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AR014406A1 - SULFONYL PHENYLAMINES REPLACED AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM - Google Patents

SULFONYL PHENYLAMINES REPLACED AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM

Info

Publication number
AR014406A1
AR014406A1 ARP980106523A ARP980106523A AR014406A1 AR 014406 A1 AR014406 A1 AR 014406A1 AR P980106523 A ARP980106523 A AR P980106523A AR P980106523 A ARP980106523 A AR P980106523A AR 014406 A1 AR014406 A1 AR 014406A1
Authority
AR
Argentina
Prior art keywords
alkyl
alkoxy
substituted
carbamoyl
amino
Prior art date
Application number
ARP980106523A
Other languages
Spanish (es)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR014406A1 publication Critical patent/AR014406A1/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88Nitrogen atoms, e.g. allantoin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/14Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/42Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Sulfonilfenilaminas sustituidas de la formula (I), en donde: X es S o NH, e Y y Z son cada uno CH; o X es NH, y una de las variables Y y Z es N, y la otraes CH; R1 y R2, independientemente uno del otro, presentan hidrogeno, alquilo (C1-7), o alquilo (C1-7) sustituido por hidroxi, halogeno, alcoxi (C1-7),carboxi, alcoxi (C1-7)-carbonilo, carbamoílo, alquilo (C1-7)-carbamoílo, dialquilo (C1-7)-carbamoílo, cicloalquilo (C3-8), o por cicloalquilo (C3-8) queestá sustituido por alcoxi (C1-7)-carbonilo, o representan alcanoílo (C2-7); mientras que cuando menos una de las variables R1 y R2 es diferente dehidrogeno; o el grupo NR1R2 es alquileno (C2-6)-amino lineal que está insustituido o sustituido por alquilo (C1-7), hidroxialquilo (C1-7), alcoxi(C1-7), alcoxi (C1-7)-alquilo (C1-7), alcoxi (C1-7)-alcoxi (C1-7)-alquilo (C1-7), tioalquilo (C1-7)-alquilo (C1-7), alcano (C1-7)-sulfinilalquilo (C1-7),alcano (C1-7)-sulfonilalquilo (C1-7), aminoalquilo (C1-7), alquilo (C1-7)- aminoalquilo (C1-7), dialquilo (C1-7)-aminoalquilo (C1-7), hidroxi, ciano,amino, alquilo (C1-7)-amino, dialquilo (C1-7)-amino, alcanoílo (C1-7), hidroxilimino-alquilo (C2-7), carboxi, alcoxi (C1-7)-carbonilo, carbamoílo,alquilo (C1-7)-carbamoílo, dialquilo (C1-7)-carbamoílo, o por oxo, o es morfolino, tiomorfolino, 4-alquilo (C1-7)-piperazino, 4-piridil-piperazino,tetrahidroquinolin-1-ilo, tetrahidroiso-quinolin-2-ilo, dihidroindol-1-ilo, o dihidroindol-1-ilo sustituido por alcoxi (C1-7)-carbonilo, o es un grupo de laformula (II); y en donde el anillo A, aparte de estar sustituido por -SO2NR1R2 y -NH-, está insustituido o sustituido una o más veces por un sustituyenteseleccionado a partir del grupo que consisteen alquilo (C1-7), alcoxi (C1-7), alcoxi (C1-7)-alcoxi (C1-7), hidroxi, halogeno, y CF3; y en donde el anillo BSubstituted sulfonylphenylamines of the formula (I), wherein: X is S or NH, and Y and Z are each CH; or X is NH, and one of the variables Y and Z is N, and the other is CH; R1 and R2, independently of each other, have hydrogen, (C1-7) alkyl, or (C1-7) alkyl substituted by hydroxy, halogen, (C1-7) alkoxy, carboxy, (C1-7) alkoxycarbonyl, carbamoyl, (C1-7) alkyl -carbamoyl, dialkyl (C1-7) -carbamoyl, cycloalkyl (C3-8), or by cycloalkyl (C3-8) which is substituted by (C1-7) alkoxycarbonyl, or represent alkanoyl (C2-7); while at least one of the variables R1 and R2 is different from hydrogen; or the NR1R2 group is linear (C2-6) alkyleneamino which is unsubstituted or substituted by (C1-7) alkyl, hydroxy (C1-7) alkyl, (C1-7) alkoxy, (C1-7) alkoxy ( C1-7), (C1-7) alkoxy-(C1-7) alkoxy-(C1-7) alkyl, thioalkyl (C1-7) -alkyl (C1-7), alkane (C1-7) -sulfinylalkyl (C1 -7), (C1-7) alkane-sulfonyl (C1-7) alkyl, amino (C1-7) alkyl, (C1-7) alkyl-amino (C1-7), dialkyl (C1-7) -aminoalkyl (C1- 7), hydroxy, cyano, amino, (C1-7) -amino, dialkyl (C1-7) -amino, (C1-7) alkanoyl, hydroxyimino-(C2-7) alkyl, carboxy, (C1-7) alkoxy ) -carbonyl, carbamoyl, (C1-7) alkyl -carbamoyl, dialkyl (C1-7) -carbamoyl, or by oxo, or is morpholino, thiomorpholino, 4-alkyl (C1-7) -piperazino, 4-pyridyl-piperazino , tetrahydroquinolin-1-yl, tetrahydroiso-quinolin-2-yl, dihydroindole-1-yl, or dihydroindole-1-yl substituted by (C1-7) alkoxycarbonyl, or is a group of laformula (II); and wherein ring A, apart from being substituted by -SO2NR1R2 and -NH-, is unsubstituted or substituted one or more times by a substituent selected from the group consisting of (C1-7) alkyl, (C1-7) alkoxy, (C1-7) alkoxy (C1-7) alkoxy, hydroxy, halogen, and CF3; and where ring B

ARP980106523A 1997-12-22 1998-12-18 SULFONYL PHENYLAMINES REPLACED AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM AR014406A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19757248 1997-12-22

Publications (1)

Publication Number Publication Date
AR014406A1 true AR014406A1 (en) 2001-02-28

Family

ID=7853006

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980106523A AR014406A1 (en) 1997-12-22 1998-12-18 SULFONYL PHENYLAMINES REPLACED AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM

Country Status (6)

Country Link
AR (1) AR014406A1 (en)
AU (1) AU2415299A (en)
CO (1) CO5011105A1 (en)
PE (1) PE20000127A1 (en)
WO (1) WO1999032466A1 (en)
ZA (1) ZA9811705B (en)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2350714A1 (en) 1998-11-10 2000-05-18 Merck & Co., Inc. Spiro-indolines as y5 receptor antagonists
FR2792314B1 (en) * 1999-04-15 2001-06-01 Adir NOVEL AMINOTRIAZOLE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
US6218408B1 (en) 1999-06-30 2001-04-17 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (bicyclics)
US6340683B1 (en) 1999-04-22 2002-01-22 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (triazines)
US6989379B1 (en) 1999-04-22 2006-01-24 H. Lundbick A/S Selective NPY (Y5) antagonists
EP1183245B1 (en) * 1999-04-22 2007-05-09 H. Lundbeck A/S Selective npy (y5) antagonists
US6225330B1 (en) 1999-06-30 2001-05-01 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (tricyclics)
US6214853B1 (en) 1999-06-30 2001-04-10 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (bicyclics)
US6222040B1 (en) 1999-06-30 2001-04-24 Synaptic Pharmaceutical Corporation Selective NPY (Y5) antagonists (tricyclics)
US7273880B2 (en) 1999-06-30 2007-09-25 H. Lunbeck A/S Selective NPY (Y5) antagonists
DK1249233T3 (en) * 1999-11-26 2008-11-17 Shionogi & Co NPYY5 receptor antagonists
JP2003525291A (en) * 2000-03-01 2003-08-26 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 2,4-disubstituted thiazolyl derivatives
FR2815346B1 (en) * 2000-10-13 2004-02-20 Servier Lab NOVEL AMINOTRIAZOLONE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
WO2002078697A1 (en) * 2001-03-29 2002-10-10 Smithkline Beecham Corporation Compounds and methods
CA2403307A1 (en) 2001-10-23 2003-04-23 Neurogen Corporation Substituted 2-cyclohexyl-4-phenyl-1h-imidazole derivatives
TW200303742A (en) * 2001-11-21 2003-09-16 Novartis Ag Organic compounds
BRPI0409447A (en) * 2003-04-14 2006-04-18 Inst For Pharm Discovery Inc substituted phenylalkanoic acids
EA200501710A1 (en) 2003-04-30 2006-06-30 ДЗЕ ИНСТИТЬЮТС ФОР ФАРМАСЬЮТИКАЛ ДИСКАВЕРИ, ЭлЭлСи SUBSTITUTED CARBON ACIDS
WO2006042215A1 (en) 2004-10-08 2006-04-20 Janssen Pharmaceutica, N.V. 1,2,4-triazolylaminoaryl (heteroaryl) sulfonamide derivatives
GB0526257D0 (en) 2005-12-22 2006-02-01 Novartis Ag Organic compounds
US9353078B2 (en) * 2013-10-01 2016-05-31 New York University Amino, amido and heterocyclic compounds as modulators of rage activity and uses thereof
EP4077290A1 (en) 2019-12-20 2022-10-26 Ikena Oncology, Inc. 4-phenyl-n-(phenyl)thiazol-2-amine derivatives and related compounds as aryl hydrocarbon receptor (ahr) agonists for the treatment of e.g. angiogenesis implicated or inflammatory disorders
WO2025017207A1 (en) * 2023-07-20 2025-01-23 Cemm - Forschungszentrum Für Molekulare Medizin Gmbh Inhibitors of smndc1 and their therapeutic use

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US3776765A (en) * 1972-02-28 1973-12-04 Cities Service Co Process for protecting a substrate with an n{11 substituted aminoarylsulfonamide intumescent agent
FR2701480B1 (en) * 1993-02-15 1995-05-24 Sanofi Elf Compounds with a sulfamoyl and amidino group, process for their preparation and pharmaceutical compositions containing them.
AU3201095A (en) * 1994-07-27 1996-02-22 G.D. Searle & Co. Substituted thiazoles for the treatment of inflammation

Also Published As

Publication number Publication date
ZA9811705B (en) 1999-09-07
AU2415299A (en) 1999-07-12
PE20000127A1 (en) 2000-03-14
CO5011105A1 (en) 2001-02-28
WO1999032466A1 (en) 1999-07-01

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