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AR012247A1 - Composiciones farmaceuticas y su uso para la preparacion de medicamentos destinados a prevenir y tratar las enfermedades tromboembolicas arteriales - Google Patents

Composiciones farmaceuticas y su uso para la preparacion de medicamentos destinados a prevenir y tratar las enfermedades tromboembolicas arteriales

Info

Publication number
AR012247A1
AR012247A1 ARP980102794A ARP980102794A AR012247A1 AR 012247 A1 AR012247 A1 AR 012247A1 AR P980102794 A ARP980102794 A AR P980102794A AR P980102794 A ARP980102794 A AR P980102794A AR 012247 A1 AR012247 A1 AR 012247A1
Authority
AR
Argentina
Prior art keywords
preparation
prevent
thromboembolic diseases
pharmaceutical compositions
treat arterial
Prior art date
Application number
ARP980102794A
Other languages
English (en)
Original Assignee
Dupuis Laurent
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dupuis Laurent filed Critical Dupuis Laurent
Publication of AR012247A1 publication Critical patent/AR012247A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7024Esters of saccharides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/702Oligosaccharides, i.e. having three to five saccharide radicals attached to each other by glycosidic linkages
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Utilizacion de uno o varios inhibidores selectivos directos o indirectos del factor Sa que actuan vía la antitrombina III, solos o en combinacion conuno o varios compuestos de actividad antagregante plaquetaria, para la preparacion de medicamentos distinados a prevenir y a tratar las enfermedadestromboembolicas arteriales. Composiciones farmacéuticas para la preparacion de medicamentos destinados a prevenir y tratar enfermedades tromboembolicasarteriales, composiciones que contienenuno o varios inhibidores selectivos directos o indirectos del factor Xa que actua vía la antitrombina III enasociacion con uno o varios compuestos de actividad antiagregante plaquetaria y eventualente uno o varios vehículos farmacéuticamente aceptables.
ARP980102794A 1997-06-13 1998-06-12 Composiciones farmaceuticas y su uso para la preparacion de medicamentos destinados a prevenir y tratar las enfermedades tromboembolicas arteriales AR012247A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9707368A FR2764511B1 (fr) 1997-06-13 1997-06-13 Compositions pour le traitement et la prevention de la thrombose arterielle et utilisation d'un inhibiteur du facteur xa seul et/ou en combinaison avec un antiagregant plaquettaire

Publications (1)

Publication Number Publication Date
AR012247A1 true AR012247A1 (es) 2000-09-27

Family

ID=9507960

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980102794A AR012247A1 (es) 1997-06-13 1998-06-12 Composiciones farmaceuticas y su uso para la preparacion de medicamentos destinados a prevenir y tratar las enfermedades tromboembolicas arteriales

Country Status (42)

Country Link
US (2) US6541488B1 (es)
EP (1) EP0986376B1 (es)
JP (1) JP3988803B2 (es)
KR (1) KR100598451B1 (es)
CN (1) CN1253150C (es)
AR (1) AR012247A1 (es)
AT (1) ATE384528T1 (es)
AU (1) AU728826B2 (es)
BR (1) BR9810520A (es)
CA (1) CA2293415C (es)
CO (1) CO4940476A1 (es)
CY (1) CY1107912T1 (es)
CZ (1) CZ299518B6 (es)
DE (1) DE69839046T2 (es)
DK (1) DK0986376T3 (es)
DZ (1) DZ2512A1 (es)
EE (1) EE04737B1 (es)
ES (1) ES2299209T3 (es)
FR (1) FR2764511B1 (es)
GT (1) GT199800171A (es)
HR (1) HRP980322B1 (es)
HU (1) HU227956B1 (es)
ID (1) ID29309A (es)
IL (1) IL133452A (es)
IS (1) IS2619B (es)
ME (1) ME00685B (es)
MY (1) MY124648A (es)
NO (1) NO323739B1 (es)
NZ (1) NZ501452A (es)
PL (1) PL193405B1 (es)
PT (1) PT986376E (es)
RS (1) RS49902B (es)
RU (1) RU2212886C2 (es)
SA (1) SA98190552B1 (es)
SI (1) SI0986376T1 (es)
SK (1) SK286311B6 (es)
TR (1) TR199903087T2 (es)
TW (1) TW565442B (es)
UA (1) UA70919C2 (es)
UY (1) UY25044A1 (es)
WO (1) WO1998056365A1 (es)
ZA (1) ZA985137B (es)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2764511B1 (fr) * 1997-06-13 2000-09-08 Sanofi Sa Compositions pour le traitement et la prevention de la thrombose arterielle et utilisation d'un inhibiteur du facteur xa seul et/ou en combinaison avec un antiagregant plaquettaire
EP1156803A4 (en) 1999-02-09 2004-03-17 Bristol Myers Squibb Co FXA LACTAM INHIBITORS AND METHOD
US6344450B1 (en) 1999-02-09 2002-02-05 Bristol-Myers Squibb Company Lactam compounds and their use as inhibitors of serine proteases and method
FR2793687B1 (fr) * 1999-04-26 2001-08-24 Sanofi Sa Nouvelle composition injectable d'un anticoagulant
FR2800074B1 (fr) * 1999-10-22 2001-12-21 Aventis Pharma Sa Nouveaux oligosaccharides, leur preparation et les compositions pharmaceutiques les contenant
US6544981B2 (en) 2000-06-09 2003-04-08 Bristol-Myers Squibb Company Lactam inhibitors of factor Xa and method
US6511973B2 (en) 2000-08-02 2003-01-28 Bristol-Myers Squibb Co. Lactam inhibitors of FXa and method
ATE352309T1 (de) * 2001-02-28 2007-02-15 John H Griffin Plasmaglucosylceramiddefizienz als risikofaktor für thrombose und modulator von anticoagulant protein c
UA80399C2 (en) * 2001-11-13 2007-09-25 Glaxo Group Ltd Use of specific dose of fondaparinux sodium for the treatment of acs
AU2003270861A1 (en) 2002-10-02 2004-04-23 Bristol-Myers Squibb Company Novel combination of a factor xa inhibitor and clopidogrel
CA2507026A1 (en) * 2002-11-22 2004-06-10 Takeda Pharmaceutical Company Limited Imidazole derivatives, their production and use
RU2245162C2 (ru) * 2003-01-04 2005-01-27 Козлов Владимир Александрович Способ терапии инфаркта миокарда
WO2005027896A1 (ja) * 2003-09-19 2005-03-31 Kissei Pharmaceutical Co., Ltd. 併用医薬
WO2005087266A1 (en) * 2004-03-05 2005-09-22 Vddi Pharmaceuticals Combination therapy for inhibition of platelet aggregation
KR101099884B1 (ko) * 2004-04-23 2011-12-28 히또시 기야 동화상데이터의 부호화방법, 복호화방법, 이들을 실행하는단말장치, 및 쌍방향 대화형 시스템
TWI396686B (zh) 2004-05-21 2013-05-21 Takeda Pharmaceutical 環狀醯胺衍生物、以及其製品和用法
US7563780B1 (en) * 2004-06-18 2009-07-21 Advanced Cardiovascular Systems, Inc. Heparin prodrugs and drug delivery stents formed therefrom
JP5557410B2 (ja) * 2004-07-13 2014-07-23 第一三共株式会社 経口投与による血栓・塞栓の予防治療剤
US20070105825A1 (en) * 2004-09-16 2007-05-10 Yuji Hoyano Concurrent drugs
US20090111769A1 (en) * 2005-10-10 2009-04-30 De Kort Martin Antithrombotic Compound
CA2735983A1 (en) * 2008-09-10 2010-03-18 Transpharma Medical Ltd. Transdermal delivery of oligosaccharides
RU2410104C1 (ru) * 2009-07-10 2011-01-27 Учреждение Российской академии медицинских наук Научный центр неврологии РАМН СПОСОБ СНИЖЕНИЯ АГРЕГАЦИОННОЙ АКТИВНОСТИ ТРОМБОЦИТОВ in vitro
WO2011149110A1 (en) 2010-05-28 2011-12-01 Daiichi Sankyo Company, Limited Novel composition for the prevention and/or treatment of thromboembolism
KR101968190B1 (ko) * 2014-10-30 2019-04-11 청두 바이위 파머수티컬 씨오., 엘티디 징코라이드 B(Ginkgolide B)와 Ⅹa 인자 억제제를 포함한 약물 조성물 및 그 제조방법과 용도
CN106860868B (zh) * 2015-12-11 2019-11-22 北京百奥药业有限责任公司 沙班类药物与蚓激酶的药物组合物、制剂及其应用
US11654036B2 (en) 2020-05-26 2023-05-23 Elixir Medical Corporation Anticoagulant compounds and methods and devices for their use

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE419871B (sv) * 1975-12-01 1981-08-31 Pharmacia Ab Sett att bestemma aktiviteten hos faktor xa-inhibitor i blod
DE3038163A1 (de) * 1980-10-09 1982-05-06 Boehringer Mannheim Gmbh, 6800 Mannheim Thrombininhibitor, seine herstellung und verwendung
FR2548189B1 (fr) * 1983-07-01 1986-04-11 Choay Sa Nouveaux produits contenant des oligosaccharides, leur preparation et leurs applications biologiques et biochimiques
RU2045264C1 (ru) * 1983-12-15 1995-10-10 Белорусский научно-исследовательский институт кардиологии Антиагрегационное средство
ZA928276B (en) * 1991-10-31 1993-05-06 Daiichi Seiyaku Co Aromatic amidine derivates and salts thereof.
FR2728901B1 (fr) * 1994-12-28 1997-03-28 Sanofi Sa Derives de phenyl-4-thiazoles substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
SI0946185T2 (sl) 1996-11-27 2010-08-31 Aventis Pharma Inc Farmacevtski sestavek, ki obsega spojino z anti-Xa-aktivnostjo in antagonistično spojino za agregacijo ploščic
FR2764511B1 (fr) * 1997-06-13 2000-09-08 Sanofi Sa Compositions pour le traitement et la prevention de la thrombose arterielle et utilisation d'un inhibiteur du facteur xa seul et/ou en combinaison avec un antiagregant plaquettaire

Also Published As

Publication number Publication date
PL337288A1 (en) 2000-08-14
EE9900574A (et) 2000-08-15
SI0986376T1 (sl) 2008-06-30
CN1274281A (zh) 2000-11-22
HRP980322A2 (en) 1999-04-30
SK286311B6 (en) 2008-07-07
TW565442B (en) 2003-12-11
ES2299209T3 (es) 2008-05-16
SA98190552B1 (ar) 2006-09-09
DE69839046T2 (de) 2009-01-15
ID29309A (id) 2001-08-16
YU63699A (sh) 2002-06-19
JP3988803B2 (ja) 2007-10-10
HUP0002175A3 (en) 2003-05-28
PL193405B1 (pl) 2007-02-28
ME00685B (me) 2008-08-07
BR9810520A (pt) 2000-09-19
UA70919C2 (uk) 2004-11-15
NO323739B1 (no) 2007-07-02
ATE384528T1 (de) 2008-02-15
IL133452A0 (en) 2001-04-30
MY124648A (en) 2006-06-30
UY25044A1 (es) 2000-10-31
AU7924698A (en) 1998-12-30
EP0986376A1 (fr) 2000-03-22
CN1253150C (zh) 2006-04-26
CA2293415A1 (en) 1998-12-17
CZ299518B6 (cs) 2008-08-20
CO4940476A1 (es) 2000-07-24
KR100598451B1 (ko) 2006-07-10
KR20010013690A (ko) 2001-02-26
EP0986376B1 (fr) 2008-01-23
ZA985137B (en) 1999-01-07
PT986376E (pt) 2008-04-01
HUP0002175A1 (hu) 2000-11-28
JP2002504110A (ja) 2002-02-05
RS49902B (sr) 2008-08-07
CZ446099A3 (cs) 2000-04-12
HU227956B1 (en) 2012-07-30
NO996137D0 (no) 1999-12-10
IS2619B (is) 2010-05-15
WO1998056365A1 (fr) 1998-12-17
HK1032750A1 (en) 2001-08-03
DE69839046D1 (de) 2008-03-13
US20040092477A1 (en) 2004-05-13
FR2764511A1 (fr) 1998-12-18
EE04737B1 (et) 2006-12-15
FR2764511B1 (fr) 2000-09-08
IS5280A (is) 1999-11-30
RU2212886C2 (ru) 2003-09-27
US6541488B1 (en) 2003-04-01
SK170999A3 (en) 2000-07-11
DZ2512A1 (fr) 2003-02-01
GT199800171A (es) 2000-04-21
IL133452A (en) 2004-09-27
CY1107912T1 (el) 2013-09-04
HRP980322B1 (en) 2003-12-31
NO996137L (no) 2000-02-14
CA2293415C (en) 2011-08-09
DK0986376T3 (da) 2008-05-13
AU728826B2 (en) 2001-01-18
TR199903087T2 (xx) 2000-05-22
NZ501452A (en) 2002-06-28

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