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NO20076425L - Fremgangsmater for behandling av drug-resistent cancer - Google Patents

Fremgangsmater for behandling av drug-resistent cancer

Info

Publication number
NO20076425L
NO20076425L NO20076425A NO20076425A NO20076425L NO 20076425 L NO20076425 L NO 20076425L NO 20076425 A NO20076425 A NO 20076425A NO 20076425 A NO20076425 A NO 20076425A NO 20076425 L NO20076425 L NO 20076425L
Authority
NO
Norway
Prior art keywords
compound
resistant cancer
methods
treating drug
tautomer
Prior art date
Application number
NO20076425A
Other languages
English (en)
Inventor
Glenn C Michelson
Vivien W Chan
Carla C Heise
Marion Wiesmann
Timothy D Dawes
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20076425L publication Critical patent/NO20076425L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4425—Pyridinium derivatives, e.g. pralidoxime, pyridostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

En fremgangsmåte for behandling av medikamentresistent cancer inkluderer: administrere til en pasient med behov derav, en forbindelse av formel 1, en tautomer av forbindelsen, et salt av forbindelsen, et salt av tautomeren, en blanding derav, eller en farmasøytisk sammensetning omfattende forbindelsen, tautomeren, saltet av forbindelsen, saltet av tautomeren eller blandingen, hvor pasienten er en cancerpasient med medikamentresistent cancer, hvor forbindelsen av formel I er som definert i søknaden.
NO20076425A 2005-05-13 2007-12-13 Fremgangsmater for behandling av drug-resistent cancer NO20076425L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68072205P 2005-05-13 2005-05-13
PCT/US2006/017922 WO2006124413A2 (en) 2005-05-13 2006-05-10 Methods for treating drug resistant cancer

Publications (1)

Publication Number Publication Date
NO20076425L true NO20076425L (no) 2008-01-30

Family

ID=37431829

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20076425A NO20076425L (no) 2005-05-13 2007-12-13 Fremgangsmater for behandling av drug-resistent cancer

Country Status (22)

Country Link
US (1) US8299081B2 (no)
EP (1) EP1885187B1 (no)
JP (2) JP5344910B2 (no)
KR (1) KR101319122B1 (no)
CN (1) CN101222850B (no)
AU (1) AU2006247803B2 (no)
BR (1) BRPI0610360A2 (no)
CA (1) CA2608171C (no)
DK (1) DK1885187T3 (no)
ES (1) ES2440799T3 (no)
IL (1) IL187327A (no)
MA (1) MA29543B1 (no)
MX (1) MX2007014206A (no)
NO (1) NO20076425L (no)
NZ (1) NZ564144A (no)
PL (1) PL1885187T3 (no)
PT (1) PT1885187E (no)
RU (1) RU2426539C2 (no)
SI (1) SI1885187T1 (no)
TN (1) TNSN07419A1 (no)
WO (1) WO2006124413A2 (no)
ZA (1) ZA200709620B (no)

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CN104093402A (zh) * 2012-01-31 2014-10-08 诺华股份有限公司 Rtk抑制剂与抗雌激素的组合及其治疗癌症的应用
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Also Published As

Publication number Publication date
RU2007145932A (ru) 2009-06-20
JP2013173787A (ja) 2013-09-05
KR20080033902A (ko) 2008-04-17
HK1110477A1 (en) 2008-07-18
TNSN07419A1 (en) 2009-03-17
IL187327A0 (en) 2008-04-13
KR101319122B1 (ko) 2013-10-23
WO2006124413A3 (en) 2007-06-07
JP2008540543A (ja) 2008-11-20
AU2006247803A1 (en) 2006-11-23
CA2608171C (en) 2014-02-04
RU2426539C2 (ru) 2011-08-20
US8299081B2 (en) 2012-10-30
EP1885187A4 (en) 2009-05-13
JP5344910B2 (ja) 2013-11-20
DK1885187T3 (da) 2013-12-09
MX2007014206A (es) 2008-02-07
SI1885187T1 (sl) 2013-12-31
BRPI0610360A2 (pt) 2010-06-15
AU2006247803B2 (en) 2011-12-22
US20090215793A1 (en) 2009-08-27
IL187327A (en) 2015-05-31
CA2608171A1 (en) 2006-11-23
ZA200709620B (en) 2008-10-29
EP1885187B1 (en) 2013-09-25
PL1885187T3 (pl) 2014-03-31
MA29543B1 (fr) 2008-06-02
CN101222850B (zh) 2012-10-03
EP1885187A2 (en) 2008-02-13
CN101222850A (zh) 2008-07-16
WO2006124413A2 (en) 2006-11-23
NZ564144A (en) 2009-11-27
ES2440799T3 (es) 2014-01-30
PT1885187E (pt) 2013-12-16

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