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NO20044808L - Heterosykliske sulfonamider som er hepatitt C virus inhibitorer - Google Patents

Heterosykliske sulfonamider som er hepatitt C virus inhibitorer

Info

Publication number
NO20044808L
NO20044808L NO20044808A NO20044808A NO20044808L NO 20044808 L NO20044808 L NO 20044808L NO 20044808 A NO20044808 A NO 20044808A NO 20044808 A NO20044808 A NO 20044808A NO 20044808 L NO20044808 L NO 20044808L
Authority
NO
Norway
Prior art keywords
hepatitis
virus inhibitors
heterocyclic sulfonamides
analogs
compounds
Prior art date
Application number
NO20044808A
Other languages
English (en)
Inventor
Jeffrey Allen Campbell
Andrew Charles Good
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20044808L publication Critical patent/NO20044808L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0808—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C07K5/06165—Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biophysics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

Det beskrives tripeptidforbindelser, blandinger som inneholder slike forbindelser og fremgangsmåter for anvendelse av slike forbindelser til behandlingen av hepatitt C virus (HCV-infeksjon). Særlig beskrives nye tripeptidanaloger, farmasøytiske blandinger som inneholder slike analoger og fremgangsmåter for bruk av disse analogene ved behandlingen av HCV-infeksjon.
NO20044808A 2002-05-20 2004-11-04 Heterosykliske sulfonamider som er hepatitt C virus inhibitorer NO20044808L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38210402P 2002-05-20 2002-05-20
PCT/US2003/015786 WO2003099316A1 (en) 2002-05-20 2003-05-20 Heterocyclicsulfonamide hepatitis c virus inhibitors

Publications (1)

Publication Number Publication Date
NO20044808L true NO20044808L (no) 2004-12-17

Family

ID=29584359

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20044808A NO20044808L (no) 2002-05-20 2004-11-04 Heterosykliske sulfonamider som er hepatitt C virus inhibitorer

Country Status (11)

Country Link
US (1) US6869964B2 (no)
EP (1) EP1506000B9 (no)
JP (1) JP4312711B2 (no)
AT (1) ATE481106T1 (no)
AU (1) AU2003248535A1 (no)
DE (1) DE60334205D1 (no)
ES (1) ES2350201T3 (no)
IS (1) IS7532A (no)
NO (1) NO20044808L (no)
PL (1) PL211889B1 (no)
WO (1) WO2003099316A1 (no)

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