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NO953447L - New 4-aminopyridines, processes for their preparation and drugs containing them - Google Patents

New 4-aminopyridines, processes for their preparation and drugs containing them

Info

Publication number
NO953447L
NO953447L NO953447A NO953447A NO953447L NO 953447 L NO953447 L NO 953447L NO 953447 A NO953447 A NO 953447A NO 953447 A NO953447 A NO 953447A NO 953447 L NO953447 L NO 953447L
Authority
NO
Norway
Prior art keywords
atom
group
compounds
alkyl
aminopyridines
Prior art date
Application number
NO953447A
Other languages
Norwegian (no)
Other versions
NO953447D0 (en
Inventor
Wolfgang Von Der Saal
Reinhard Heck
Herbert Leinert
Thomas Poll
Karlheinz Stegmeier
Helmut Michel
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE4306506A external-priority patent/DE4306506A1/en
Priority claimed from DE19934312966 external-priority patent/DE4312966A1/en
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Publication of NO953447D0 publication Critical patent/NO953447D0/en
Publication of NO953447L publication Critical patent/NO953447L/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/74Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Nye 4-aminopyridiner med generell formel I (I) hvori R1 betegner gruppen R6-SO-NR7-, R6- S02-NR7-, R'-NR7-SO-, R6-NR7-S02-, R6-SO-0-, R6-SO,-0-, R6-0-SO- eller R6-O-SO,, R2 betegner et hydrogen- eller halogenatom, en cyano-, alkyl-, alkoksy- eller halogenalkyl- gruppe, X betegner et oksygenatom, et svovelatom eller NH-gruppen, RJ og R4 er like eller forskjellige og betegner hydrogenatomer eller alkylgrupper, R5 betegner et hydrogenatom, en alkylgruppe eller en aralkyl- gruppe. R6 betegner en alifatisk eller syklisk, eventuelt substituert rest, R7 betegner et hydrogenatom eller en alifatisk eller syklisk, eventuelt substituert rest, Y betegner en lineær eller for- grenet alkylenkjede, R8 og R9 er like eller forskjellige og betegner hydrogenatomer, aralkyl-, sykloalkyl- eller alkylgrupper som kan være en- eller flersubstituert med halogen, hydroksy, alkoksy, alkylkarbonyloksy, amin eller karboksy, eller R8 og R* danner sammen med N-atomet de er bundet til, en mettet ring som kan inneholde et ytterligere oksygen-, svovel- eller nitrogenatom, så vel som hydrater, solvater og fysio- logisk forenlige salter derav, og også optisk aktive former, racemater og dia- stereomerblandinger av disse forbind- elser. Fremgangsmåter for fremstilling av de ovennevnte forbindelser, lege- midler som inneholder slike forbindelser samt anvendelse av disse forbind- elser ved fremstilling av legemidler er også beskrevet.Novel 4-aminopyridines of general formula I (I) wherein R 1 represents the group R 6 -SO-NR 7 , R6-SO, -O-, R6-O-SO- or R6-O-SO4, R2 represents a hydrogen or halogen atom, a cyano, alkyl, alkoxy or haloalkyl group, X represents an oxygen atom, a sulfur atom or the NH group, R 1 and R 4 are the same or different and represent hydrogen atoms or alkyl groups, R 5 represents a hydrogen atom, an alkyl group or an aralkyl group. R6 represents an aliphatic or cyclic, optionally substituted residue, R7 represents a hydrogen atom or an aliphatic or cyclic, optionally substituted residue, Y represents a linear or branched alkylene chain, R8 and R9 are the same or different and represent hydrogen atoms, aralkyl, cycloalkyl - or alkyl groups which may be mono- or poly-substituted with halogen, hydroxy, alkoxy, alkylcarbonyloxy, amine or carboxy, or R8 and R * together with the N atom to which they are attached form a saturated ring which may contain an additional oxygen, sulfur or nitrogen atom, as well as hydrates, solvates and physiologically compatible salts thereof, and also optically active forms, racemates and diastereomeric mixtures of these compounds. Methods for the preparation of the above compounds, drugs containing such compounds and the use of these compounds in the manufacture of drugs are also described.

NO953447A 1993-03-03 1995-09-01 New 4-aminopyridines, processes for their preparation and drugs containing them NO953447L (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE4306506A DE4306506A1 (en) 1993-03-03 1993-03-03 Novel 4-alkylaminopyridines - processes for their preparation and medicaments containing these compounds
DE19934312966 DE4312966A1 (en) 1993-04-21 1993-04-21 Novel 4-aminopyridines - process for their preparation and medicaments containing these compounds
PCT/EP1994/000608 WO1994020467A1 (en) 1993-03-03 1994-03-02 New 4-aminopyridines, process for preparing the same and medicaments containing the same

Publications (2)

Publication Number Publication Date
NO953447D0 NO953447D0 (en) 1995-09-01
NO953447L true NO953447L (en) 1995-09-01

Family

ID=25923593

Family Applications (1)

Application Number Title Priority Date Filing Date
NO953447A NO953447L (en) 1993-03-03 1995-09-01 New 4-aminopyridines, processes for their preparation and drugs containing them

Country Status (22)

Country Link
EP (1) EP0687253B1 (en)
JP (1) JPH08507503A (en)
KR (1) KR100252551B1 (en)
CN (1) CN1046710C (en)
AT (1) ATE174590T1 (en)
AU (1) AU682026B2 (en)
CA (1) CA2156729A1 (en)
CZ (1) CZ225495A3 (en)
DE (1) DE59407494D1 (en)
DK (1) DK0687253T3 (en)
ES (1) ES2127919T3 (en)
FI (1) FI954105A7 (en)
GR (1) GR3029691T3 (en)
HU (1) HUT72898A (en)
IL (1) IL108786A (en)
NO (1) NO953447L (en)
NZ (1) NZ262725A (en)
PL (1) PL176455B1 (en)
RU (1) RU2126388C1 (en)
SK (1) SK108295A3 (en)
TW (1) TW257757B (en)
WO (1) WO1994020467A1 (en)

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AU725403B2 (en) * 1996-09-13 2000-10-12 Merck & Co., Inc. Thrombin inhibitors
GB9821483D0 (en) 1998-10-03 1998-11-25 Glaxo Group Ltd Chemical compounds
UA56197C2 (en) 1996-11-08 2003-05-15 Зенека Лімітед Heterocyclic derivatives
TW499412B (en) 1996-11-26 2002-08-21 Dimensional Pharm Inc Aminoguanidines and alkoxyguanidines as protease inhibitors
US6127191A (en) * 1996-12-03 2000-10-03 3-Dimensional Pharmaceuticals, Inc. Aminobenzenedicarboxylic acid-based combinatorial libraries
AU5999698A (en) 1997-02-13 1998-09-08 Zeneca Limited Heterocyclic compounds useful as oxido-squalene cyclase inhibitors
US6391880B1 (en) 1997-02-13 2002-05-21 Zeneca Limited Heterocyclic compounds useful as oxido-squalene cyclase inhibitors
GB9715895D0 (en) 1997-07-29 1997-10-01 Zeneca Ltd Heterocyclic compounds
JP4327915B2 (en) * 1998-03-30 2009-09-09 株式会社デ・ウエスタン・セラピテクス研究所 Sulfonamide derivatives
ID27509A (en) 1998-10-06 2001-04-12 Dainippon Pharmaceutical Co SUBSTITUTION OF PYRIDINE SUBSTITUTED-2,3 THE PROCESS OF MAKING, PHARMACEUTICAL COMPOSITION THAT CONTAINS THE COMPOUND, AND THE COMPOUND
GB9902989D0 (en) 1999-02-11 1999-03-31 Zeneca Ltd Heterocyclic derivatives
AR023510A1 (en) 1999-04-21 2002-09-04 Astrazeneca Ab A TEAM OF PARTS, PHARMACEUTICAL FORMULATION AND USE OF A THROMBIN INHIBITOR.
MXPA03000963A (en) 2000-08-04 2004-04-05 Dimensional Pharm Inc Cyclic oxyguanidine protease inhibitors.
AU9233101A (en) * 2000-10-04 2002-04-15 Kissei Pharmaceutical 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation
EP1399137A4 (en) * 2001-05-07 2005-12-14 Smithkline Beecham Corp Sulfonamides
EP1385495A4 (en) * 2001-05-07 2005-12-21 Smithkline Beecham Corp Sulfonamides
ATE402700T1 (en) 2002-08-27 2008-08-15 Merck Patent Gmbh GLYCINAMIDE DERIVATIVES AS RAF-KINASE INHIBITORS
WO2004026823A1 (en) * 2002-09-20 2004-04-01 Pfizer Products Inc. Amide and sulfonamide ligands for the estrogen receptor
AU2004291262C1 (en) 2003-11-05 2011-08-11 F. Hoffmann-La Roche Ag Phenyl derivatives as PPAR agonists
WO2008104994A2 (en) * 2007-02-28 2008-09-04 Advinus Therapeutics Private Limited 2,2,2-tri-substituted acetamide derivatives as glucokinase activators, their process and pharmaceutical application
RU2354647C2 (en) * 2007-06-28 2009-05-10 Общество С Ограниченной Ответственностью "Бионика" New compounds with thrombin inhibiting function, and based pharmaceutical compositions
RU2353619C2 (en) * 2007-06-28 2009-04-27 Общество С Ограниченной Ответственностью "Бионика" Novel compounds possessing anticoagulant function, based on them pharmaceutical compositions for treatment of thrombotic conditions and plasma-substituting solution for correction of hypercoagulation disorders in hemodilution
GB0815782D0 (en) 2008-08-29 2008-10-08 Xention Ltd Novel potassium channel blockers
GB0815784D0 (en) 2008-08-29 2008-10-08 Xention Ltd Novel potassium channel blockers
GB0815781D0 (en) 2008-08-29 2008-10-08 Xention Ltd Novel potassium channel blockers
US8265575B2 (en) * 2009-06-16 2012-09-11 Mediatek Inc. Methods for handling a transmitting process and communication apparatuses utilizing the same
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RU2685261C1 (en) * 2018-04-05 2019-04-17 Общество с ограниченной ответственностью "ФК ЛАБОРАТОРИЗ" 4-amino-1-{2-[3-methyl-5-(benzenesulfonyloxy]phenoxy]ethyl}-pyridium chloride substance, having the biologically active agent properties, influencing the mammals blood coagulability naturally running processes, anticoagulant on its basis and its obtaining method by chemical synthesis
CN109172573B (en) * 2018-09-12 2021-01-26 黑龙江中桂制药有限公司 Oral antithrombotic drug and application thereof
CN110669337B (en) * 2019-07-08 2020-09-25 中国科学院长春应用化学研究所 Aromatic diamine monomer and preparation method thereof
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Also Published As

Publication number Publication date
SK108295A3 (en) 1996-06-05
CN1046710C (en) 1999-11-24
WO1994020467A1 (en) 1994-09-15
CZ225495A3 (en) 1996-01-17
CA2156729A1 (en) 1994-09-15
DK0687253T3 (en) 1999-08-23
FI954105A0 (en) 1995-09-01
EP0687253B1 (en) 1998-12-16
HUT72898A (en) 1996-06-28
JPH08507503A (en) 1996-08-13
CN1119858A (en) 1996-04-03
ATE174590T1 (en) 1999-01-15
NO953447D0 (en) 1995-09-01
NZ262725A (en) 1997-05-26
RU2126388C1 (en) 1999-02-20
ES2127919T3 (en) 1999-05-01
TW257757B (en) 1995-09-21
KR100252551B1 (en) 2000-05-01
HU9502568D0 (en) 1995-11-28
GR3029691T3 (en) 1999-06-30
DE59407494D1 (en) 1999-01-28
IL108786A (en) 1999-04-11
PL310520A1 (en) 1995-12-27
PL176455B1 (en) 1999-05-31
IL108786A0 (en) 1994-06-24
AU6257494A (en) 1994-09-26
EP0687253A1 (en) 1995-12-20
AU682026B2 (en) 1997-09-18
KR960701019A (en) 1996-02-24
FI954105A7 (en) 1995-09-01

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