NO974057L - Bisykliske takykinin-antagonister, fremstilling derav og deres anvendelse i farmasöytisk sammensetning - Google Patents

Bisykliske takykinin-antagonister, fremstilling derav og deres anvendelse i farmasöytisk sammensetning

Info

Publication number: NO974057L
Authority: NO; Norway
Prior art keywords: bisyclic; preparation; pharmaceutical composition; tachykinin antagonists; tachykinin
Prior art date: 1995-03-13

Application number

NO974057A

Other languages

English (en)

Other versions

NO319290B1 (no

NO974057D0 (no

Inventor

Federico Arcamone

Carlo Alberto Maggi

Laura Quartara

Danilo Giannotti

Original Assignee

Menarini Farma Ind

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-03-13

Filing date

1997-09-03

Publication date

1997-11-07

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11351134&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO974057(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1997-09-03 Application filed by Menarini Farma Ind filed Critical Menarini Farma Ind

1997-09-03 Publication of NO974057D0 publication Critical patent/NO974057D0/no

1997-11-07 Publication of NO974057L publication Critical patent/NO974057L/no

2005-07-11 Publication of NO319290B1 publication Critical patent/NO319290B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/22—Tachykinins, e.g. Eledoisins, Substance P; Related peptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/64—Cyclic peptides containing only normal peptide links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Cardiology (AREA)
Biomedical Technology (AREA)
Oncology (AREA)
Pulmonology (AREA)
Communicable Diseases (AREA)
Rheumatology (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Virology (AREA)
Physical Education & Sports Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

NO19974057A 1995-03-13 1997-09-03 Bisykliske forbindelser, farmasoytiske sammensetninger som inneholder disse og anvendelse av forbindelsen til fremstillingen av et legemiddel. NO319290B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT95FI000044A IT1277835B1 (it)	1995-03-13	1995-03-13	Composti biciclici, loro preparazione ed uso in composizioni farmaceutiche
PCT/EP1996/001028 WO1996028467A1 (en)	1995-03-13	1996-03-11	Bicyclic tachykinins antagonists, preparation thereof and their use in pharmaceutical composition

Publications (3)

Publication Number	Publication Date
NO974057D0 NO974057D0 (no)	1997-09-03
NO974057L true NO974057L (no)	1997-11-07
NO319290B1 NO319290B1 (no)	2005-07-11

Family

ID=11351134

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO19974057A NO319290B1 (no)	1995-03-13	1997-09-03	Bisykliske forbindelser, farmasoytiske sammensetninger som inneholder disse og anvendelse av forbindelsen til fremstillingen av et legemiddel.

Country Status (33)

Country	Link
US (1)	US6150325A (no)
EP (1)	EP0815126B1 (no)
JP (1)	JP4618821B2 (no)
KR (1)	KR100405009B1 (no)
CN (1)	CN1189477C (no)
AR (1)	AR004476A1 (no)
AT (1)	ATE198481T1 (no)
AU (1)	AU696528B2 (no)
BG (1)	BG63208B1 (no)
BR (1)	BR9607348A (no)
CZ (1)	CZ287372B6 (no)
DE (1)	DE69611438T2 (no)
DK (1)	DK0815126T3 (no)
EA (1)	EA000697B1 (no)
EE (1)	EE03618B1 (no)
ES (1)	ES2155187T3 (no)
GE (1)	GEP20002271B (no)
GR (1)	GR3035676T3 (no)
HR (1)	HRP960117B1 (no)
HU (1)	HU222051B1 (no)
IL (1)	IL117395A (no)
IT (1)	IT1277835B1 (no)
MX (1)	MX9706927A (no)
NO (1)	NO319290B1 (no)
NZ (1)	NZ303982A (no)
PL (1)	PL184147B1 (no)
PT (1)	PT815126E (no)
RO (1)	RO118297B1 (no)
SK (1)	SK281899B6 (no)
TW (1)	TW565572B (no)
UA (1)	UA48962C2 (no)
WO (1)	WO1996028467A1 (no)
ZA (1)	ZA961983B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6017705A (en) *	1995-03-14	2000-01-25	Ludwig Institute For Cancer Research	Isolated nucleic acid molecules which are members of the MAGE-B family and uses thereof
IT1291776B1 (it) *	1997-02-07	1999-01-21	Menarini Ricerche Spa	Composti monociclici a quattro residui bifunzionali, aventi azione nk-2 antagonista
IT1304888B1 (it) *	1998-08-05	2001-04-05	Menarini Ricerche Spa	Composti monociclici ad azione nk-2 antagonista e formulazioni che licontengono
US20020016283A1 (en) *	2000-06-12	2002-02-07	Guttuso Thomas J.	Method of treating symptoms of hormonal variation, including hot flashes, using tachykinin receptor antagonist
EP1297826A1 (en) *	2001-09-27	2003-04-02	Menarini Ricerche S.p.A.	Nasal pharmaceutical compositions containing a NK-2 antagonist
ITFI20020239A1 (it) *	2002-12-06	2004-06-07	Menarini Ricerche Spa	Processo per la preparazione di composti peptidici biciclici.
ITFI20040221A1 (it) *	2004-10-27	2005-01-27	Guidotti & C Spa	Composizioni farmaceutiche a base di nk2 antagonisti per uso pediatrico
ITRM20120331A1 (it)	2012-07-12	2014-01-13	Guidotti & C Spa Labor	Composizioni pediatriche orali liquide contenenti nepadutant.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1262902B (it) *	1992-04-15	1996-07-22	Menarini Farma Ind	Composti triciclici antagonisti delle tachichinine, loro preparazione e loro uso in composizioni farmaceutiche.

1995
- 1995-03-13 IT IT95FI000044A patent/IT1277835B1/it active IP Right Grant
1996
- 1996-03-01 AR ARP960101616A patent/AR004476A1/es active IP Right Grant
- 1996-03-07 IL IL11739596A patent/IL117395A/xx not_active IP Right Cessation
- 1996-03-11 MX MX9706927A patent/MX9706927A/es unknown
- 1996-03-11 ES ES96907421T patent/ES2155187T3/es not_active Expired - Lifetime
- 1996-03-11 SK SK1212-97A patent/SK281899B6/sk not_active IP Right Cessation
- 1996-03-11 DK DK96907421T patent/DK0815126T3/da active
- 1996-03-11 CN CNB961937629A patent/CN1189477C/zh not_active Expired - Lifetime
- 1996-03-11 PL PL96322105A patent/PL184147B1/pl unknown
- 1996-03-11 EA EA199700223A patent/EA000697B1/ru not_active IP Right Cessation
- 1996-03-11 AU AU51059/96A patent/AU696528B2/en not_active Expired
- 1996-03-11 WO PCT/EP1996/001028 patent/WO1996028467A1/en not_active Ceased
- 1996-03-11 EE EE9700230A patent/EE03618B1/xx unknown
- 1996-03-11 UA UA97104990A patent/UA48962C2/uk unknown
- 1996-03-11 BR BR9607348A patent/BR9607348A/pt active IP Right Grant
- 1996-03-11 GE GEAP19963873A patent/GEP20002271B/en unknown
- 1996-03-11 CZ CZ19972862A patent/CZ287372B6/cs not_active IP Right Cessation
- 1996-03-11 JP JP52726796A patent/JP4618821B2/ja not_active Expired - Lifetime
- 1996-03-11 RO RO97-01700A patent/RO118297B1/ro unknown
- 1996-03-11 KR KR1019970706419A patent/KR100405009B1/ko not_active Expired - Lifetime
- 1996-03-11 EP EP96907421A patent/EP0815126B1/en not_active Expired - Lifetime
- 1996-03-11 PT PT96907421T patent/PT815126E/pt unknown
- 1996-03-11 NZ NZ303982A patent/NZ303982A/en not_active IP Right Cessation
- 1996-03-11 AT AT96907421T patent/ATE198481T1/de active
- 1996-03-11 HU HU9801835A patent/HU222051B1/hu active IP Right Grant
- 1996-03-11 DE DE69611438T patent/DE69611438T2/de not_active Expired - Lifetime
- 1996-03-12 ZA ZA9601983A patent/ZA961983B/xx unknown
- 1996-03-13 TW TW085103008A patent/TW565572B/zh not_active IP Right Cessation
- 1996-03-13 HR HR960117A patent/HRP960117B1/xx not_active IP Right Cessation
1997
- 1997-08-22 BG BG101849A patent/BG63208B1/bg unknown
- 1997-09-03 NO NO19974057A patent/NO319290B1/no not_active IP Right Cessation
- 1997-09-09 US US08/929,215 patent/US6150325A/en not_active Expired - Lifetime
2001
- 2001-03-30 GR GR20010400526T patent/GR3035676T3/el unknown

Also Published As

Publication number	Publication date
JP4618821B2 (ja)	2011-01-26
ITFI950044A0 (it)	1995-03-13
AU696528B2 (en)	1998-09-10
PT815126E (pt)	2001-06-29
HUP9801835A2 (hu)	1999-01-28
HRP960117A2 (en)	1997-08-31
UA48962C2 (uk)	2002-09-16
CN1183786A (zh)	1998-06-03
EE9700230A (et)	1998-04-15
CN1189477C (zh)	2005-02-16
DE69611438T2 (de)	2001-06-13
EE03618B1 (et)	2002-02-15
CZ287372B6 (en)	2000-11-15
RO118297B1 (ro)	2003-04-30
ZA961983B (en)	1997-09-29
IL117395A (en)	1999-12-31
BG63208B1 (bg)	2001-06-29
KR19980703011A (ko)	1998-09-05
JPH11501643A (ja)	1999-02-09
DE69611438D1 (de)	2001-02-08
NO319290B1 (no)	2005-07-11
SK281899B6 (sk)	2001-09-11
KR100405009B1 (ko)	2004-05-20
MX9706927A (es)	1997-11-29
GEP20002271B (en)	2000-10-25
HU222051B1 (hu)	2003-04-28
HRP960117B1 (en)	2001-06-30
IT1277835B1 (it)	1997-11-12
DK0815126T3 (da)	2001-05-07
EP0815126B1 (en)	2001-01-03
NO974057D0 (no)	1997-09-03
WO1996028467A1 (en)	1996-09-19
NZ303982A (en)	1998-04-27
PL322105A1 (en)	1998-01-05
AU5105996A (en)	1996-10-02
CZ286297A3 (cs)	1998-02-18
ES2155187T3 (es)	2001-05-01
IL117395A0 (en)	1996-07-23
GR3035676T3 (en)	2001-06-29
TW565572B (en)	2003-12-11
ITFI950044A1 (it)	1996-09-13
EA199700223A1 (ru)	1998-04-30
PL184147B1 (pl)	2002-09-30
ATE198481T1 (de)	2001-01-15
US6150325A (en)	2000-11-21
SK121297A3 (en)	1998-02-04
HUP9801835A3 (en)	2000-05-29
AR004476A1 (es)	1998-12-16
BG101849A (en)	1998-04-30
BR9607348A (pt)	1997-12-30
EA000697B1 (ru)	2000-02-28
EP0815126A1 (en)	1998-01-07

Publication	Publication Date	Title
EE03680B1 (et)	2002-04-15	Asendatud püridiinid, nende kasutamine ja farmatseutilised kompositsioonid
FI961270A7 (fi)	1996-05-03	Takykiniinien antagonisteja ja 3-(5-tetratsolyyli-bentsyyli)amino-piperidiinijohdannaisia
DK0723774T3 (da)	2001-01-29	Anvendelse af en antagonist for CGRP i en kosmetisk, farmaceutisk eller dermatologisk sammensætning og den opnåede sammensæ
DK0817779T3 (da)	2000-06-19	Nye taxoider, deres fremstilling og farmaceutiske præparater deraf
DK0876362T3 (da)	2004-02-02	Nye taxoider, deres fremstilling og farmaceutiske præparater deraf
DK0832104T3 (da)	2003-01-06	Dolastatinderivater, deres fremstilling og anvendelse
DK1019358T3 (da)	2003-09-01	3,3-diarylpropylaminer, deres anvendelse og fremstilling
NO981522L (no)	1998-04-03	Aminosyrederivater, deres fremstilling og anvendelse som endotelinantagonister
NO975020D0 (no)	1997-10-31	Azacykloalkanderivater, fremstilling derav og deres anvendelse i terapi
FI973221L (fi)	1997-10-20	1-aryyli-2-asyyliammo-etaaniyhdisteitä ja niiden käyttö neurokiniiniantagonisteina, erityisesti neurokiniini 1 antagonisteina
FI972988L (fi)	1997-09-11	Menetelmiä ja farmaseuttisia koostumuksia, joissa käytetään desmetyyliselegiliiniä
NO951418D0 (no)	1995-04-11	Peptidderivater, deres fremstilling og anvendelse som terapeutika
NO974057L (no)	1997-11-07	Bisykliske takykinin-antagonister, fremstilling derav og deres anvendelse i farmasöytisk sammensetning
DK60893D0 (da)	1993-05-26	Piperidinderivater, deres fremstilling og anvendelse
NO931364L (no)	1993-10-18	Tachykinin reseptorantagonister, isokinoloner og deres fremstilling
NO954763D0 (no)	1995-11-24	Piperidinderivater, deres fremstilling og anvendelse
NO985807D0 (no)	1998-12-11	Transdermale systemer inneholdende 2 aktive ingredienser i separate seksjoner, deres fremstillingsprosess og deres anvendelse som medikament
NO902248D0 (no)	1990-05-22	Renininhiberende peptider, deres fremstilling og anvendelse i legemidler.
DK0726250T3 (da)	2001-01-08	Substituerede benzensulfonylurinstoffer og -thiourinstoffer, fremgangsmåder til deres fremstilling og deres anvendelse til
NO973230D0 (no)	1997-07-11	Nye peptider, deres fremstilling og anvendelse
DK489889D0 (da)	1989-10-04	Dihydropyridinamider, deres fremstilling og anvendelse i laegemidler
NO982349D0 (no)	1998-05-22	Nye kinoksalindionderivater, deres fremstilling og anvendelse i legemidler
FR2774990B1 (fr)	2000-07-28	Nouveaux peptides, utilisation en therapeutique et compositions pharmaceutiques les renfermant
FI941915A7 (fi)	1994-10-28	2-amino-4-heteroaryyli-1,4-dihydropyridiineja, menetelmiä niiden valmistamiseksi ja niiden käyttö lääkeaineissa
SI0815126T1 (en)	2001-06-30	Bicyclic tachykinins antagonists, preparation thereof and their use in pharmaceutical composition

Legal Events

Date	Code	Title	Description
2016-03-21	MK1K	Patent expired