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NO20055591D0 - Antivirale fosfonatanaloger - Google Patents

Antivirale fosfonatanaloger

Info

Publication number
NO20055591D0
NO20055591D0 NO20055591A NO20055591A NO20055591D0 NO 20055591 D0 NO20055591 D0 NO 20055591D0 NO 20055591 A NO20055591 A NO 20055591A NO 20055591 A NO20055591 A NO 20055591A NO 20055591 D0 NO20055591 D0 NO 20055591D0
Authority
NO
Norway
Prior art keywords
compounds
phosphonate analogues
antiviral phosphonate
antiviral
analogues
Prior art date
Application number
NO20055591A
Other languages
English (en)
Other versions
NO338306B1 (no
NO20055591L (no
Inventor
David Oare
Aesop Cho
William John Watkins
William A Lee
Alan X Huang
Choung U Kim
Constantine G Boojamra
Lee S Chong
James M Chen
Xiaowu Chen
Maria Fardis
Haolun Jin
Richard L Mackman
Hyung-Jung Pyun
Sundaramoorthi Swaminathan
Jennifer R Zhang
Carina E Cannizzaro
Thorsten A Kirschberg
Ralph F Hirschmann
Christopher P Lee
Original Assignee
Usprasad Vidya K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Usprasad Vidya K filed Critical Usprasad Vidya K
Publication of NO20055591D0 publication Critical patent/NO20055591D0/no
Publication of NO20055591L publication Critical patent/NO20055591L/no
Publication of NO338306B1 publication Critical patent/NO338306B1/no

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    • C07F9/02—Phosphorus compounds
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C07F9/65616—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system having three or more than three double bonds between ring members or between ring members and non-ring members, e.g. purine or analogs
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
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    • A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
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