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NO20075258L - Vannfrie krystallinske former av N-(1-(2-etoksyetyl)-5-(N-etyl-N-metylamino)-7-(4-metylpyndin-2-yl-amino)-1H-pyrazolo(4,3-d)pyrimidin-3-carbonyl)metansulfonamid - Google Patents

Vannfrie krystallinske former av N-(1-(2-etoksyetyl)-5-(N-etyl-N-metylamino)-7-(4-metylpyndin-2-yl-amino)-1H-pyrazolo(4,3-d)pyrimidin-3-carbonyl)metansulfonamid

Info

Publication number
NO20075258L
NO20075258L NO20075258A NO20075258A NO20075258L NO 20075258 L NO20075258 L NO 20075258L NO 20075258 A NO20075258 A NO 20075258A NO 20075258 A NO20075258 A NO 20075258A NO 20075258 L NO20075258 L NO 20075258L
Authority
NO
Norway
Prior art keywords
methanesulfonamide
methylpyridin
pyrazolo
ethoxyethyl
methylamino
Prior art date
Application number
NO20075258A
Other languages
English (en)
Inventor
David Andrew Entwistle
Peter Wallance Marshall
Stefan Colin Taylor
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO20075258L publication Critical patent/NO20075258L/no

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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Abstract

Det beskrives (1) vannfrie krystallinske former av N-[1-(2-etoksyetyl)-5-(N-etyl-N-metylamino)-7-(4-metylpyridin-2-yl-amino)-lH-pyrazolo[4,3-d]pyrimidin-3-karbonyl]-metansulfonamid, (2) farmasøytiske sammensetninger omfattende minst en slik form, (3) fremgangsmåter for behandling av fosfodiesterase 5-medierte tilstander ved anvendelse av minst en slik form, og (4) fremgangsmåte for fremstilling av slike former.
NO20075258A 2005-05-12 2007-10-12 Vannfrie krystallinske former av N-(1-(2-etoksyetyl)-5-(N-etyl-N-metylamino)-7-(4-metylpyndin-2-yl-amino)-1H-pyrazolo(4,3-d)pyrimidin-3-carbonyl)metansulfonamid NO20075258L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68044505P 2005-05-12 2005-05-12
US68171105P 2005-05-17 2005-05-17
PCT/IB2006/001233 WO2006120552A2 (en) 2005-05-12 2006-05-03 ANHYDROUS CRYSTALLINE FORMS OF N-[1-(2-ETHOXYETHYL)-5-(N-ETHYL-N-METHYLAMINO)-7-(4-METHYLPYRIDIN-2-yl-AMINO)-1H-PYRAZOLO[4,3-d]PYRIMIDINE-3-CARBONYL]METHANESULFONAMIDE

Publications (1)

Publication Number Publication Date
NO20075258L true NO20075258L (no) 2007-11-15

Family

ID=37106941

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20075258A NO20075258L (no) 2005-05-12 2007-10-12 Vannfrie krystallinske former av N-(1-(2-etoksyetyl)-5-(N-etyl-N-metylamino)-7-(4-metylpyndin-2-yl-amino)-1H-pyrazolo(4,3-d)pyrimidin-3-carbonyl)metansulfonamid

Country Status (23)

Country Link
US (3) US8227475B2 (no)
EP (1) EP1881985B1 (no)
JP (2) JP4271695B2 (no)
KR (1) KR100939890B1 (no)
AT (1) ATE493413T1 (no)
AU (1) AU2006245416B2 (no)
BR (1) BRPI0609225A2 (no)
CA (1) CA2608018C (no)
CR (1) CR9505A (no)
CY (1) CY1111171T1 (no)
DE (1) DE602006019231D1 (no)
DK (1) DK1881985T3 (no)
EA (1) EA012577B1 (no)
IL (1) IL186693A (no)
MA (1) MA29447B1 (no)
MX (1) MX2007013215A (no)
NO (1) NO20075258L (no)
NZ (1) NZ564187A (no)
PL (1) PL1881985T3 (no)
PT (1) PT1881985E (no)
TN (1) TNSN07414A1 (no)
TW (1) TWI380986B (no)
WO (1) WO2006120552A2 (no)

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KR20080004593A (ko) 2008-01-09
AU2006245416A1 (en) 2006-11-16
IL186693A0 (en) 2008-02-09
JP4996631B2 (ja) 2012-08-08
ATE493413T1 (de) 2011-01-15
JP2006316058A (ja) 2006-11-24
TNSN07414A1 (fr) 2009-03-17
WO2006120552A3 (en) 2007-01-18
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CA2608018A1 (en) 2006-11-16
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BRPI0609225A2 (pt) 2010-03-09
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