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AP2593A - Crystalline pyridazine compound - Google Patents

Crystalline pyridazine compound

Info

Publication number
AP2593A
AP2593A AP2009005078A AP2009005078A AP2593A AP 2593 A AP2593 A AP 2593A AP 2009005078 A AP2009005078 A AP 2009005078A AP 2009005078 A AP2009005078 A AP 2009005078A AP 2593 A AP2593 A AP 2593A
Authority
AP
ARIPO
Prior art keywords
crystalline
pyridazine compound
pyridazine
compound
crystalline pyridazine
Prior art date
Application number
AP2009005078A
Other languages
English (en)
Other versions
AP2009005078A0 (en
Inventor
Eric D Dowdy
Kenneth M Kent
Norma J Tom
Original Assignee
Gilead Sciences Inc
Ku Leuven Res And Dev
Puerstinger Gerhard
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39790369&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2593(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc, Ku Leuven Res And Dev, Puerstinger Gerhard filed Critical Gilead Sciences Inc
Publication of AP2009005078A0 publication Critical patent/AP2009005078A0/en
Application granted granted Critical
Publication of AP2593A publication Critical patent/AP2593A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
AP2009005078A 2007-07-06 2008-07-03 Crystalline pyridazine compound AP2593A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US95859507P 2007-07-06 2007-07-06
PCT/US2008/008259 WO2009009001A1 (fr) 2007-07-06 2008-07-03 Composé cristallin de pyridazine

Publications (2)

Publication Number Publication Date
AP2009005078A0 AP2009005078A0 (en) 2009-12-31
AP2593A true AP2593A (en) 2013-02-07

Family

ID=39790369

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2009005078A AP2593A (en) 2007-07-06 2008-07-03 Crystalline pyridazine compound

Country Status (19)

Country Link
US (2) US8106054B2 (fr)
EP (1) EP2170881A1 (fr)
JP (2) JP5366944B2 (fr)
KR (1) KR101229528B1 (fr)
CN (1) CN101778847B (fr)
AP (1) AP2593A (fr)
AR (1) AR066158A1 (fr)
AU (1) AU2008275756B2 (fr)
BR (1) BRPI0814801A2 (fr)
CA (1) CA2691917C (fr)
CO (1) CO6251293A2 (fr)
EA (2) EA201270275A1 (fr)
EC (1) ECSP109919A (fr)
IL (1) IL202694A0 (fr)
MX (1) MX2009013833A (fr)
TW (1) TWI447116B (fr)
UA (1) UA99466C2 (fr)
WO (1) WO2009009001A1 (fr)
ZA (1) ZA201000826B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0215293D0 (en) 2002-07-03 2002-08-14 Rega Foundation Viral inhibitors
EP2161273B1 (fr) 2003-12-22 2015-04-15 K.U.Leuven Research & Development Composés d'Imidazo[4,5-c]pyridine et procédés de traitement anti-viral
ATE426601T1 (de) 2004-12-21 2009-04-15 Gilead Sciences Inc Imidazoa4,5-cupyridinverbindung und verfahren zur antiviralen behandlung
TWI360549B (en) 2006-07-07 2012-03-21 Gilead Sciences Inc Novel pyridazine compound and use thereof
SI2094702T1 (sl) 2006-12-14 2016-03-31 Gilead Sciences, Inc. Virusni inhibitorji
UA99466C2 (en) 2007-07-06 2012-08-27 Гилиад Сайенсиз, Инк. Crystalline pyridazine compound
BR112012014729A2 (pt) 2009-12-18 2016-03-29 Boehringer Ingelheim Int terapia combinada contra hcv
EP2571882A1 (fr) 2010-05-21 2013-03-27 Gilead Sciences, Inc. Inhibiteurs heterocycliques de virus de la famille flaviviridae
TW201306841A (zh) 2010-12-20 2013-02-16 Gilead Sciences Inc 治療c型肝炎病毒(hcv)之方法
US20120204871A1 (en) * 2011-02-10 2012-08-16 Julio Cesar Vega Stable, non-corrosive formulations for pressurized metered dose inhalers
SG11201400664WA (en) 2011-09-16 2014-04-28 Gilead Pharmassett Llc Methods for treating hcv
US20140212491A1 (en) 2013-01-31 2014-07-31 Gilead Pharmasset Llc Combination formulation of two antiviral compounds
US20190022116A1 (en) 2014-12-26 2019-01-24 Emory University N4-Hydroxycytidine and Derivatives and Anti-Viral Uses Related Thereto
DK3706762T3 (da) 2017-12-07 2024-12-16 Univ Emory N4-hydroxycytidin og derivater og antivirale anvendelser relateret dertil
CN114195812A (zh) * 2021-12-30 2022-03-18 大连联化化学有限公司 一种合成2,4-二三氟甲基苯硼酸的方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005063744A2 (fr) * 2003-12-22 2005-07-14 K.U. Leuven Research & Development Composes d'imidazo[4,5-c]pyridine et methodes de traitement antiviral
WO2008005519A2 (fr) * 2006-07-07 2008-01-10 Gilead Sciences, Inc. Nouveau composé à base de pyrizadine et son utilisation

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Patent Citations (2)

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Publication number Priority date Publication date Assignee Title
WO2005063744A2 (fr) * 2003-12-22 2005-07-14 K.U. Leuven Research & Development Composes d'imidazo[4,5-c]pyridine et methodes de traitement antiviral
WO2008005519A2 (fr) * 2006-07-07 2008-01-10 Gilead Sciences, Inc. Nouveau composé à base de pyrizadine et son utilisation

Also Published As

Publication number Publication date
JP5366944B2 (ja) 2013-12-11
US20120108601A1 (en) 2012-05-03
ZA201000826B (en) 2010-11-24
AU2008275756A1 (en) 2009-01-15
BRPI0814801A2 (pt) 2017-03-28
EA018173B1 (ru) 2013-06-28
KR20100044201A (ko) 2010-04-29
JP2013216695A (ja) 2013-10-24
CA2691917C (fr) 2013-12-03
KR101229528B1 (ko) 2013-02-04
AU2008275756B2 (en) 2012-01-19
TWI447116B (zh) 2014-08-01
EA201270275A1 (ru) 2012-09-28
AP2009005078A0 (en) 2009-12-31
CN101778847A (zh) 2010-07-14
AR066158A1 (es) 2009-07-29
MX2009013833A (es) 2010-03-10
UA99466C2 (en) 2012-08-27
EA200971080A1 (ru) 2010-08-30
US8569488B2 (en) 2013-10-29
US8106054B2 (en) 2012-01-31
US20090036460A1 (en) 2009-02-05
IL202694A0 (en) 2010-06-30
ECSP109919A (es) 2010-04-30
WO2009009001A1 (fr) 2009-01-15
TW200918531A (en) 2009-05-01
EP2170881A1 (fr) 2010-04-07
JP2010532757A (ja) 2010-10-14
CA2691917A1 (fr) 2009-01-15
CN101778847B (zh) 2013-07-24
WO2009009001A9 (fr) 2010-11-11
CO6251293A2 (es) 2011-02-21

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