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NO20061543L - Modulators of ATPBinding Cassette Transportm - Google Patents

Modulators of ATPBinding Cassette Transportm

Info

Publication number
NO20061543L
NO20061543L NO20061543A NO20061543A NO20061543L NO 20061543 L NO20061543 L NO 20061543L NO 20061543 A NO20061543 A NO 20061543A NO 20061543 A NO20061543 A NO 20061543A NO 20061543 L NO20061543 L NO 20061543L
Authority
NO
Norway
Prior art keywords
modulators
transportm
cassette
atpbinding
atpbinding cassette
Prior art date
Application number
NO20061543A
Other languages
English (en)
Inventor
Mark T Miller
Sara S Hadida Ruah
Ashavini K Singh
Thomas Cleveland
Lewis R Makings
Matthew Hamilton
Peter D J Grootenhuis
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20061543L publication Critical patent/NO20061543L/no

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D295/145—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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Abstract

Den foreliggende oppfinnelsen vedrører modulatorer av ATP-bindingskassett- ("ABC") transportere eller fragmenter derav, inkludert CF-transmembranregulator ("CFTR"), sammensetninger derav og tilhørende fremgangsmåter. Den foreliggende oppfinnelsen vedrører også fremgangsmåter for å behandle ABC-transportermedierte sykdommer anvendende slike modulatorer.
NO20061543A 2003-09-06 2006-04-05 Modulators of ATPBinding Cassette Transportm NO20061543L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50044403P 2003-09-06 2003-09-06
PCT/US2004/029206 WO2005026137A2 (en) 2003-09-06 2004-09-07 Modulators of atp-binding cassette transporters

Publications (1)

Publication Number Publication Date
NO20061543L true NO20061543L (no) 2006-06-06

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ID=34312193

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20061543A NO20061543L (no) 2003-09-06 2006-04-05 Modulators of ATPBinding Cassette Transportm

Country Status (13)

Country Link
US (6) US7973169B2 (no)
EP (1) EP1664006A2 (no)
JP (1) JP2007504255A (no)
KR (1) KR20060088537A (no)
CN (1) CN1898221A (no)
AU (1) AU2004272599A1 (no)
CA (1) CA2537841A1 (no)
IL (1) IL174128A0 (no)
MX (1) MXPA06002567A (no)
NO (1) NO20061543L (no)
RU (1) RU2006111093A (no)
WO (1) WO2005026137A2 (no)
ZA (1) ZA200602755B (no)

Cited By (1)

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NO338017B1 (no) * 2003-12-26 2016-07-18 Kyowa Hakko Kirin Co Ltd Tiazolderivater, farmasøytiske preparater inneholdende slike, og anvendelse derav

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