5-il)-4(eh)- pirimidinona o tiona |
Country Status (24)
| Country | Link |
|---|---|
| EP (1) | EP0908457B1 (es) |
| JP (1) | JP2001516758A (es) |
| KR (1) | KR20010030612A (es) |
| CN (1) | CN1273585A (es) |
| AR (3) | AR015168A1 (es) |
| AT (1) | ATE227721T1 (es) |
| AU (2) | AU9392598A (es) |
| BG (1) | BG104336A (es) |
| BR (1) | BR9813017A (es) |
| CA (1) | CA2246221A1 (es) |
| CZ (1) | CZ2000861A3 (es) |
| DE (1) | DE69809370T2 (es) |
| ES (1) | ES2185118T3 (es) |
| HU (1) | HUP0004477A3 (es) |
| IL (1) | IL125947A0 (es) |
| MX (1) | MXPA00002661A (es) |
| NZ (1) | NZ331825A (es) |
| PL (1) | PL339350A1 (es) |
| SK (1) | SK3552000A3 (es) |
| TR (1) | TR200000679T2 (es) |
| TW (1) | TW474927B (es) |
| WO (1) | WO1999014216A1 (es) |
| YU (1) | YU15800A (es) |
| ZA (1) | ZA988435B (es) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6140270A (en) * | 1998-09-14 | 2000-10-31 | American Cyanamid Company | Process for the preparation of 6-(perfluoroalkyl) uracil compounds from 2-(N,N-disubstituted) amino-4-(perfluoroalkyl)-1,3-oxazin-6-one compounds |
| IL144776A0 (en) * | 1999-02-16 | 2002-06-30 | Basf Ag | Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils |
| EP1274708A1 (en) * | 2000-04-17 | 2003-01-15 | Basf Aktiengesellschaft | Herbicidal 3-heterocyclic substituted benzisothiazole and benzisoxazole compounds |
| US20040097728A1 (en) * | 2000-09-08 | 2004-05-20 | Gerhard Hamprecht | Method for producing anellated tetrahydro-{1h}-triazoles |
| HUP0401298A3 (en) | 2001-08-30 | 2008-03-28 | Alizyme Therapeutics Ltd | Thieno [1,3] oxazin-4-ones with lipase inhibiting activity, process for their preparation and pharmaceutical compositions containing them |
| WO2003087072A1 (en) * | 2002-03-29 | 2003-10-23 | Mochida Pharmaceutical Co., Ltd. | Therapeutic agent for endothelial disorder |
| BR0315932A (pt) | 2002-10-30 | 2005-09-13 | Basf Ag | Processo para a preparação de iso (tio) cianatos de fenila, composto, e, processo para a preparação do mesmo |
| KR102027598B1 (ko) | 2011-05-17 | 2019-10-01 | 프린시피아 바이오파마, 인코퍼레이티드 | 타이로신 키나아제 저해제 |
| US9580427B2 (en) | 2011-05-17 | 2017-02-28 | The Regents Of The University Of California | Kinase inhibitors |
| US9376438B2 (en) | 2011-05-17 | 2016-06-28 | Principia Biopharma, Inc. | Pyrazolopyrimidine derivatives as tyrosine kinase inhibitors |
| CN104822681B (zh) | 2012-09-10 | 2018-01-30 | 普林斯匹亚生物制药公司 | 作为激酶抑制剂的吡唑并嘧啶化合物 |
| US8957080B2 (en) | 2013-04-09 | 2015-02-17 | Principia Biopharma Inc. | Tyrosine kinase inhibitors |
| DE102013226249A1 (de) * | 2013-12-17 | 2015-06-18 | Wacker Chemie Ag | Polyetherreste aufweisende Organopolysiloxangele |
| EP3107544B1 (en) | 2014-02-21 | 2020-10-07 | Principia Biopharma Inc. | Salts and solid form of a btk inhibitor |
| CA2970723C (en) | 2014-12-18 | 2023-09-05 | Principia Biopharma Inc. | Treatment of pemphigus |
| EP3313839A1 (en) | 2015-06-24 | 2018-05-02 | Principia Biopharma Inc. | Tyrosine kinase inhibitors |
| IL293621B2 (en) | 2016-06-29 | 2023-09-01 | Principia Biopharma Inc | Modified release formulations of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[4,3-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4 -Methyl-4-[4-(oxane-3-yl)piperazine-1-yl)penta-2-ananitrile |
| EP3648605A1 (en) * | 2017-07-03 | 2020-05-13 | Bayer CropScience Aktiengesellschaft | Novel isothiazolo-based bicycles, processes for their preparation and their use as herbicides and/or plant growth regulators |
| CN109776302A (zh) * | 2017-11-13 | 2019-05-21 | 中国科学院化学研究所 | 一种由木质素为甲基源制备重要化学品的方法 |
| IL291994A (en) | 2019-10-14 | 2022-06-01 | Principia Biopharma Inc | Methods for treating immune thrombocytopenia by administering (r)-2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine- 1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile |
| CN115461341A (zh) | 2020-01-22 | 2022-12-09 | 普林斯匹亚生物制药公司 | 2-[3-[4-氨基-3-(2-氟-4-苯氧基-苯基)-1h-吡唑并[3,4-d]嘧啶-1-基]哌啶-1-羰基]-4-甲基-4-[4-(氧杂环丁烷-3-基)哌嗪-1-基]戊-2-烯腈的晶型 |
| CN114276287B (zh) * | 2021-12-27 | 2023-10-03 | 浙江工业大学 | N-(取代苄氧基)酰胺类化合物及其制备方法和应用 |
| CN116354953B (zh) * | 2022-12-31 | 2024-07-16 | 西北农林科技大学 | 含苯并噻唑类化合物的除草组合物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU627906B2 (en) * | 1989-07-14 | 1992-09-03 | Nissan Chemical Industries Ltd. | Uracil derivatives and herbicides containing the same as active ingredient |
| IL97102A0 (en) * | 1990-02-16 | 1992-03-29 | Ici Plc | Heterocyclic compounds |
| US5484763A (en) * | 1995-02-10 | 1996-01-16 | American Cyanamid Company | Substituted benzisoxazole and benzisothiazole herbicidal agents |
| US5753595A (en) * | 1995-08-31 | 1998-05-19 | Fmc Corporation | Herbicidal 3-(substituted benzoxazol-7-yl) and 3-(Substituted benzothiazol-7-yl)-1-substituted-6-trifluoromethyl-2 4-(1h 3h)pyrimidinediones |
| EP0853620A1 (en) * | 1995-10-04 | 1998-07-22 | Fmc Corporation | Herbicidal heterocyclic benzisoxazoles and benzisoxazolidinones |
-
1998
- 1998-08-27 IL IL12594798A patent/IL125947A0/xx unknown
- 1998-09-02 CA CA002246221A patent/CA2246221A1/en not_active Abandoned
- 1998-09-09 NZ NZ331825A patent/NZ331825A/xx unknown
- 1998-09-15 YU YU15800A patent/YU15800A/sh unknown
- 1998-09-15 PL PL98339350A patent/PL339350A1/xx unknown
- 1998-09-15 WO PCT/US1998/019251 patent/WO1999014216A1/en not_active Ceased
- 1998-09-15 CN CN98809898A patent/CN1273585A/zh active Pending
- 1998-09-15 CZ CZ2000861A patent/CZ2000861A3/cs unknown
- 1998-09-15 SK SK355-2000A patent/SK3552000A3/sk unknown
- 1998-09-15 JP JP2000511765A patent/JP2001516758A/ja active Pending
- 1998-09-15 TR TR2000/00679T patent/TR200000679T2/xx unknown
- 1998-09-15 AU AU93925/98A patent/AU9392598A/en not_active Abandoned
- 1998-09-15 ZA ZA9808435A patent/ZA988435B/xx unknown
- 1998-09-15 AU AU84239/98A patent/AU737864B2/en not_active Ceased
- 1998-09-15 BR BR9813017-0A patent/BR9813017A/pt not_active IP Right Cessation
- 1998-09-15 HU HU0004477A patent/HUP0004477A3/hu unknown
- 1998-09-16 ES ES98307495T patent/ES2185118T3/es not_active Expired - Lifetime
- 1998-09-16 AR ARP980104611A patent/AR015168A1/es unknown
- 1998-09-16 TW TW087115446A patent/TW474927B/zh not_active IP Right Cessation
- 1998-09-16 EP EP98307495A patent/EP0908457B1/en not_active Expired - Lifetime
- 1998-09-16 DE DE69809370T patent/DE69809370T2/de not_active Expired - Fee Related
- 1998-09-16 AT AT98307495T patent/ATE227721T1/de not_active IP Right Cessation
-
1999
- 1999-11-04 AR ARP990105577A patent/AR021500A2/es unknown
- 1999-11-04 AR ARP990105578A patent/AR021081A2/es unknown
-
2000
- 2000-03-16 KR KR20007002805A patent/KR20010030612A/ko not_active Withdrawn
- 2000-03-16 MX MXPA00002661 patent/MXPA00002661A/es unknown
- 2000-04-13 BG BG104336A patent/BG104336A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SK3552000A3 (en) | 2001-01-18 |
| HUP0004477A2 (hu) | 2001-02-28 |
| JP2001516758A (ja) | 2001-10-02 |
| ATE227721T1 (de) | 2002-11-15 |
| PL339350A1 (en) | 2000-12-18 |
| AU8423998A (en) | 1999-04-01 |
| IL125947A0 (en) | 1999-04-11 |
| TW474927B (en) | 2002-02-01 |
| TR200000679T2 (tr) | 2000-08-21 |
| BR9813017A (pt) | 2000-08-15 |
| KR20010030612A (en) | 2001-04-16 |
| NZ331825A (en) | 2000-04-28 |
| DE69809370T2 (de) | 2003-03-27 |
| EP0908457B1 (en) | 2002-11-13 |
| AR015168A1 (es) | 2001-04-18 |
| BG104336A (en) | 2001-09-28 |
| AR021081A2 (es) | 2002-06-12 |
| WO1999014216A1 (en) | 1999-03-25 |
| HUP0004477A3 (en) | 2002-01-28 |
| CA2246221A1 (en) | 1999-03-17 |
| DE69809370D1 (de) | 2002-12-19 |
| CN1273585A (zh) | 2000-11-15 |
| AU737864B2 (en) | 2001-08-30 |
| ZA988435B (en) | 2000-03-15 |
| CZ2000861A3 (cs) | 2000-08-16 |
| ES2185118T3 (es) | 2003-04-16 |
| EP0908457A1 (en) | 1999-04-14 |
| AU9392598A (en) | 1999-04-05 |
| MXPA00002661A (es) | 2001-10-31 |
| YU15800A (sh) | 2002-11-15 |
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