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NO20084590L - Styryl pyridine derivatives and their use in binding and imaging of amyloid plaques - Google Patents

Styryl pyridine derivatives and their use in binding and imaging of amyloid plaques

Info

Publication number
NO20084590L
NO20084590L NO20084590A NO20084590A NO20084590L NO 20084590 L NO20084590 L NO 20084590L NO 20084590 A NO20084590 A NO 20084590A NO 20084590 A NO20084590 A NO 20084590A NO 20084590 L NO20084590 L NO 20084590L
Authority
NO
Norway
Prior art keywords
imaging
binding
pyridine derivatives
amyloid plaques
compounds
Prior art date
Application number
NO20084590A
Other languages
Norwegian (no)
Other versions
NO342090B1 (en
Inventor
Hank F Kung
Mei-Ping Kung
Original Assignee
Univ Pennsylvania
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Pennsylvania filed Critical Univ Pennsylvania
Publication of NO20084590L publication Critical patent/NO20084590L/en
Publication of NO342090B1 publication Critical patent/NO342090B1/en

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/92Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
    • C07D211/94Oxygen atom, e.g. piperidine N-oxide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62Oxygen or sulfur atoms
    • C07D213/63One oxygen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0455Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Physics & Mathematics (AREA)
  • Epidemiology (AREA)
  • Optics & Photonics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Denne oppfinnelsen vedrører en fremgangsmåte for avbilding av amyloidavsetninger, og styrylpyridinforbindel-ser og fremgangsmåter for fremstilling av radioaktivt merkede styrylpyridin-forbindelser som kan anvendes ved avbilding av amyloidavsetninger. Denne oppfinnelsen vedrører også forbindelser og fremgangsmåter for fremstiling av forbindelser for inhibering av aggre-gasjonen av amyloidproteiner for å danne amyloidavsetninger, og en fremgangsmåte for avlevering av et terapeutisk middel til amyloidavsetninger,This invention relates to a method for imaging amyloid deposits, and to styrylpyridine compounds and methods for preparing radiolabelled styrylpyridine compounds which may be used in imaging amyloid deposits. This invention also relates to compounds and methods for preparing compounds for inhibiting the aggregation of amyloid proteins to form amyloid deposits, and to a method of delivering a therapeutic agent to amyloid deposits.

NO20084590A 2006-03-30 2008-10-29 Styryl pyridine derivatives and their use for bonding and imaging of amyloid plaques NO342090B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78715606P 2006-03-30 2006-03-30
PCT/US2007/007400 WO2007126733A2 (en) 2006-03-30 2007-03-26 Styrylpyridine derivatives and their use for binding and imaging amyloid plaques

Publications (2)

Publication Number Publication Date
NO20084590L true NO20084590L (en) 2008-12-29
NO342090B1 NO342090B1 (en) 2018-03-19

Family

ID=38326579

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20084590A NO342090B1 (en) 2006-03-30 2008-10-29 Styryl pyridine derivatives and their use for bonding and imaging of amyloid plaques
NO2018030C NO2018030I1 (en) 2006-03-30 2018-09-11 Florbetapir (18F)

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2018030C NO2018030I1 (en) 2006-03-30 2018-09-11 Florbetapir (18F)

Country Status (34)

Country Link
US (3) US7687052B2 (en)
EP (3) EP2363391A1 (en)
JP (1) JP5290954B2 (en)
KR (1) KR101376807B1 (en)
CN (1) CN101522624B (en)
AT (1) ATE539060T1 (en)
AU (1) AU2007243712B2 (en)
BR (1) BRPI0710225B1 (en)
CA (1) CA2644530C (en)
CR (1) CR10329A (en)
CY (3) CY1113048T1 (en)
DK (2) DK1999109T3 (en)
EA (1) EA017898B1 (en)
EC (1) ECSP088783A (en)
ES (2) ES2378785T3 (en)
FR (1) FR13C0034I2 (en)
GT (1) GT200800201A (en)
HR (2) HRP20120135T1 (en)
HU (2) HUE032660T2 (en)
IL (1) IL193567A (en)
LT (1) LT2363392T (en)
LU (1) LU92232I2 (en)
MX (1) MX2008012527A (en)
NO (2) NO342090B1 (en)
NZ (1) NZ570887A (en)
PL (2) PL1999109T3 (en)
PT (2) PT1999109E (en)
RS (2) RS52222B (en)
SG (1) SG173338A1 (en)
SI (2) SI2363392T1 (en)
TW (1) TWI399366B (en)
UA (1) UA97802C2 (en)
WO (1) WO2007126733A2 (en)
ZA (1) ZA200807955B (en)

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Publication number Publication date
CN101522624A (en) 2009-09-02
CA2644530A1 (en) 2007-11-08
EP2363392B1 (en) 2017-05-03
CY2013024I2 (en) 2015-11-04
US8506929B2 (en) 2013-08-13
HRP20120135T1 (en) 2012-03-31
TWI399366B (en) 2013-06-21
ECSP088783A (en) 2008-10-31
TW200838852A (en) 2008-10-01
EA200870389A1 (en) 2009-04-28
US20130129624A1 (en) 2013-05-23
CA2644530C (en) 2015-05-19
ES2378785T3 (en) 2012-04-17
JP5290954B2 (en) 2013-09-18
JP2009532349A (en) 2009-09-10
CN101522624B (en) 2013-11-06
SG173338A1 (en) 2011-08-29
SI2363392T1 (en) 2017-09-29
ZA200807955B (en) 2012-11-28
US20080038195A1 (en) 2008-02-14
LU92232I9 (en) 2019-01-15
EP1999109A2 (en) 2008-12-10
CY2013024I1 (en) 2015-11-04
AU2007243712B2 (en) 2013-01-10
PT1999109E (en) 2012-03-16
WO2007126733A2 (en) 2007-11-08
KR20080106564A (en) 2008-12-08
WO2007126733A3 (en) 2008-03-06
IL193567A (en) 2014-03-31
EA017898B1 (en) 2013-04-30
ES2628882T3 (en) 2017-08-04
ATE539060T1 (en) 2012-01-15
FR13C0034I1 (en) 2013-08-09
NZ570887A (en) 2011-05-27
GT200800201A (en) 2009-08-20
IL193567A0 (en) 2009-05-04
LT2363392T (en) 2017-07-25
FR13C0034I2 (en) 2014-03-07
SI1999109T1 (en) 2012-04-30
US7687052B2 (en) 2010-03-30
CY1113048T1 (en) 2015-11-04
HUE032660T2 (en) 2017-10-30
HRP20170857T1 (en) 2017-12-01
US8840866B2 (en) 2014-09-23
EP2363391A1 (en) 2011-09-07
DK2363392T3 (en) 2017-07-03
UA97802C2 (en) 2012-03-26
KR101376807B1 (en) 2014-03-20
EP1999109B1 (en) 2011-12-28
EP2363392A1 (en) 2011-09-07
BRPI0710225A2 (en) 2011-08-02
US20090123369A1 (en) 2009-05-14
DK1999109T3 (en) 2012-04-02
MX2008012527A (en) 2008-10-14
CR10329A (en) 2008-10-29
RS56171B1 (en) 2017-11-30
RS52222B (en) 2012-10-31
HUS1300028I1 (en) 2017-08-28
AU2007243712A1 (en) 2007-11-08
PL2363392T3 (en) 2017-10-31
BRPI0710225B1 (en) 2021-07-13
PL1999109T3 (en) 2012-05-31
PT2363392T (en) 2017-06-15
NO2018030I1 (en) 2018-09-11
CY1119048T1 (en) 2018-01-10
LU92232I2 (en) 2013-08-26
NO342090B1 (en) 2018-03-19

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