NO943803D0 - Acylaminoindolderivater som 5-HT 1 agonister - Google Patents

Acylaminoindolderivater som 5-HT 1 agonister

Info

Publication number: NO943803D0
Authority: NO; Norway
Prior art keywords: aryl; alkyl; alkylaryl; hydrogen; pct
Prior art date: 1992-04-10

Application number

NO943803A

Other languages

English (en)

Other versions

NO943803L (no

NO309860B1 (no

Inventor

John E Macor

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-04-10

Filing date

1994-10-07

Publication date

1994-10-07

1994-10-07 Application filed by Pfizer filed Critical Pfizer

1994-10-07 Publication of NO943803L publication Critical patent/NO943803L/no

1994-10-07 Publication of NO943803D0 publication Critical patent/NO943803D0/no

2001-04-09 Publication of NO309860B1 publication Critical patent/NO309860B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Diabetes (AREA)
Heart & Thoracic Surgery (AREA)
Child & Adolescent Psychology (AREA)
Cardiology (AREA)
Hematology (AREA)
Obesity (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Supply Devices, Intensifiers, Converters, And Telemotors (AREA)
Materials For Photolithography (AREA)
Soft Magnetic Materials (AREA)

NO943803A 1992-04-10 1994-10-07 Acylaminoindolderivater som 5-HT 1 agonister og farmasøytisk preparat NO309860B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US86638292A	1992-04-10	1992-04-10
PCT/US1993/001807 WO1993021180A1 (en)	1992-04-10	1993-03-04	Acylaminoindole derivatives as 5-ht1 agonists

Publications (3)

Publication Number	Publication Date
NO943803L NO943803L (no)	1994-10-07
NO943803D0 true NO943803D0 (no)	1994-10-07
NO309860B1 NO309860B1 (no)	2001-04-09

Family

ID=25347493

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO943803A NO309860B1 (no)	1992-04-10	1994-10-07	Acylaminoindolderivater som 5-HT 1 agonister og farmasøytisk preparat

Country Status (31)

Country	Link
US (1)	US5498626A (no)
EP (1)	EP0635015B1 (no)
JP (1)	JP2544704B2 (no)
KR (1)	KR0179074B1 (no)
CN (1)	CN1038506C (no)
AT (1)	ATE148465T1 (no)
AU (1)	AU670270B2 (no)
BR (1)	BR9306221A (no)
CA (1)	CA2132706C (no)
CZ (1)	CZ282653B6 (no)
DE (1)	DE69307875T2 (no)
DK (1)	DK0635015T3 (no)
EG (1)	EG20466A (no)
ES (1)	ES2097496T3 (no)
FI (2)	FI111256B (no)
GR (1)	GR3022767T3 (no)
HR (1)	HRP930753B1 (no)
HU (1)	HUT64060A (no)
IL (1)	IL105309A0 (no)
MX (1)	MX9301996A (no)
MY (1)	MY115278A (no)
NO (1)	NO309860B1 (no)
NZ (1)	NZ251047A (no)
PL (1)	PL172232B1 (no)
RU (1)	RU2110516C1 (no)
SK (1)	SK278182B6 (no)
TW (1)	TW394769B (no)
UA (1)	UA34452C2 (no)
WO (1)	WO1993021180A1 (no)
YU (1)	YU48916B (no)
ZA (1)	ZA932536B (no)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5559246A (en) *	1990-10-15	1996-09-24	Pfizer Inc.	Indole derivatives
US5607951A (en) *	1990-10-15	1997-03-04	Pfizer Inc	Indole derivatives
US5545644A (en) *	1990-10-15	1996-08-13	Pfizer Inc.	Indole derivatives
US5559129A (en) *	1990-10-15	1996-09-24	Pfizer Inc	Indole derivatives
US5578612A (en) *	1990-10-15	1996-11-26	Pfizer Inc.	Indole derivatives
US6380233B1 (en)	1992-04-07	2002-04-30	Pfizer Inc	Indole derivatives as 5-HT1 agonists
JP2644088B2 (ja)	1992-04-07	1997-08-25	フアイザー・インコーポレイテツド	５−ｈｔ１作動薬としてのインドール誘導体
ES2070772B1 (es) *	1993-08-09	1996-02-16	Pfizer	Derivados de acilaminoindol
KR100191973B1 (ko) *	1993-08-31	1999-06-15	디. 제이. 우드, 스피겔 알렌 제이	5-아릴인돌 유도체
GB9402016D0 (en) *	1994-02-02	1994-03-30	Merck Sharp & Dohme	Therapeutic agents
GB9402011D0 (en) *	1994-02-02	1994-03-30	Merck Sharp & Dohme	Therapeutic agents
FI971334L (fi) *	1994-08-03	1997-04-01	Asta Medica Ag	Indoli-, indatsoli-, pyridopyrroli- ja pyridopyratsolijohdannaiset, joilla on antiastmaattinen, antiallerginen, anti-inflammatorinen ja immunomoduloiva vaikutus
GB9417310D0 (en)	1994-08-27	1994-10-19	Pfizer Ltd	Therapeutic agents
GB9420503D0 (en) *	1994-10-11	1994-11-23	Pfizer Ltd	Therapeutic agents
GB9420529D0 (en)	1994-10-12	1994-11-30	Pfizer Ltd	Indoles
AU3170099A (en) *	1998-04-16	1999-11-08	Yamanouchi Pharmaceutical Co., Ltd.	Remedies for obesity
US5994352A (en) *	1998-11-13	1999-11-30	Pfizer Inc.	5-arylindole derivatives
US20050032750A1 (en) *	2003-01-22	2005-02-10	Steiner Mitchell S.	Treating androgen deficiency in female (ADIF)-associated conditions with SARMS
CN101939306A (zh) *	2007-12-07	2011-01-05	美国辉瑞有限公司	反式-n-异丁基-3-氟-3-[3-氟-4-(吡咯烷-1-基-甲基)-苯基]环丁烷甲酰胺的甲苯磺酸盐
US20140206667A1 (en)	2012-11-14	2014-07-24	Michela Gallagher	Methods and compositions for treating schizophrenia
CN103408535B (zh) *	2013-08-13	2016-03-02	张家港威胜生物医药有限公司	一种依来曲普坦中间体-5-溴-3-(n-甲基吡咯啉-2-基甲基)-1h-吲哚合成工艺

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA795239B (en) *	1978-10-12	1980-11-26	Glaxo Group Ltd	Heterocyclic compounds
ZA815541B (en) *	1980-08-12	1983-03-30	Glaxo Group Ltd	Heterocyclic compounds
CH652394A5 (fr) *	1980-08-12	1985-11-15	Glaxo Group Ltd	Derives indoliques, leur preparation et medicaments les renfermant.
GB8600397D0 (en) *	1986-01-08	1986-02-12	Glaxo Group Ltd	Chemical compounds
GB8719167D0 (en) *	1987-08-13	1987-09-23	Glaxo Group Ltd	Chemical compounds
GB8724912D0 (en) *	1987-10-23	1987-11-25	Wellcome Found	Indole derivatives
GB8819024D0 (en) *	1988-08-10	1988-09-14	Glaxo Group Ltd	Chemical compounds
IL96891A0 (en) *	1990-01-17	1992-03-29	Merck Sharp & Dohme	Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them
CA2042295A1 (fr) *	1990-05-15	1991-11-16	Jacques Chauveau	Derives de mediateurs endogenes, leurs sels, procede de preparation, applications, et compositions les renfermant
HU219974B (hu) *	1990-06-07	2001-10-28	Astrazeneca Ab,	Heterociklusos csoporttal helyettesített indolszármazék, előállítása és a vegyületet hatóanyagként tartalmazó gyógyszerkészítmények
HU225055B1 (en) *	1990-10-15	2006-05-29	Pfizer	Indole derivatives, their intermediates, process for production them and pharmaceutical compositions containing the compounds
US5208248A (en) *	1991-01-11	1993-05-04	Merck Sharpe & Dohme, Ltd.	Indazole-substituted five-membered heteroaromatic compounds
SK278998B6 (sk) *	1991-02-01	1998-05-06	Merck Sharp & Dohme Limited	Deriváty imidazolu, triazolu a tetrazolu, spôsob i
EP0619805B1 (en) *	1991-11-25	2000-03-15	Pfizer Inc.	5-(hetero- or carbocyclylamino)-indole derivatives, their preparation and their use as 5-ht1 agonists

1993
- 1993-03-04 DK DK93907096.7T patent/DK0635015T3/da active
- 1993-03-04 JP JP5518302A patent/JP2544704B2/ja not_active Expired - Fee Related
- 1993-03-04 PL PL93305558A patent/PL172232B1/pl not_active IP Right Cessation
- 1993-03-04 UA UA94105907A patent/UA34452C2/uk unknown
- 1993-03-04 DE DE69307875T patent/DE69307875T2/de not_active Expired - Fee Related
- 1993-03-04 CZ CZ942477A patent/CZ282653B6/cs not_active IP Right Cessation
- 1993-03-04 EP EP93907096A patent/EP0635015B1/en not_active Expired - Lifetime
- 1993-03-04 NZ NZ251047A patent/NZ251047A/en unknown
- 1993-03-04 AU AU37821/93A patent/AU670270B2/en not_active Ceased
- 1993-03-04 RU RU94045902/04A patent/RU2110516C1/ru not_active IP Right Cessation
- 1993-03-04 CA CA002132706A patent/CA2132706C/en not_active Expired - Fee Related
- 1993-03-04 BR BR9306221A patent/BR9306221A/pt not_active Application Discontinuation
- 1993-03-04 ES ES93907096T patent/ES2097496T3/es not_active Expired - Lifetime
- 1993-03-04 WO PCT/US1993/001807 patent/WO1993021180A1/en not_active Ceased
- 1993-03-04 US US08/295,792 patent/US5498626A/en not_active Expired - Fee Related
- 1993-03-04 AT AT93907096T patent/ATE148465T1/de not_active IP Right Cessation
- 1993-03-04 SK SK1207-94A patent/SK278182B6/sk unknown
- 1993-03-04 KR KR1019940703551A patent/KR0179074B1/ko not_active Expired - Fee Related
- 1993-03-09 TW TW082101732A patent/TW394769B/zh active
- 1993-04-02 HR HR930753A patent/HRP930753B1/xx not_active IP Right Cessation
- 1993-04-05 IL IL105309A patent/IL105309A0/xx not_active IP Right Cessation
- 1993-04-06 MX MX9301996A patent/MX9301996A/es unknown
- 1993-04-07 EG EG21493A patent/EG20466A/xx active
- 1993-04-08 MY MYPI93000646A patent/MY115278A/en unknown
- 1993-04-08 ZA ZA932536A patent/ZA932536B/xx unknown
- 1993-04-08 FI FI931613A patent/FI111256B/fi not_active IP Right Cessation
- 1993-04-09 CN CN93104439A patent/CN1038506C/zh not_active Expired - Fee Related
- 1993-04-09 YU YU25593A patent/YU48916B/sh unknown
- 1993-04-09 HU HU9301048A patent/HUT64060A/hu unknown
1994
- 1994-10-07 NO NO943803A patent/NO309860B1/no not_active IP Right Cessation
1997
- 1997-03-07 GR GR970400451T patent/GR3022767T3/el unknown
2001
- 2001-02-05 FI FI20010214A patent/FI20010214A7/fi unknown

Also Published As

Publication number	Publication date
NZ251047A (en)	1996-09-25
JPH07501831A (ja)	1995-02-23
AU670270B2 (en)	1996-07-11
CZ282653B6 (cs)	1997-08-13
HRP930753A2 (en)	1994-10-31
HU9301048D0 (en)	1993-06-28
TW394769B (en)	2000-06-21
CA2132706C (en)	1998-08-04
CA2132706A1 (en)	1993-10-28
IL105309A0 (en)	1993-08-18
FI20010214L (fi)	2001-02-05
EP0635015A1 (en)	1995-01-25
EP0635015B1 (en)	1997-01-29
MY115278A (en)	2003-05-31
FI20010214A7 (fi)	2001-02-05
SK278182B6 (en)	1996-03-06
NO943803L (no)	1994-10-07
ZA932536B (en)	1994-10-08
JP2544704B2 (ja)	1996-10-16
EG20466A (en)	1999-05-31
MX9301996A (es)	1994-03-31
KR0179074B1 (ko)	1999-03-20
WO1993021180A1 (en)	1993-10-28
RU94045902A (ru)	1996-08-27
FI931613L (fi)	1993-10-11
ES2097496T3 (es)	1997-04-01
DE69307875T2 (de)	1997-05-22
HUT64060A (en)	1993-11-29
HRP930753B1 (en)	2000-10-31
AU3782193A (en)	1993-11-18
CZ247794A3 (en)	1995-07-12
DE69307875D1 (de)	1997-03-13
RU2110516C1 (ru)	1998-05-10
CN1080288A (zh)	1994-01-05
KR950700903A (ko)	1995-02-20
UA34452C2 (uk)	2001-03-15
CN1038506C (zh)	1998-05-27
BR9306221A (pt)	1998-06-30
GR3022767T3 (en)	1997-06-30
YU48916B (sh)	2002-11-15
FI111256B (fi)	2003-06-30
ATE148465T1 (de)	1997-02-15
PL172232B1 (pl)	1997-08-29
DK0635015T3 (da)	1997-03-17
SK120794A3 (en)	1995-05-10
US5498626A (en)	1996-03-12
FI931613A0 (fi)	1993-04-08
YU25593A (sh)	1996-10-09
NO309860B1 (no)	2001-04-09

Publication	Publication Date	Title
NO943803D0 (no)	1994-10-07	Acylaminoindolderivater som 5-HT 1 agonister
MX9206762A (es)	1993-05-01	Derivados de indol
MY108909A (en)	1996-11-30	Indole derivatives
MY111683A (en)	2000-11-30	Indole derivatives.
CA2117643A1 (en)	1993-09-16	Indole Derivatives

Legal Events

Date	Code	Title	Description
2004-12-27	MM1K	Lapsed by not paying the annual fees