NO944680L - New thienothiazine derivatives, a process for their preparation and their use - Google Patents
New thienothiazine derivatives, a process for their preparation and their useInfo
- Publication number
- NO944680L NO944680L NO944680A NO944680A NO944680L NO 944680 L NO944680 L NO 944680L NO 944680 A NO944680 A NO 944680A NO 944680 A NO944680 A NO 944680A NO 944680 L NO944680 L NO 944680L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- halogen
- new
- thienothiazine derivatives
- thienothiazine
- Prior art date
Links
- TZIJDLHRFZUDHD-UHFFFAOYSA-N 2h-thieno[2,3-e]thiazine Chemical class C1=CNSC2=C1SC=C2 TZIJDLHRFZUDHD-UHFFFAOYSA-N 0.000 title 1
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000002950 monocyclic group Chemical group 0.000 abstract 1
- 125000003367 polycyclic group Chemical group 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Det er beskrevet tienotlazlnderlvater med formel (I) (D hvori X betyr en enkeltblnding eller en 5 - 12-leddet, mono- eller polycykllsk, eventuelt delvis hydrert aryl- eller heteroarylrest som eventuelt kan være substituert med halogen, laverealkyl eller laverealkoksy, Y betyr en enkeltbindlng eller et heteroatom, R betyr en mono- eller polycyklisk, eventuelt delvis hydrert 5 - 12-leddet aryl- eller heteroarylrest som eventuelt kan være substituert en eller flere ganger med halogen, laverealkyl eller laverealkoksy, A betyr halogen, og B betyr hydrogen eller halogen. Det er videre beskrevet en fremgangsmåte for fremstilling av forbindelsene samt deres anvendelse som farmasøy-tika.Thienothiazol substituents of formula (I) (D) are disclosed in which a single bond or a heteroatom, R means a mono- or polycyclic, optionally partially hydrated 5-12 membered aryl or heteroaryl radical which may or may not be substituted one or more times by halogen, lower alkyl or lower alkoxy, A means halogen, and B means hydrogen or a halogen A process for the preparation of the compounds as well as their use as pharmaceuticals is further described.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AT0246193A AT400845B (en) | 1993-12-06 | 1993-12-06 | NEW THIENOTHIAZINE DERIVATIVES, A METHOD FOR THEIR PRODUCTION AND THEIR USE |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO944680D0 NO944680D0 (en) | 1994-12-05 |
| NO944680L true NO944680L (en) | 1995-06-07 |
Family
ID=3534780
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO944680A NO944680L (en) | 1993-12-06 | 1994-12-05 | New thienothiazine derivatives, a process for their preparation and their use |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP0657459A1 (en) |
| JP (1) | JPH07252260A (en) |
| CN (1) | CN1111634A (en) |
| AT (1) | AT400845B (en) |
| CA (1) | CA2137443A1 (en) |
| NO (1) | NO944680L (en) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19632556A1 (en) | 1996-08-13 | 1998-02-19 | Bayer Ag | Process for the production of high-rubber ABS molding compounds |
| US20010049379A1 (en) | 1997-08-27 | 2001-12-06 | Lowe John Adams | 2-aminopyridines containing fused ring substituents |
| HN1998000118A (en) * | 1997-08-27 | 1999-02-09 | Pfizer Prod Inc | 2 - AMINOPYRIDINES CONTAINING SUBSTITUTES FOR CONDENSED RINGS. |
| BR112013006272A2 (en) | 2010-09-17 | 2019-09-24 | Purdue Pharma Lp | pyridine compounds and their uses |
| US9656959B2 (en) * | 2010-12-22 | 2017-05-23 | Purdue Pharma L.P. | Substituted pyridines as sodium channel blockers |
| TWI644899B (en) | 2013-02-04 | 2018-12-21 | 健生藥品公司 | Flap modulators |
| JP6424173B2 (en) | 2013-02-04 | 2018-11-14 | ヤンセン ファーマシューティカ エヌ．ベー． | FLAP regulator |
| CN111646987B (en) * | 2020-06-05 | 2022-06-24 | 湖南师范大学 | 5-aminothiazole non-steroidal anti-inflammatory compound and preparation method and application thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU518216B2 (en) * | 1977-09-06 | 1981-09-17 | Hafslund Nycomed Pharma Aktiengesellschaft | Thienothiazine derivatives |
| DE69027594T2 (en) * | 1989-11-30 | 1996-10-31 | Nippon Hypox Lab Inc | A MEDICINE CONTAINING THIAZINE DIOXIDE DERIVATIVE |
| AT399880B (en) * | 1992-07-03 | 1995-08-25 | Chem Pharm Forsch Gmbh | NEW THIENOTHIAZINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE |
-
1993
- 1993-12-06 AT AT0246193A patent/AT400845B/en not_active IP Right Cessation
-
1994
- 1994-11-21 EP EP94118276A patent/EP0657459A1/en not_active Withdrawn
- 1994-12-05 CN CN94119890A patent/CN1111634A/en active Pending
- 1994-12-05 NO NO944680A patent/NO944680L/en unknown
- 1994-12-05 JP JP6300976A patent/JPH07252260A/en not_active Withdrawn
- 1994-12-06 CA CA002137443A patent/CA2137443A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2137443A1 (en) | 1995-06-07 |
| CN1111634A (en) | 1995-11-15 |
| EP0657459A1 (en) | 1995-06-14 |
| JPH07252260A (en) | 1995-10-03 |
| NO944680D0 (en) | 1994-12-05 |
| AT400845B (en) | 1996-03-25 |
| ATA246193A (en) | 1995-08-15 |
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