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AR027066A1 - Forma de dosificacion de farmaco en capas impulsada por hidrogel - Google Patents

Forma de dosificacion de farmaco en capas impulsada por hidrogel

Info

Publication number
AR027066A1
AR027066A1 ARP000106853A ARP000106853A AR027066A1 AR 027066 A1 AR027066 A1 AR 027066A1 AR P000106853 A ARP000106853 A AR P000106853A AR P000106853 A ARP000106853 A AR P000106853A AR 027066 A1 AR027066 A1 AR 027066A1
Authority
AR
Argentina
Prior art keywords
dosage form
hour
weight
environment
sertraline
Prior art date
Application number
ARP000106853A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AR027066A1 publication Critical patent/AR027066A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Obesity (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

Una forma de dosificacion de liberacion controlada para sertralina tiene un nucleo que comprende una composicion que contiene sertralina y una composicionhinchable en agua, en donde la composicion hinchable en agua está situada en una region separada dentro del nucleo. Un revestimiento en torno al nucleo espermeable al agua, insoluble en agua, y tiene al menos una abertura de suministro a través del mismo. En una realizacion, la forma de dosificacion liberasertralina hacia el entorno de uso con una velocidad media de 6 a 10% en peso por hora desde la segunda hasta la décima hora después de la introduccion en unentorno de uso, y menos de aproximadamente 25% en peso durante las dos primeras horas y al menos 70% en peso al cabo de la décima ho ra, en donde losporcentajes corresponden a la masa de fármaco liberado desde el comprimido dividida por la masa total de fármaco originalmente presente en el comprimido. Enotra realizacion, la forma de dosificacion libera menos de aproximadamente 25% en peso de sertralina hacia el entorno de uso al cabo de la segunda hora despuésde la introduccion de la forma de dosificacion en el entorno de uso, y suministra al menos 25% en peso desde la octava hora hasta la vigesimocuarta.
ARP000106853A 1999-12-23 2000-12-21 Forma de dosificacion de farmaco en capas impulsada por hidrogel AR027066A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17210899P 1999-12-23 1999-12-23

Publications (1)

Publication Number Publication Date
AR027066A1 true AR027066A1 (es) 2003-03-12

Family

ID=22626396

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000106853A AR027066A1 (es) 1999-12-23 2000-12-21 Forma de dosificacion de farmaco en capas impulsada por hidrogel

Country Status (15)

Country Link
US (1) US6899896B2 (es)
EP (1) EP1239839A2 (es)
JP (1) JP2003518487A (es)
AR (1) AR027066A1 (es)
AU (1) AU1724301A (es)
BR (1) BR0016707A (es)
CA (1) CA2395231C (es)
CO (1) CO5271728A1 (es)
GT (1) GT200000220A (es)
MX (1) MXPA02006335A (es)
PA (1) PA8508901A1 (es)
PE (1) PE20010983A1 (es)
TN (1) TNSN00251A1 (es)
UY (1) UY26493A1 (es)
WO (1) WO2001047498A2 (es)

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ATE395044T1 (de) 2002-02-01 2008-05-15 Pfizer Prod Inc Pharmazeutische zusammensetzungen amorpher dispersionen von wirkstoffen und lipophiler mikrophasenbildender materialien
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US8637512B2 (en) 2002-07-29 2014-01-28 Glaxo Group Limited Formulations and method of treatment
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US8084058B2 (en) 2002-09-20 2011-12-27 Watson Pharmaceuticals, Inc. Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
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CN100563637C (zh) * 2006-10-13 2009-12-02 北京红林制药有限公司 一种控释给药的药芯组合物和控释制剂及其制备方法
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WO2011078993A1 (en) 2009-12-21 2011-06-30 Aptapharma, Inc. Functionally-coated multilayer tablets
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Also Published As

Publication number Publication date
UY26493A1 (es) 2001-07-31
JP2003518487A (ja) 2003-06-10
EP1239839A2 (en) 2002-09-18
CA2395231C (en) 2006-08-15
CO5271728A1 (es) 2003-04-30
WO2001047498A2 (en) 2001-07-05
PE20010983A1 (es) 2001-10-01
AU1724301A (en) 2001-07-09
MXPA02006335A (es) 2002-12-13
PA8508901A1 (es) 2003-12-10
BR0016707A (pt) 2002-09-03
CA2395231A1 (en) 2001-07-05
TNSN00251A1 (fr) 2002-05-30
GT200000220A (es) 2002-06-14
US20010044474A1 (en) 2001-11-22
WO2001047498A3 (en) 2001-11-15
US6899896B2 (en) 2005-05-31

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