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NO20020260D0 - 11<beta>-aryl-17,17-spirotiolansubstituerte steroider - Google Patents

11<beta>-aryl-17,17-spirotiolansubstituerte steroider

Info

Publication number
NO20020260D0
NO20020260D0 NO20020260A NO20020260A NO20020260D0 NO 20020260 D0 NO20020260 D0 NO 20020260D0 NO 20020260 A NO20020260 A NO 20020260A NO 20020260 A NO20020260 A NO 20020260A NO 20020260 D0 NO20020260 D0 NO 20020260D0
Authority
NO
Norway
Prior art keywords
spirothiolane
beta
aryl
substituted steroids
compounds
Prior art date
Application number
NO20020260A
Other languages
English (en)
Other versions
NO321524B1 (no
NO20020260L (no
Inventor
Edgar C Cook
Rupa S Shetty
John A Kepler
David Y-W Lee
Original Assignee
Res Triangle Inst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Res Triangle Inst filed Critical Res Triangle Inst
Publication of NO20020260D0 publication Critical patent/NO20020260D0/no
Publication of NO20020260L publication Critical patent/NO20020260L/no
Publication of NO321524B1 publication Critical patent/NO321524B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J33/00Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20020260A 1999-07-21 2002-01-17 11<beta>-aryl-17,17-spirotiolansubstituerte steroider, anvendelse derav samt fremgangsmate for fremstilling av et C17-cyklisk spirotiolan av en steroidforbindelse. NO321524B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/357,923 US6043235A (en) 1999-07-21 1999-07-21 11β-aryl-17, 17-spirothiolane-substituted steroids
PCT/US2000/019537 WO2001007462A1 (en) 1999-07-21 2000-07-20 11β-ARYL-17,17-SPIROTHIOLANE-SUBSTITUTED STEROIDS

Publications (3)

Publication Number Publication Date
NO20020260D0 true NO20020260D0 (no) 2002-01-17
NO20020260L NO20020260L (no) 2002-03-14
NO321524B1 NO321524B1 (no) 2006-05-15

Family

ID=23407590

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20020260A NO321524B1 (no) 1999-07-21 2002-01-17 11<beta>-aryl-17,17-spirotiolansubstituerte steroider, anvendelse derav samt fremgangsmate for fremstilling av et C17-cyklisk spirotiolan av en steroidforbindelse.

Country Status (14)

Country Link
US (1) US6043235A (no)
EP (1) EP1196428B1 (no)
JP (1) JP4768181B2 (no)
KR (1) KR100616025B1 (no)
AT (1) ATE277071T1 (no)
AU (1) AU774472B2 (no)
CA (1) CA2379995C (no)
DE (1) DE60014096T2 (no)
DK (1) DK1196428T3 (no)
ES (1) ES2228584T3 (no)
HK (1) HK1044542B (no)
NO (1) NO321524B1 (no)
PT (1) PT1196428E (no)
WO (1) WO2001007462A1 (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6262042B1 (en) 1998-05-29 2001-07-17 Research Triangle Institute 17β-amino and hydroxylamino-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties
CN103893211A (zh) 2006-03-07 2014-07-02 吉塔·什罗夫 包含人胚胎干细胞和其衍生物的组合物、其使用方法和制备方法
KR200451979Y1 (ko) * 2008-04-11 2011-01-24 정종오 회전형 광고장치
DE102009034367A1 (de) * 2009-07-20 2011-01-27 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-benzyliden-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten
DE102009034526A1 (de) * 2009-07-21 2011-02-10 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-ethinylphenyl-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2344286A1 (fr) * 1976-03-16 1977-10-14 Roussel Uclaf Nouveaux derives 17-spirosultines, les g-hydroxy acides correspondants, leur procede de preparation et leur application comme medicament
FR2374037A1 (fr) * 1976-10-27 1978-07-13 Roussel Uclaf Nouveaux derives steroides 17-spirosultines les g-hydroxy acides correspondants, leur procede de preparation et leur application comme medicament
ZA929315B (en) * 1991-12-20 1993-05-24 Akzo Nv 17-spirofuran-3'-ylidene steroids.
IL115659A (en) * 1994-10-27 2000-06-01 Akzo Nobel Nv Steroids with a 17-spiromethylene lactone or lactol group process for their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
ES2228584T3 (es) 2005-04-16
HK1044542B (en) 2005-02-25
US6043235A (en) 2000-03-28
DE60014096T2 (de) 2005-10-06
DE60014096D1 (de) 2004-10-28
DK1196428T3 (da) 2005-01-24
HK1044542A1 (en) 2002-10-25
PT1196428E (pt) 2005-02-28
AU6220000A (en) 2001-02-13
CA2379995A1 (en) 2001-02-01
KR100616025B1 (ko) 2006-08-30
CA2379995C (en) 2008-10-14
JP2003531815A (ja) 2003-10-28
EP1196428A4 (en) 2002-10-16
EP1196428A1 (en) 2002-04-17
ATE277071T1 (de) 2004-10-15
EP1196428B1 (en) 2004-09-22
WO2001007462A1 (en) 2001-02-01
JP4768181B2 (ja) 2011-09-07
NO321524B1 (no) 2006-05-15
KR20020092893A (ko) 2002-12-12
NO20020260L (no) 2002-03-14
AU774472B2 (en) 2004-07-01

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Legal Events

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