AR013559A1 - USO DE DERIVADOS DE PIRROLIDINA PARA LA PREPARACIoN DE MEDICAMENNTOS DESTINADOS AL TRATAMIENTO DEL ABUSO DE DROGAS O DE SUSTANCIAS QUE DAN ORIGEN A LA ADICCIoN O AL USO EXCESIVO DE DROGAS , CON EXCEPCIoN DEL ABUSO DEL ALCOHOL, MEDIANTE LA REDUCCIoN DE LA AUTO-MEDICACIoN DE DICHAS DROGAS POR PARTE DE - Google Patents
USO DE DERIVADOS DE PIRROLIDINA PARA LA PREPARACIoN DE MEDICAMENNTOS DESTINADOS AL TRATAMIENTO DEL ABUSO DE DROGAS O DE SUSTANCIAS QUE DAN ORIGEN A LA ADICCIoN O AL USO EXCESIVO DE DROGAS , CON EXCEPCIoN DEL ABUSO DEL ALCOHOL, MEDIANTE LA REDUCCIoN DE LA AUTO-MEDICACIoN DE DICHAS DROGAS POR PARTE DEInfo
- Publication number
- AR013559A1 AR013559A1 ARP970100466A ARP970100466A AR013559A1 AR 013559 A1 AR013559 A1 AR 013559A1 AR P970100466 A ARP970100466 A AR P970100466A AR P970100466 A ARP970100466 A AR P970100466A AR 013559 A1 AR013559 A1 AR 013559A1
- Authority
- AR
- Argentina
- Prior art keywords
- drugs
- abuse
- drug
- substances
- preparation
- Prior art date
Links
- 239000003814 drug Substances 0.000 title abstract 4
- 229940079593 drug Drugs 0.000 title abstract 4
- 206010013654 Drug abuse Diseases 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- 239000000126 substance Substances 0.000 title abstract 2
- 208000011117 substance-related disease Diseases 0.000 title abstract 2
- 238000011282 treatment Methods 0.000 title abstract 2
- 206010012335 Dependence Diseases 0.000 title 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 title 1
- RWRDLPDLKQPQOW-UHFFFAOYSA-N Pyrrolidine Chemical class C1CCNC1 RWRDLPDLKQPQOW-UHFFFAOYSA-N 0.000 title 1
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 208000007848 Alcoholism Diseases 0.000 abstract 1
- 206010001584 alcohol abuse Diseases 0.000 abstract 1
- 208000025746 alcohol use disease Diseases 0.000 abstract 1
- 150000003235 pyrrolidines Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/401—Proline; Derivatives thereof, e.g. captopril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Addiction (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Aplicacion de derivados de la pirrolidina de la formula general I sus rascémicos y enantiomeros cuando contienen uno o varios centros asimétricos ysus sales, en la preparacion de medicamentos destinados al tratamiento del abuso de drogaso de sustancias que dan origen a farmacomanías o a su consumoexcesivo, excepto el abuso del alcohol.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9601481A FR2744361B1 (fr) | 1996-02-07 | 1996-02-07 | Application de derives de pyrrolidine a la preparation de medicaments destines au traitement de l'abus de drogues ou de substances donnant lieu a des pharmacomanies ou a un usage excessif |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR013559A1 true AR013559A1 (es) | 2001-01-10 |
Family
ID=9488931
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP970100466A AR013559A1 (es) | 1996-02-07 | 1997-06-02 | USO DE DERIVADOS DE PIRROLIDINA PARA LA PREPARACIoN DE MEDICAMENNTOS DESTINADOS AL TRATAMIENTO DEL ABUSO DE DROGAS O DE SUSTANCIAS QUE DAN ORIGEN A LA ADICCIoN O AL USO EXCESIVO DE DROGAS , CON EXCEPCIoN DEL ABUSO DEL ALCOHOL, MEDIANTE LA REDUCCIoN DE LA AUTO-MEDICACIoN DE DICHAS DROGAS POR PARTE DE |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US6150387A (es) |
| EP (1) | EP0879054B1 (es) |
| JP (1) | JP2000504681A (es) |
| AR (1) | AR013559A1 (es) |
| AU (1) | AU1727297A (es) |
| DE (1) | DE69738320T2 (es) |
| DK (1) | DK0879054T3 (es) |
| ES (1) | ES2297850T3 (es) |
| FR (1) | FR2744361B1 (es) |
| PT (1) | PT879054E (es) |
| TW (1) | TW514528B (es) |
| WO (1) | WO1997028798A1 (es) |
| ZA (1) | ZA97872B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6512120B1 (en) | 2001-03-12 | 2003-01-28 | Ortho Mcneil Pharmaceutical, Inc. | Methods for the synthesis of densely functionalized pyrrolidine intermediates |
| US6697016B1 (en) * | 2002-09-30 | 2004-02-24 | Motorola, Inc. | Self adjustment of a frequency offset in a GPS receiver |
| US7405210B2 (en) * | 2003-05-21 | 2008-07-29 | Osi Pharmaceuticals, Inc. | Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phosphorylase |
| ATE483708T1 (de) | 2004-03-08 | 2010-10-15 | Prosidion Ltd | Pyrrolopyridin-2-carbonsäurehydrazide als inhibitoren von glykogenphosphorylase |
| ES2324173T3 (es) | 2004-12-02 | 2009-07-31 | Prosidion Limited | Amidas del acido pirrolopiridin-2-carboxilico. |
| US8247438B2 (en) | 2008-02-27 | 2012-08-21 | Neuropill, Inc. | Methods for treating schizophrenia |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| WO2020212951A1 (en) | 2019-04-17 | 2020-10-22 | Compass Pathfinder Limited | Methods for treating anxiety disorders, headache disorders, and eating disorders with psilocybin |
| CN115667217A (zh) | 2020-05-19 | 2023-01-31 | 赛本爱尔兰有限公司 | 氘化的色胺衍生物和使用方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2678938B1 (fr) * | 1991-07-10 | 1993-10-08 | Rhone Poulenc Rorer Sa | Derives de pyrrolidine, leur preparation et les medicaments les contenant. |
| EP0617621A4 (en) * | 1991-12-20 | 1995-04-05 | Merck Sharp & Dohme | CENTRAL CHOLECYSTOKININE ANTAGONISTS WITH PHARMACEUTICAL EFFECTIVENESS. |
| FR2700167B1 (fr) * | 1993-01-07 | 1995-02-03 | Rhone Poulenc Rorer Sa | Dérivés de pyrrolidine et thiazolidine, leur préparation et les médicaments les contenant. |
| FR2700168B1 (fr) * | 1993-01-07 | 1995-02-03 | Rhone Poulenc Rorer Sa | Dérivés de thiazolidine, leur préparation et les médicaments les contenant. |
| FR2700165B1 (fr) * | 1993-01-07 | 1995-02-17 | Rhone Poulenc Rorer Sa | Dérivés de pyrrolidine, leur préparation et les médicaments les contenant. |
| FR2734724B1 (fr) * | 1995-06-01 | 1997-07-04 | Rhone Poulenc Rorer Sa | Application de derives de pyrrolidine a la preparation de medicaments destines au traitement de l'alcoolisme |
-
1996
- 1996-02-07 FR FR9601481A patent/FR2744361B1/fr not_active Expired - Fee Related
-
1997
- 1997-01-31 TW TW086101166A patent/TW514528B/zh not_active IP Right Cessation
- 1997-02-03 DE DE69738320T patent/DE69738320T2/de not_active Expired - Lifetime
- 1997-02-03 PT PT97904476T patent/PT879054E/pt unknown
- 1997-02-03 DK DK97904476T patent/DK0879054T3/da active
- 1997-02-03 WO PCT/FR1997/000209 patent/WO1997028798A1/fr not_active Ceased
- 1997-02-03 ES ES97904476T patent/ES2297850T3/es not_active Expired - Lifetime
- 1997-02-03 US US09/117,931 patent/US6150387A/en not_active Expired - Fee Related
- 1997-02-03 JP JP9528214A patent/JP2000504681A/ja not_active Ceased
- 1997-02-03 EP EP97904476A patent/EP0879054B1/fr not_active Expired - Lifetime
- 1997-02-03 ZA ZA9700872A patent/ZA97872B/xx unknown
- 1997-02-03 AU AU17272/97A patent/AU1727297A/en not_active Abandoned
- 1997-06-02 AR ARP970100466A patent/AR013559A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO1997028798A1 (fr) | 1997-08-14 |
| US6150387A (en) | 2000-11-21 |
| DE69738320T2 (de) | 2008-10-09 |
| TW514528B (en) | 2002-12-21 |
| ES2297850T3 (es) | 2008-05-01 |
| DE69738320D1 (de) | 2008-01-10 |
| FR2744361A1 (fr) | 1997-08-08 |
| EP0879054A1 (fr) | 1998-11-25 |
| EP0879054B1 (fr) | 2007-11-28 |
| FR2744361B1 (fr) | 1998-02-27 |
| ZA97872B (en) | 1997-08-04 |
| PT879054E (pt) | 2008-03-05 |
| AU1727297A (en) | 1997-08-28 |
| DK0879054T3 (da) | 2008-04-07 |
| JP2000504681A (ja) | 2000-04-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Refusal |