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NO20081523L - Fremstilling og anvendelse av tetrahydropyrrolo(3,2-C)Pyridin-4-on-derivater for behandling av fedme, psykiatriske og neurologiske forstyrrelser - Google Patents

Fremstilling og anvendelse av tetrahydropyrrolo(3,2-C)Pyridin-4-on-derivater for behandling av fedme, psykiatriske og neurologiske forstyrrelser

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Publication number
NO20081523L
NO20081523L NO20081523A NO20081523A NO20081523L NO 20081523 L NO20081523 L NO 20081523L NO 20081523 A NO20081523 A NO 20081523A NO 20081523 A NO20081523 A NO 20081523A NO 20081523 L NO20081523 L NO 20081523L
Authority
NO
Norway
Prior art keywords
pyridin
tetrahydropyrrolo
psychiatric
obesity
preparation
Prior art date
Application number
NO20081523A
Other languages
English (en)
Inventor
Leifeng Cheng
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37781800&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20081523(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20081523L publication Critical patent/NO20081523L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Abstract

Foreliggende oppfinnelse angår 4,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-on- og 4,5-dihydropyrrolo[3,2-c]pyridin-4-on-forbindelser med formel I og fremgangsmåter for fremstilling av slike forbindelser, anvendelse av dem ved behandling av fedme, psykiatriske og nevrologiske lidelser, metoder for deres terapeutiske anvendelse og farmasøytiske preparater inneholdende dem.
NO20081523A 2005-10-06 2008-03-28 Fremstilling og anvendelse av tetrahydropyrrolo(3,2-C)Pyridin-4-on-derivater for behandling av fedme, psykiatriske og neurologiske forstyrrelser NO20081523L (no)

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PCT/GB2006/003695 WO2007039740A2 (en) 2005-10-06 2006-10-05 Preparation and use of tetrahydropyrrolo [3, 2-c] pyridin-4-one derivatives for treatment of obesity, psychiatric and neurological disorders

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US7875626B2 (en) 2011-01-25
ATE440099T1 (de) 2009-09-15
TW200730525A (en) 2007-08-16
AU2006298530A1 (en) 2007-04-12
DE602006008641D1 (de) 2009-10-01
EP1937679B1 (en) 2009-08-19
US20080009513A1 (en) 2008-01-10
EP1937679A2 (en) 2008-07-02
ES2329616T3 (es) 2009-11-27
ZA200802946B (en) 2009-03-25
RU2008109185A (ru) 2009-11-20
US7576095B2 (en) 2009-08-18
HK1122808A1 (en) 2009-05-29
RU2415856C2 (ru) 2011-04-10
ECSP088413A (es) 2008-05-30
US20080312269A1 (en) 2008-12-18
CA2624495A1 (en) 2007-04-12
CN101277957A (zh) 2008-10-01
AR056560A1 (es) 2007-10-10
IL190025A0 (en) 2008-08-07
AU2006298530B2 (en) 2009-10-29
WO2007039740A2 (en) 2007-04-12
UY29838A1 (es) 2007-05-31
WO2007039740A3 (en) 2007-05-31
JP4277062B2 (ja) 2009-06-10
JP2009504722A (ja) 2009-02-05
KR20080058456A (ko) 2008-06-25

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