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NO930222D0 - Quinuclidin-derivater - Google Patents

Quinuclidin-derivater

Info

Publication number
NO930222D0
NO930222D0 NO1993930222A NO930222A NO930222D0 NO 930222 D0 NO930222 D0 NO 930222D0 NO 1993930222 A NO1993930222 A NO 1993930222A NO 930222 A NO930222 A NO 930222A NO 930222 D0 NO930222 D0 NO 930222D0
Authority
NO
Norway
Prior art keywords
quinuclidine derivatives
quinuclidine
derivatives
migraine
antagonists
Prior art date
Application number
NO1993930222A
Other languages
English (en)
Other versions
NO930222L (no
NO302172B1 (no
Inventor
Iii John A Lowe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO930222L publication Critical patent/NO930222L/no
Publication of NO930222D0 publication Critical patent/NO930222D0/no
Publication of NO302172B1 publication Critical patent/NO302172B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Soft Magnetic Materials (AREA)
  • Paper (AREA)
  • Control Of Electric Motors In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO930222A 1990-07-23 1993-01-22 Quinuclidin-derivater NO302172B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55744290A 1990-07-23 1990-07-23
PCT/US1991/003369 WO1992001688A1 (en) 1990-07-23 1991-05-14 Quinuclidine derivatives

Publications (3)

Publication Number Publication Date
NO930222L NO930222L (no) 1993-01-22
NO930222D0 true NO930222D0 (no) 1993-01-22
NO302172B1 NO302172B1 (no) 1998-02-02

Family

ID=24225412

Family Applications (1)

Application Number Title Priority Date Filing Date
NO930222A NO302172B1 (no) 1990-07-23 1993-01-22 Quinuclidin-derivater

Country Status (25)

Country Link
US (5) US5422354A (no)
EP (1) EP0540526B1 (no)
JP (1) JP2514137B2 (no)
CN (1) CN1058405A (no)
AT (1) ATE116317T1 (no)
AU (1) AU660416B2 (no)
BR (1) BR9106665A (no)
CA (1) CA2086434C (no)
DE (1) DE69106365T2 (no)
DK (1) DK0540526T3 (no)
ES (1) ES2065691T3 (no)
FI (1) FI114473B (no)
GR (1) GR3015144T3 (no)
HU (1) HUT62584A (no)
IE (1) IE65000B1 (no)
IL (1) IL98860A (no)
MX (1) MX9100308A (no)
MY (1) MY107157A (no)
NO (1) NO302172B1 (no)
NZ (1) NZ239063A (no)
PL (1) PL167568B1 (no)
PT (1) PT98393B (no)
WO (1) WO1992001688A1 (no)
YU (1) YU128091A (no)
ZA (1) ZA915727B (no)

Families Citing this family (76)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2086434C (en) * 1990-07-23 1998-09-22 John A. Lowe, Iii Quinuclidine derivatives
US5716965A (en) * 1991-05-22 1998-02-10 Pfizer Inc. Substituted 3-aminoquinuclidines
SK282203B6 (sk) * 1991-06-20 2001-12-03 Pfizer Inc. Fluoroalkoxybenzylamínové deriváty heterocyklov obsahujúcich dusík, spôsob ich prípravy, medziprodukty, spôsob prípravy medziproduktov, použitie a farmaceutický prostriedok
TW202432B (no) * 1991-06-21 1993-03-21 Pfizer
CA2118704C (en) * 1991-09-26 1997-01-21 John A. Lowe, Iii Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists
ES2111650T3 (es) * 1991-11-12 1998-03-16 Pfizer Derivados aciclicos de etilenodiamina como antagonistas de receptores de la sustancia p.
JP2757234B2 (ja) * 1992-05-18 1998-05-25 ファイザー インク． Ｐ物質拮抗薬としての架橋アザ二環式誘導体
JPH07506379A (ja) * 1992-08-04 1995-07-13 ファイザー・インコーポレーテッド 物質ｐ受容体アンタゴニストとしての３−ベンジルアミノ−２−フェニル−ピペリジン
AU4224993A (en) * 1992-08-19 1994-03-15 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles
PT675886E (pt) * 1992-12-10 2000-12-29 Pfizer Heterociclos nao aromaticos com substituintes aminometileno e sua utilizacao como antagonistas da substancia p
US5830854A (en) * 1992-12-14 1998-11-03 Merck Sharp & Dohme, Limited Method of treating cystic fibrosis using a tachykinin receptor antagonist
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EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
FR2725900B1 (fr) * 1994-10-21 1997-07-18 Sanofi Sa Utilisation d'antagonistes des recepteurs nk1 pour la preparation de medicaments a action cardioregulatrice
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UA105182C2 (ru) 2008-07-03 2014-04-25 Ньюрексон, Інк. Бензоксазины, бензотиазины и родственные соединения, которые имеют ингибирующую nos активность
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Family Cites Families (8)

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US2455949A (en) * 1947-06-02 1948-12-14 Parke Davis & Co Dialkylaminoalkyl benzahydryl ethers and salts thereof
US3560510A (en) * 1969-03-05 1971-02-02 Aldrich Chem Co Inc 2-benzhydrylquinuclidines
GB1527489A (en) * 1976-08-05 1978-10-04 Andreu Sa Dr Amine compound
US4246201A (en) * 1979-06-11 1981-01-20 Alfa Farmaceutici, S.P.A. Substituted N-(3-phenylthiopropyl)-3,3-diphenyl-propylamines possessing pharmacological activity
WO1990005525A1 (en) * 1988-11-23 1990-05-31 Pfizer Inc. Quinuclidine derivatives as substance p antagonists
UA41251C2 (uk) * 1990-01-04 2001-09-17 Пфайзер, Інк. Гідровані азотвмісні гетероциклічні сполуки, похідні піперидину, фармацевтична композиція та спосіб пригнічення активності речовини р в організмі
US5451586A (en) * 1990-06-01 1995-09-19 Pfizer Inc. 3-amino-2-aryl quinuclidines
CA2086434C (en) * 1990-07-23 1998-09-22 John A. Lowe, Iii Quinuclidine derivatives

Also Published As

Publication number Publication date
PT98393B (pt) 1999-01-29
CA2086434A1 (en) 1992-01-24
ES2065691T3 (es) 1995-02-16
ZA915727B (en) 1993-02-24
NO930222L (no) 1993-01-22
JP2514137B2 (ja) 1996-07-10
IE912560A1 (en) 1992-01-29
IL98860A0 (en) 1992-07-15
US5422354A (en) 1995-06-06
HU9300188D0 (en) 1993-04-28
US5641786A (en) 1997-06-24
EP0540526B1 (en) 1994-12-28
MX9100308A (es) 1992-02-28
US5854256A (en) 1998-12-29
US5698568A (en) 1997-12-16
PT98393A (pt) 1992-05-29
CA2086434C (en) 1998-09-22
BR9106665A (pt) 1993-06-08
GR3015144T3 (en) 1995-05-31
IE65000B1 (en) 1995-10-04
US5821248A (en) 1998-10-13
ATE116317T1 (de) 1995-01-15
NO302172B1 (no) 1998-02-02
YU128091A (sh) 1994-01-20
NZ239063A (en) 1995-09-26
FI930262L (fi) 1993-01-22
FI114473B (fi) 2004-10-29
MY107157A (en) 1995-09-30
DE69106365D1 (de) 1995-02-09
PL167568B1 (pl) 1995-09-30
IL98860A (en) 1995-11-27
CN1058405A (zh) 1992-02-05
EP0540526A1 (en) 1993-05-12
WO1992001688A1 (en) 1992-02-06
DE69106365T2 (de) 1995-05-04
DK0540526T3 (da) 1995-04-18
FI930262A0 (fi) 1993-01-22
AU7894891A (en) 1992-02-18
JPH05507687A (ja) 1993-11-04
AU660416B2 (en) 1995-06-29
HUT62584A (en) 1993-05-28

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