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NO20052733D0 - C-6 modifiserte indazolylpyrrolotriaziner - Google Patents

C-6 modifiserte indazolylpyrrolotriaziner

Info

Publication number
NO20052733D0
NO20052733D0 NO20052733A NO20052733A NO20052733D0 NO 20052733 D0 NO20052733 D0 NO 20052733D0 NO 20052733 A NO20052733 A NO 20052733A NO 20052733 A NO20052733 A NO 20052733A NO 20052733 D0 NO20052733 D0 NO 20052733D0
Authority
NO
Norway
Prior art keywords
indazolylpyrrolotriazines
modified
modified indazolylpyrrolotriazines
Prior art date
Application number
NO20052733A
Other languages
English (en)
Other versions
NO20052733L (no
Inventor
Gregory D Vite
John F Kadow
Ashvinikumar Gavai
Harold Mastalerz
Brian E Fink
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20052733D0 publication Critical patent/NO20052733D0/no
Publication of NO20052733L publication Critical patent/NO20052733L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
NO20052733A 2002-12-13 2005-06-07 C-6 modifiserte indazolylpyrrolotriaziner NO20052733L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43319002P 2002-12-13 2002-12-13
PCT/US2003/039542 WO2004054514A2 (en) 2002-12-13 2003-12-12 C-6 modified indazolylpyrrolotriazines

Publications (2)

Publication Number Publication Date
NO20052733D0 true NO20052733D0 (no) 2005-06-07
NO20052733L NO20052733L (no) 2005-07-07

Family

ID=32595133

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20052733A NO20052733L (no) 2002-12-13 2005-06-07 C-6 modifiserte indazolylpyrrolotriaziner

Country Status (27)

Country Link
US (2) US6916815B2 (no)
EP (1) EP1569937B1 (no)
JP (1) JP4511367B2 (no)
KR (1) KR101073801B1 (no)
CN (2) CN1726216A (no)
AR (1) AR042450A1 (no)
AT (1) ATE534648T1 (no)
AU (1) AU2003300877B2 (no)
BR (1) BR0316755A (no)
CA (1) CA2509650C (no)
CO (1) CO5570660A2 (no)
DK (1) DK1569937T3 (no)
ES (1) ES2374393T3 (no)
HR (1) HRP20050535A2 (no)
IS (1) IS7890A (no)
MX (1) MXPA05006164A (no)
NO (1) NO20052733L (no)
NZ (1) NZ540338A (no)
PE (1) PE20040805A1 (no)
PL (1) PL377517A1 (no)
PT (1) PT1569937E (no)
RS (1) RS20050441A (no)
RU (1) RU2356903C2 (no)
TW (1) TW200420565A (no)
UA (1) UA80591C2 (no)
WO (1) WO2004054514A2 (no)
ZA (1) ZA200504507B (no)

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TW200306841A (en) 2002-04-23 2003-12-01 Bristol Myers Squibb Co Aryl ketone pyrrolo-triazine compounds useful as kinase inhibitors
TWI329112B (en) * 2002-07-19 2010-08-21 Bristol Myers Squibb Co Novel inhibitors of kinases
US6921769B2 (en) 2002-08-23 2005-07-26 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
US7649006B2 (en) 2002-08-23 2010-01-19 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
PT1506203E (pt) 2002-08-23 2007-04-30 Sloan Kettering Inst Cancer Síntese de epotilonas, seus intermediários, seus análogos e suas utilizações
TW200420565A (en) * 2002-12-13 2004-10-16 Bristol Myers Squibb Co C-6 modified indazolylpyrrolotriazines
JP2006516653A (ja) 2003-02-05 2006-07-06 ブリストル−マイヤーズ スクイブ カンパニー キナーゼ阻害剤ピロロトリアジンの製造方法
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US7151176B2 (en) * 2004-10-21 2006-12-19 Bristol-Myers Squibb Company Pyrrolotriazine compounds
WO2006111524A2 (en) * 2005-04-18 2006-10-26 Novo Nordisk A/S Il-21 variants
US7405213B2 (en) * 2005-07-01 2008-07-29 Bristol-Myers Squibb Company Pyrrolotriazine compounds useful as kinase inhibitors and methods of treating kinase-associated conditions therewith
US7402582B2 (en) * 2005-07-01 2008-07-22 Bristol-Myers Squibb Company Pyrrolotriazine compounds useful as kinase inhibitors and methods of treating kinase-associated conditions therewith
US7880004B2 (en) 2005-09-15 2011-02-01 Bristol-Myers Squibb Company Met kinase inhibitors
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US7514435B2 (en) * 2005-11-18 2009-04-07 Bristol-Myers Squibb Company Pyrrolotriazine kinase inhibitors
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US8063208B2 (en) 2006-02-16 2011-11-22 Bristol-Myers Squibb Company Crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol
KR20080107408A (ko) 2006-03-07 2008-12-10 브리스톨-마이어스 스큅 컴퍼니 키나제 억제제로서 유용한 피롤로트리아진 아닐린 전구약물화합물
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CN105026399B (zh) * 2013-03-11 2017-06-23 百时美施贵宝公司 作为钾离子通道抑制剂的吡咯并三嗪类化合物
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Also Published As

Publication number Publication date
UA80591C2 (en) 2007-10-10
CA2509650C (en) 2007-10-30
US7148220B2 (en) 2006-12-12
CO5570660A2 (es) 2005-10-31
IS7890A (is) 2005-06-10
CN1726216A (zh) 2006-01-25
CA2509650A1 (en) 2004-07-01
JP4511367B2 (ja) 2010-07-28
HRP20050535A2 (en) 2005-12-31
EP1569937A2 (en) 2005-09-07
PE20040805A1 (es) 2004-11-20
ZA200504507B (en) 2006-08-30
NO20052733L (no) 2005-07-07
US6916815B2 (en) 2005-07-12
KR20050084242A (ko) 2005-08-26
AR042450A1 (es) 2005-06-22
US20050222153A1 (en) 2005-10-06
US20040142931A1 (en) 2004-07-22
EP1569937B1 (en) 2011-11-23
PL377517A1 (pl) 2006-02-06
AU2003300877A1 (en) 2004-07-09
BR0316755A (pt) 2005-10-25
MXPA05006164A (es) 2005-08-26
AU2003300877B2 (en) 2010-02-18
EP1569937A4 (en) 2007-08-08
RU2356903C2 (ru) 2009-05-27
TW200420565A (en) 2004-10-16
WO2004054514A2 (en) 2004-07-01
WO2004054514A3 (en) 2004-10-07
RU2005120650A (ru) 2006-01-20
NZ540338A (en) 2008-05-30
ES2374393T3 (es) 2012-02-16
KR101073801B1 (ko) 2011-10-13
RS20050441A (sr) 2007-04-10
ATE534648T1 (de) 2011-12-15
PT1569937E (pt) 2012-01-04
DK1569937T3 (da) 2012-01-02
JP2006509826A (ja) 2006-03-23
CN101723948A (zh) 2010-06-09

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