[go: up one dir, main page]

NO20043424L - Tricykliske 2-pyrimidon forbindelser nyttige som HIV revers transkriptase inhibitorer - Google Patents

Tricykliske 2-pyrimidon forbindelser nyttige som HIV revers transkriptase inhibitorer

Info

Publication number
NO20043424L
NO20043424L NO20043424A NO20043424A NO20043424L NO 20043424 L NO20043424 L NO 20043424L NO 20043424 A NO20043424 A NO 20043424A NO 20043424 A NO20043424 A NO 20043424A NO 20043424 L NO20043424 L NO 20043424L
Authority
NO
Norway
Prior art keywords
tricyclic
reverse transcriptase
compounds useful
transcriptase inhibitors
hiv reverse
Prior art date
Application number
NO20043424A
Other languages
English (en)
Inventor
Christine M Tarby
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20043424L publication Critical patent/NO20043424L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20043424A 2002-01-18 2004-08-17 Tricykliske 2-pyrimidon forbindelser nyttige som HIV revers transkriptase inhibitorer NO20043424L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34964102P 2002-01-18 2002-01-18
PCT/US2003/001604 WO2003062238A1 (en) 2002-01-18 2003-01-16 Tricyclic 2-pyrimidone compounds useful as hiv reverse transcriptase inhibitors

Publications (1)

Publication Number Publication Date
NO20043424L true NO20043424L (no) 2004-08-18

Family

ID=27613304

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20043424A NO20043424L (no) 2002-01-18 2004-08-17 Tricykliske 2-pyrimidon forbindelser nyttige som HIV revers transkriptase inhibitorer

Country Status (21)

Country Link
US (2) US6844340B2 (no)
EP (1) EP1474424A4 (no)
JP (1) JP2005519910A (no)
KR (1) KR20040077735A (no)
CN (1) CN1642954A (no)
AR (1) AR038164A1 (no)
BR (1) BR0306927A (no)
CA (1) CA2473420A1 (no)
CO (1) CO5590961A2 (no)
HR (1) HRP20040643A2 (no)
IL (1) IL162743A0 (no)
IS (1) IS7341A (no)
MX (1) MXPA04006948A (no)
NO (1) NO20043424L (no)
PE (1) PE20030987A1 (no)
PL (1) PL371418A1 (no)
RU (1) RU2004125151A (no)
TW (1) TW200306192A (no)
WO (1) WO2003062238A1 (no)
YU (1) YU62504A (no)
ZA (1) ZA200405139B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7169932B2 (en) 2001-06-11 2007-01-30 Pfizer Inc. HIV protease inhibitors, compositions containing the same, their pharmaceutical uses, material for their synthesis
HN2002000136A (es) 2001-06-11 2003-07-31 Basf Ag Inhibidores de la proteasa del virus hiv, compuestos que contienen a los mismos, sus usos farmaceuticos y los materiales para su sintesis
US7094909B2 (en) 2001-06-11 2006-08-22 Agouron Pharmaceuticals, Inc. HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
TW200306192A (en) * 2002-01-18 2003-11-16 Bristol Myers Squibb Co Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors
AR039540A1 (es) * 2002-05-13 2005-02-23 Tibotec Pharm Ltd Compuestos microbicidas con contenido de pirimidina o triazina
ES2598404T3 (es) * 2003-02-07 2017-01-27 Janssen Pharmaceutica Nv Derivados de pirimidina para la prevención de infección por el VIH
WO2008004100A2 (en) 2006-07-05 2008-01-10 Pfizer Products Inc. Therapeutic compounds
US20080119552A1 (en) * 2006-11-17 2008-05-22 Novus International Inc. Matrix-embedded compositions having organic acids and fatty acids
BRPI0906809A2 (pt) 2008-01-25 2015-07-14 High Point Pharmaceuticals Llc Compostos tricíclicos como moduladores da síntese do tnf-(alfa) e como inibidores da pde4.
AU2010334958B2 (en) 2009-12-23 2015-02-05 Katholieke Universiteit Leuven Novel antiviral compounds
CA2817165A1 (en) 2010-11-15 2012-05-24 Patrick Chaltin Novel antiviral compounds
CA2817896A1 (en) 2010-11-15 2012-05-24 Viiv Healthcare Uk Limited Inhibitors of hiv replication
CN103130787B (zh) * 2011-11-24 2015-06-10 南开大学 嘧啶酮酰胺类化合物及其制备方法、抗hiv活性和抗tmv活性
GB201509663D0 (en) * 2015-06-03 2015-07-15 Johnson Matthey Plc Benzo(h)quinoline ligands and complexes thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6593337B1 (en) * 1999-10-19 2003-07-15 Bristol-Myers Squibb Pharma Company Tricyclic compounds useful as HIV reverse transcriptase inhibitors
US6596729B2 (en) 2000-07-20 2003-07-22 Bristol-Myers Squibb Company Tricyclic-2-pyridone compounds useful as HIV reverse transcriptase inhibitors
TW200306192A (en) * 2002-01-18 2003-11-16 Bristol Myers Squibb Co Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors

Also Published As

Publication number Publication date
TW200306192A (en) 2003-11-16
CA2473420A1 (en) 2003-07-31
IL162743A0 (en) 2005-11-20
MXPA04006948A (es) 2004-12-06
US7186830B2 (en) 2007-03-06
US6844340B2 (en) 2005-01-18
US20040266778A1 (en) 2004-12-30
IS7341A (is) 2004-06-30
KR20040077735A (ko) 2004-09-06
BR0306927A (pt) 2004-11-09
CN1642954A (zh) 2005-07-20
US20030162800A1 (en) 2003-08-28
HRP20040643A2 (en) 2005-04-30
RU2004125151A (ru) 2006-02-20
ZA200405139B (en) 2006-02-22
WO2003062238A1 (en) 2003-07-31
JP2005519910A (ja) 2005-07-07
EP1474424A4 (en) 2005-12-28
PL371418A1 (en) 2005-06-13
EP1474424A1 (en) 2004-11-10
YU62504A (sh) 2006-08-17
AR038164A1 (es) 2004-12-29
CO5590961A2 (es) 2005-12-30
PE20030987A1 (es) 2003-11-15

Similar Documents

Publication Publication Date Title
NO20021835L (no) Tricykliske forbindelser nyttige som HIV-reverse transkriptase inhibitorer
NO20033857D0 (no) Benzofenoner som inhibitorer av revers transkriptase
NO20021042D0 (no) Benzofenoner som inhibitorer av revers transkriptase
NO20161397A1 (no) Ikke-nukleosidbaserte revers-transkriptase-inhibitorer
ATE425138T1 (de) N-phenyl-phenylacetamid-nichtnukleosidinhibitor n reverser transkriptase
NO20043004L (no) 4-oksokinolin forbindelse og anvendelse derav som HIV-integraseinhibitor
DK1749011T3 (da) Bicykliske heterocykler som HIV-integrasehæmmere
DK2039685T3 (da) Heterobicycliske forbindelser som P38-inhibitorer
NO20055680D0 (no) Heksahydropyridoisokinoliner som DPP-IV-inhibitorer
DK1586319T3 (da) Thiadiazolidinoner som GSK-3-inhibitorer
DK1699797T3 (da) Pyrrolotriazinforbindelser som kinasehæmmere
DK1544199T3 (da) Nitrogenholdig kondenseret ringforbindelse og anvendelse deraf som HIV-integraseinhibitor
NO20052921D0 (no) Fenylsubstituerte piperidinforbindelser for anvendelse som PPAR aktivatorer
NO20043793L (no) Nikotinamidderivater anvendelige som PDE4 inhibitorer
NO20044256L (no) Makrosykliske forbindelser som kan anvendes som farmasoytika
NO20044654L (no) Piperidinoylpiperidiner som 5-HTIF-agonister
NO20043424L (no) Tricykliske 2-pyrimidon forbindelser nyttige som HIV revers transkriptase inhibitorer
PL378556A1 (pl) Nienukleozydowe inhibitory odwrotnej transkryptazy
NO20044104L (no) Ikke-nukleoside reverstranskriptase-inhibitorer
AU2003243765A1 (en) 2,4-disubstituted-pyridine n-oxides useful as hiv reverse transcriptase inhibitors
DK1294720T3 (da) Non-nukleosid revers transkriptase-inhibitorer
DK1651641T3 (da) Nicotinamidderivater egnede som PDE4 inhibitorer
MXPA03009482A (es) Compuestos triciclicos utiles como inhibidores de la transcriptasa inversa del virus de inmunodeficiencia humana (vih).
DK1373261T3 (da) Cyklopropaheterocykler som non-nukleotid revers transkriptase-hæmmer
NO20030248D0 (no) Tricykliske pyridonforbindelser anvendelige som HIV revers- transkriptase-inhibitorer

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application