NO951811D0 - Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse - Google Patents

Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse

Info

Publication number: NO951811D0
Authority: NO; Norway
Prior art keywords: quinoline; preparation; benzimidazole derivatives; benzimidazole; derivatives
Prior art date: 1994-05-10

Application number

NO951811A

Other languages

English (en)

Other versions

NO951811L (no

Inventor

George Pascal

Mireille Sevrin

Michel Peynot

Original Assignee

Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-05-10

Filing date

1995-05-09

Publication date

1995-05-09

1995-05-09 Application filed by Synthelabo filed Critical Synthelabo

1995-05-09 Publication of NO951811D0 publication Critical patent/NO951811D0/no

1995-11-13 Publication of NO951811L publication Critical patent/NO951811L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/16—Peri-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/16—Peri-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

NO951811A 1994-05-10 1995-05-09 Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse NO951811L (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9405715A FR2719843B1 (fr)	1994-05-10	1994-05-10	Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number	Publication Date
NO951811D0 true NO951811D0 (no)	1995-05-09
NO951811L NO951811L (no)	1995-11-13

Family

ID=9463058

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO951811A NO951811L (no)	1994-05-10	1995-05-09	Kinolin- og benzimidazolderivater, deres fremstilling og anvendelse

Country Status (18)

Country	Link
US (1)	US5512590A (no)
EP (1)	EP0682025A1 (no)
JP (1)	JPH0853450A (no)
KR (1)	KR950032193A (no)
CN (1)	CN1115761A (no)
AU (1)	AU1793595A (no)
CA (1)	CA2148951A1 (no)
CZ (1)	CZ119495A3 (no)
FI (1)	FI952249A7 (no)
FR (1)	FR2719843B1 (no)
HU (1)	HUT72666A (no)
IL (1)	IL113672A (no)
NO (1)	NO951811L (no)
NZ (1)	NZ272089A (no)
PL (1)	PL308517A1 (no)
RU (1)	RU95107157A (no)
SK (1)	SK59695A3 (no)
ZA (1)	ZA953750B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0120345D0 (en) *	2001-08-21	2001-10-17	Merck Sharp & Dohme	Therapeutic agents
CA2509561A1 (en) *	2002-12-18	2004-07-15	Mallinckrodt Inc.	Synthesis of heteroaryl acetamides
ATE451371T1 (de) *	2004-06-22	2009-12-15	Mallinckrodt Inc	Synthese von heteroarylacetamiden aus reaktionsmischungen mit reduziertem wassergehalt
JP2008538748A (ja) *	2005-04-07	2008-11-06	ハイシアム，インコーポレイテッド	不安、物質乱用及び依存の予防のための改良型方法及び組成物
US7812013B2 (en)	2005-06-14	2010-10-12	Schering Corporation	Macrocyclic heterocyclic aspartyl protease inhibitors
US12522583B2 (en)	2018-11-07	2026-01-13	Dana-Farber Cancer Institute, Inc.	Benzimidazole derivatives and aza-benzimidazole derivatives as Janus kinase 2 inhibitors and uses thereof
US12415816B2 (en)	2018-11-07	2025-09-16	Dana-Farber Cancer Institute, Inc.	Benzothiazole derivatives and 7-aza-benzothiazole derivatives as janus kinase 2 inhibitors and uses thereof
WO2020097400A1 (en)	2018-11-07	2020-05-14	Dana-Farber Cancer Institute, Inc.	Imidazopyridine derivatives and aza-imidazopyridine derivatives as janus kinase 2 inhibitors and uses thereof
US20240360132A9 (en) *	2019-10-03	2024-10-31	Dana-Farber Cancer Institute, Inc.	Tricyclic kinase inhibitors and uses thereof
EP4146639A1 (en)	2020-05-06	2023-03-15	Ajax Therapeutics, Inc.	6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
TW202241889A (zh)	2020-12-23	2022-11-01	美商雅捷可斯治療公司	作為ｊａｋ２抑制劑之６－雜芳基氧基苯并咪唑及氮雜苯并咪唑
WO2023086319A1 (en)	2021-11-09	2023-05-19	Ajax Therapeutics, Inc.	6-he tero aryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
TW202325289A (zh)	2021-11-09	2023-07-01	美商雅捷可斯治療公司	Ｊａｋ２抑制劑之形式及組合物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3732243A (en) *	1970-06-23	1973-05-08	Sankyo Co	2-(p-bromophenyl)-9-dimethyl-amino-propyl-9h-imidazo(1,2-a)benzimidazole
FR2568879B1 (fr) *	1984-08-07	1986-12-12	Synthelabo	Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2593817B1 (fr) *	1986-01-31	1988-04-15	Synthelabo	Derives de tetrahydro-5,6,7,8 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
KR0167346B1 (ko) *	1989-06-09	1999-01-15	로버트 에이. 아미테이지	중추신경계 활성을 갖는 헤테로사이클릭 아민
EP0607076A1 (fr) *	1993-01-15	1994-07-20	Synthelabo	Dérivés de 9h-imidazo 1,2-a benzimidazole-3-acétamide à activité GABA

1994
- 1994-05-10 FR FR9405715A patent/FR2719843B1/fr not_active Expired - Fee Related
1995
- 1995-05-03 EP EP95401014A patent/EP0682025A1/fr not_active Withdrawn
- 1995-05-05 RU RU95107157/04A patent/RU95107157A/ru unknown
- 1995-05-09 IL IL11367295A patent/IL113672A/xx active IP Right Grant
- 1995-05-09 SK SK596-95A patent/SK59695A3/sk unknown
- 1995-05-09 PL PL95308517A patent/PL308517A1/xx unknown
- 1995-05-09 NZ NZ272089A patent/NZ272089A/xx unknown
- 1995-05-09 NO NO951811A patent/NO951811L/no unknown
- 1995-05-09 CA CA002148951A patent/CA2148951A1/en not_active Abandoned
- 1995-05-09 ZA ZA953750A patent/ZA953750B/xx unknown
- 1995-05-09 CZ CZ951194A patent/CZ119495A3/cs unknown
- 1995-05-09 CN CN95105469A patent/CN1115761A/zh active Pending
- 1995-05-09 AU AU17935/95A patent/AU1793595A/en not_active Abandoned
- 1995-05-09 US US08/437,053 patent/US5512590A/en not_active Expired - Fee Related
- 1995-05-09 KR KR1019950011237A patent/KR950032193A/ko not_active Withdrawn
- 1995-05-09 JP JP7110538A patent/JPH0853450A/ja active Pending
- 1995-05-09 HU HU9501369A patent/HUT72666A/hu unknown
- 1995-05-09 FI FI952249A patent/FI952249A7/fi unknown

Also Published As

Publication number	Publication date
NO951811L (no)	1995-11-13
FI952249A0 (fi)	1995-05-09
KR950032193A (ko)	1995-12-20
FR2719843A1 (fr)	1995-11-17
ZA953750B (en)	1996-04-02
FI952249L (fi)	1995-11-11
US5512590A (en)	1996-04-30
CA2148951A1 (en)	1995-11-11
JPH0853450A (ja)	1996-02-27
CZ119495A3 (en)	1995-12-13
NZ272089A (en)	1996-07-26
IL113672A0 (en)	1995-08-31
FR2719843B1 (fr)	1996-06-07
AU1793595A (en)	1995-11-16
IL113672A (en)	1997-11-20
SK59695A3 (en)	1995-12-06
EP0682025A1 (fr)	1995-11-15
FI952249A7 (fi)	1995-11-11
PL308517A1 (en)	1995-11-13
CN1115761A (zh)	1996-01-31
RU95107157A (ru)	1997-03-20
HUT72666A (en)	1996-05-28

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