NO316119B1 - Imidasopyrimidiner og imidasopyridiner, farmasöytisk sammensetning inneholdende samme og anvendelse av samme for fremstilling av medikamentet - Google Patents
Imidasopyrimidiner og imidasopyridiner, farmasöytisk sammensetning inneholdende samme og anvendelse av samme for fremstilling av medikamentet Download PDFInfo
- Publication number
- NO316119B1 NO316119B1 NO19996483A NO996483A NO316119B1 NO 316119 B1 NO316119 B1 NO 316119B1 NO 19996483 A NO19996483 A NO 19996483A NO 996483 A NO996483 A NO 996483A NO 316119 B1 NO316119 B1 NO 316119B1
- Authority
- NO
- Norway
- Prior art keywords
- alkyl
- ethyl
- group
- substituted
- hexane
- Prior art date
Links
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- MMSLSKDMIZOHRX-WYDAWZGFSA-N α-helical crf(9-41) Chemical compound OC(=O)C[C@H](N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(N)=O MMSLSKDMIZOHRX-WYDAWZGFSA-N 0.000 description 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5162897P | 1997-07-03 | 1997-07-03 | |
| US8066598P | 1998-04-03 | 1998-04-03 | |
| PCT/US1998/013913 WO1999001454A1 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO996483D0 NO996483D0 (no) | 1999-12-27 |
| NO996483L NO996483L (no) | 2000-03-02 |
| NO316119B1 true NO316119B1 (no) | 2003-12-15 |
Family
ID=26729655
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19996483A NO316119B1 (no) | 1997-07-03 | 1999-12-27 | Imidasopyrimidiner og imidasopyridiner, farmasöytisk sammensetning inneholdende samme og anvendelse av samme for fremstilling av medikamentet |
Country Status (20)
| Country | Link |
|---|---|
| US (3) | US6143743A (pt) |
| EP (1) | EP0994877A1 (pt) |
| JP (1) | JP2002507996A (pt) |
| KR (1) | KR20010014431A (pt) |
| CN (1) | CN1268137A (pt) |
| AR (1) | AR016307A1 (pt) |
| AU (1) | AU746706B2 (pt) |
| BR (1) | BR9810508A (pt) |
| CA (1) | CA2294117A1 (pt) |
| EE (1) | EE04280B1 (pt) |
| HR (1) | HRP980375A2 (pt) |
| HU (1) | HUP0100179A3 (pt) |
| IL (1) | IL133800A0 (pt) |
| MY (1) | MY132871A (pt) |
| NO (1) | NO316119B1 (pt) |
| NZ (1) | NZ502642A (pt) |
| PL (1) | PL337888A1 (pt) |
| SK (1) | SK179899A3 (pt) |
| TW (1) | TW589309B (pt) |
| WO (1) | WO1999001454A1 (pt) |
Families Citing this family (76)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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| KR0151819B1 (ko) * | 1994-06-11 | 1998-10-15 | 강박광 | 신규의 피리딜 n-옥사이드로 치환된 피디딜이미다졸 유도체 및 그의 제조방법 |
| PL181895B1 (pl) * | 1994-06-16 | 2001-10-31 | Pfizer | Nowe pirazolo-i pirolopirydyny _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ _ PL PL PL PL |
| SE9402431D0 (sv) * | 1994-07-08 | 1994-07-08 | Astra Ab | New tablet formulation |
| SE504459C2 (sv) * | 1994-07-15 | 1997-02-17 | Astra Ab | Förfarande för framställning av substituerade sulfoxider |
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| WO1996019478A1 (en) * | 1994-12-19 | 1996-06-27 | Novartis Ag | 6'-substituted carbocyclic nucleosides |
| SE9500422D0 (sv) * | 1995-02-06 | 1995-02-06 | Astra Ab | New oral pharmaceutical dosage forms |
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| WO1997008150A1 (en) * | 1995-08-22 | 1997-03-06 | The Du Pont Merck Pharmaceutical Company | Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors |
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-
1998
- 1998-07-02 SK SK1798-99A patent/SK179899A3/sk unknown
- 1998-07-02 HR HR60/080,665A patent/HRP980375A2/hr not_active Application Discontinuation
- 1998-07-02 BR BR9810508-6A patent/BR9810508A/pt not_active IP Right Cessation
- 1998-07-02 PL PL98337888A patent/PL337888A1/xx unknown
- 1998-07-02 CN CN98808584A patent/CN1268137A/zh active Pending
- 1998-07-02 HU HU0100179A patent/HUP0100179A3/hu unknown
- 1998-07-02 KR KR1019997012619A patent/KR20010014431A/ko not_active Ceased
- 1998-07-02 CA CA002294117A patent/CA2294117A1/en not_active Abandoned
- 1998-07-02 MY MYPI98003027A patent/MY132871A/en unknown
- 1998-07-02 US US09/109,877 patent/US6143743A/en not_active Expired - Lifetime
- 1998-07-02 WO PCT/US1998/013913 patent/WO1999001454A1/en not_active Ceased
- 1998-07-02 TW TW087110857A patent/TW589309B/zh active
- 1998-07-02 NZ NZ502642A patent/NZ502642A/en unknown
- 1998-07-02 AU AU81819/98A patent/AU746706B2/en not_active Ceased
- 1998-07-02 EP EP98931795A patent/EP0994877A1/en not_active Withdrawn
- 1998-07-02 JP JP50744099A patent/JP2002507996A/ja active Pending
- 1998-07-02 EE EEP199900607A patent/EE04280B1/xx not_active IP Right Cessation
- 1998-07-02 IL IL13380098A patent/IL133800A0/xx unknown
- 1998-07-03 AR ARP980103234A patent/AR016307A1/es not_active Application Discontinuation
- 1998-12-10 US US09/208,778 patent/US6362180B1/en not_active Expired - Lifetime
-
1999
- 1999-12-27 NO NO19996483A patent/NO316119B1/no not_active IP Right Cessation
-
2001
- 2001-11-07 US US10/053,475 patent/US6642230B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| AU8181998A (en) | 1999-01-25 |
| EE9900607A (et) | 2000-08-15 |
| US6362180B1 (en) | 2002-03-26 |
| JP2002507996A (ja) | 2002-03-12 |
| US6642230B2 (en) | 2003-11-04 |
| BR9810508A (pt) | 2000-09-05 |
| HUP0100179A3 (en) | 2002-12-28 |
| US6143743A (en) | 2000-11-07 |
| CA2294117A1 (en) | 1999-01-14 |
| TW589309B (en) | 2004-06-01 |
| WO1999001454A1 (en) | 1999-01-14 |
| AU746706B2 (en) | 2002-05-02 |
| CN1268137A (zh) | 2000-09-27 |
| MY132871A (en) | 2007-10-31 |
| NO996483L (no) | 2000-03-02 |
| KR20010014431A (ko) | 2001-02-26 |
| US20030114468A1 (en) | 2003-06-19 |
| SK179899A3 (en) | 2001-12-03 |
| NO996483D0 (no) | 1999-12-27 |
| EP0994877A1 (en) | 2000-04-26 |
| HUP0100179A2 (hu) | 2001-11-28 |
| PL337888A1 (en) | 2000-09-11 |
| EE04280B1 (et) | 2004-04-15 |
| AR016307A1 (es) | 2001-07-04 |
| HRP980375A2 (en) | 1999-04-30 |
| NZ502642A (en) | 2002-06-28 |
| IL133800A0 (en) | 2001-04-30 |
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