NO20014603D0 - Tienopyrimidinforbindelser, deres fremstilling og anvendelse - Google Patents

Tienopyrimidinforbindelser, deres fremstilling og anvendelse

Info

Publication number: NO20014603D0
Authority: NO; Norway
Prior art keywords: tienopyrimidine; compounds; preparation; tienopyrimidine compounds
Prior art date: 1999-03-24

Application number

NO20014603A

Other languages

English (en)

Other versions

NO20014603L (no

Inventor

Shuichi Furuya

Nobuhiro Suzuki

Nobuo Choh

Yoshi Nara

Original Assignee

Takeda Chemical Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-03-24

Filing date

2001-09-21

Publication date

2001-09-21

2001-09-21 Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd

2001-09-21 Publication of NO20014603D0 publication Critical patent/NO20014603D0/no

2001-11-26 Publication of NO20014603L publication Critical patent/NO20014603L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Reproductive Health (AREA)
Diabetes (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

NO20014603A 1999-03-24 2001-09-21 Tienopyrimidinforbindelser, deres fremstilling og anvendelse NO20014603L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP7937199		1999-03-24
JP2000018019		2000-01-25
PCT/JP2000/001777 WO2000056739A1 (en)	1999-03-24	2000-03-23	Thienopyrimidine compounds, their production and use

Publications (2)

Publication Number	Publication Date
NO20014603D0 true NO20014603D0 (no)	2001-09-21
NO20014603L NO20014603L (no)	2001-11-26

Family

ID=26420391

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20014603A NO20014603L (no)	1999-03-24	2001-09-21	Tienopyrimidinforbindelser, deres fremstilling og anvendelse

Country Status (28)

Country	Link
US (1)	US6340686B1 (no)
EP (1)	EP1163244B1 (no)
JP (1)	JP3240293B2 (no)
KR (2)	KR100533483B1 (no)
CN (1)	CN1349536A (no)
AR (1)	AR023152A1 (no)
AT (1)	ATE261449T1 (no)
AU (1)	AU764019B2 (no)
BR (1)	BR0009297A (no)
CA (1)	CA2368108C (no)
CZ (1)	CZ294747B6 (no)
DE (1)	DE60008862T2 (no)
DK (1)	DK1163244T3 (no)
ES (1)	ES2212992T3 (no)
HK (1)	HK1042495B (no)
HU (1)	HUP0200550A3 (no)
ID (1)	ID30393A (no)
IL (1)	IL145549A (no)
MX (1)	MXPA01009566A (no)
MY (1)	MY124726A (no)
NO (1)	NO20014603L (no)
NZ (1)	NZ514737A (no)
OA (1)	OA11920A (no)
PL (1)	PL351202A1 (no)
PT (1)	PT1163244E (no)
SK (1)	SK13552001A3 (no)
TW (1)	TWI225863B (no)
WO (1)	WO2000056739A1 (no)

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US6828415B2 (en) *	1993-02-19	2004-12-07	Zentaris Gmbh	Oligopeptide lyophilisate, their preparation and use
EP1266898A4 (en) *	2000-02-29	2003-05-21	Takeda Chemical Industries Ltd	PROCESSES FOR PRODUCING THIENOPYRAMIDINE DERIVATIVES
EP1393747A4 (en) *	2000-04-13	2004-03-03	Takeda Chemical Industries Ltd	AGENT FOR PREVENTION / TREATMENT OF ALZHEIMER DISEASE
EP1291023A1 (en) *	2000-06-14	2003-03-12	Takeda Chemical Industries, Ltd.	Sustained release compositions
EP1319409A4 (en) *	2000-09-22	2006-05-03	Takeda Pharmaceutical	SOLID PREPARATIONS
WO2002043766A1 (en) *	2000-11-29	2002-06-06	Takeda Chemical Industries, Ltd.	Medicinal compositions and process for producing the same
WO2002047722A1 (en) *	2000-12-15	2002-06-20	Takeda Chemical Industries, Ltd.	Medicinal compositions of nonpeptidyl gonadotropin-releasing hormone agonist or antagonist, process for producing the same and use thereof
WO2002078669A1 (fr) *	2001-03-30	2002-10-10	Takeda Chemical Industries, Ltd.	Solutions medicinales
AU2002324586B2 (en)	2001-08-02	2008-04-24	Neurocrine Biosciences, Inc.	1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
US6939883B2 (en)	2001-08-02	2005-09-06	Neurocrine Biosciences, Inc.	Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
EP1411941A2 (en)	2001-08-02	2004-04-28	Neurocrine Biosciences, Inc.	Pyridinone and pyridazinone derivatives as gonadotropin-releasing hormone receptor antagonists
JP2005500356A (ja) *	2001-08-02	2005-01-06	ニューロクラインバイオサイエンシーズ，インコーポレイテッド	ゴナドトロピン放出ホルモンレセプターアンタゴニスト
CA2455235A1 (en)	2001-08-02	2003-02-13	Joseph Pontillo	1,2,4-triazin-3,5-diones as gonadotropin-releasing hormone receptor (gnrh) antagonists
WO2003064429A1 (en)	2002-01-30	2003-08-07	Takeda Chemical Industries, Ltd.	Thienopyrimidines, process for preparing the same and use thereof
EP1495768A4 (en)	2002-04-12	2007-12-05	Takeda Pharmaceutical	MEANS FOR THE PREVENTION / TREATMENT OF HITZEWALLUNGEN
US7317010B2 (en) *	2002-08-21	2008-01-08	Astrazeneca Ab	Thieno-pyrrole compounds as antagonists of gonadotropin releasing hormone
CA2514407C (en)	2003-01-29	2012-01-03	Takeda Pharmaceutical Company Limited	Thienopyrimidine compounds and use thereof
GB0307777D0 (en)	2003-04-04	2003-05-07	Medical Res Council	Conjugate compounds
US20060083017A1 (en) *	2004-10-18	2006-04-20	Bwt Propety, Inc.	Solid-state lighting apparatus for navigational aids
RU2419435C2 (ru) *	2005-07-22	2011-05-27	Такеда Фармасьютикал Компани Лимитед	Предотвращающий преждевременную овуляцию агент
US20110172249A1 (en)	2008-09-03	2011-07-14	Takeda Pharmaceutical Company Limted	Method for improving absorbability of preparation, and preparation having improved absorbability
CN105732649B (zh) *	2012-02-28	2019-02-05	株式会社蒂奥姆生物	促性腺激素释放激素受体拮抗剂、其制备方法和包含该拮抗剂的药物组合物
PL3415517T3 (pl)	2012-09-28	2022-07-04	Takeda Pharmaceutical Company Limited	Postać krystaliczna 1-(4-1-(2,6-difluorobenzylo)-5-dimetyloaminometylo-3-(6-metoksypirydazyn-3-ylo)-2,4-diokso-1,2,3,4-tetrahydrotieno(2,3-d)-pirymidyn-6-ylo)fenylo)-3-metoksymocznika
PL4233847T3 (pl)	2015-02-26	2024-11-18	Takeda Pharmaceutical Company Limited	Tabletka zawierająca pochodną metoksymocznika i cząstki mannitolu
SI3518932T1 (sl)	2016-09-30	2025-03-31	Takeda Pharmaceutical Company Limited	Zdravljenje raka prostate
CN110312512B (zh)	2016-09-30	2023-05-09	梦欧文科学有限责任公司	用于治疗子宫肌瘤和子宫内膜异位症的方法
KR101973074B1 (ko) *	2018-11-30	2019-04-26	주식회사 티움바이오	퓨로피리미딘 화합물의 염 및 결정형, 및 이를 포함하는 약학적 조성물
WO2021018105A1 (en) *	2019-07-29	2021-02-04	Sunshine Lake Pharma Co., Ltd.	Substituted pyrimidinedione compounds and uses thereof
JP2022551316A (ja)	2019-10-10	2022-12-08	ミオバントサイエンシズゲーエムベーハー	Ｎ－（４－（１－（２，６－ジフルオロベンジル）－５－（（ジメチルアミノ）メチル）－３－（６－メトキシ－３－ピリダジニル）－２，４－ジオキソ－１，２，３，４－テトラヒドロチエノ［２，３－ｄ］ピリミジン－６－イル）フェニル）－Ｎ’－メトキシ尿素の結晶形
CN111574534B (zh) *	2020-05-25	2021-06-04	东莞市东阳光新药研发有限公司	苯基取代的噻吩并[2,3-d]嘧啶-2,4(1H,3H)-二酮类化合物及其用途
CN111909168B (zh) *	2020-07-31	2022-02-01	广东东阳光药业有限公司	含氮杂环基取代的嘧啶二酮类化合物及其用途
CN111925379B (zh) *	2020-07-31	2022-02-15	广东东阳光药业有限公司	含氮杂芳基取代的嘧啶二酮类化合物及其用途
CN112047957B (zh) *	2020-09-09	2022-02-01	广东东阳光药业有限公司	取代的嘧啶二酮类化合物及其用途
CN113754679B (zh) *	2020-09-09	2023-04-07	广东东阳光药业有限公司	取代的嘧啶二酮类化合物及其用途
CN113429423B (zh) *	2020-12-30	2022-05-17	上海博志研新药物技术有限公司	瑞卢戈利中间体及其制备方法
CN115260211B (zh) *	2021-04-29	2024-02-06	长春金赛药业有限责任公司	含噻吩稠环类衍生物、药物组合物及其制备方法和应用
CN113717149A (zh) *	2021-09-29	2021-11-30	成都伊诺达博医药科技有限公司	一种瑞卢戈利关键中间体及其制备方法

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UY23948A1 (es) *	1995-02-08	2001-10-25	Takeda Chemical Industries Ltd	Derivados de anillos condensados de tiofeno su producción y uso.
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EP0816316A4 (en) *	1995-03-10	1999-06-02	Nitto Chemical Industry Co Ltd	Process for producing 1,2-ethanediol derivatives

2000
- 2000-03-08 TW TW089104127A patent/TWI225863B/zh not_active IP Right Cessation
- 2000-03-21 MY MYPI20001112 patent/MY124726A/en unknown
- 2000-03-23 SK SK1355-2001A patent/SK13552001A3/sk unknown
- 2000-03-23 DE DE60008862T patent/DE60008862T2/de not_active Expired - Lifetime
- 2000-03-23 MX MXPA01009566A patent/MXPA01009566A/es active IP Right Grant
- 2000-03-23 ES ES00911308T patent/ES2212992T3/es not_active Expired - Lifetime
- 2000-03-23 KR KR10-2000-7011511A patent/KR100533483B1/ko not_active Expired - Fee Related
- 2000-03-23 BR BR0009297-5A patent/BR0009297A/pt not_active IP Right Cessation
- 2000-03-23 ID IDW00200102298A patent/ID30393A/id unknown
- 2000-03-23 EP EP00911308A patent/EP1163244B1/en not_active Expired - Lifetime
- 2000-03-23 PL PL00351202A patent/PL351202A1/xx not_active Application Discontinuation
- 2000-03-23 KR KR10-2000-7011508A patent/KR100370981B1/ko not_active Expired - Fee Related
- 2000-03-23 CZ CZ20013419A patent/CZ294747B6/cs not_active IP Right Cessation
- 2000-03-23 NZ NZ514737A patent/NZ514737A/en unknown
- 2000-03-23 IL IL14554900A patent/IL145549A/xx not_active IP Right Cessation
- 2000-03-23 WO PCT/JP2000/001777 patent/WO2000056739A1/en not_active Ceased
- 2000-03-23 JP JP2000087051A patent/JP3240293B2/ja not_active Expired - Fee Related
- 2000-03-23 DK DK00911308T patent/DK1163244T3/da active
- 2000-03-23 OA OA1200100243A patent/OA11920A/en unknown
- 2000-03-23 PT PT00911308T patent/PT1163244E/pt unknown
- 2000-03-23 HU HU0200550A patent/HUP0200550A3/hu unknown
- 2000-03-23 AT AT00911308T patent/ATE261449T1/de not_active IP Right Cessation
- 2000-03-23 HK HK02104325.6A patent/HK1042495B/en not_active IP Right Cessation
- 2000-03-23 CN CN00807210A patent/CN1349536A/zh active Pending
- 2000-03-23 AU AU33262/00A patent/AU764019B2/en not_active Ceased
- 2000-03-23 CA CA002368108A patent/CA2368108C/en not_active Expired - Fee Related
- 2000-03-24 AR ARP000101320A patent/AR023152A1/es not_active Application Discontinuation
- 2000-05-16 US US09/571,215 patent/US6340686B1/en not_active Expired - Lifetime
2001
- 2001-09-21 NO NO20014603A patent/NO20014603L/no unknown

Also Published As

Publication number	Publication date
MXPA01009566A (es)	2002-05-14
MY124726A (en)	2006-06-30
CZ20013419A3 (cs)	2002-02-13
CZ294747B6 (cs)	2005-03-16
HK1042495A1 (en)	2002-08-16
US6340686B1 (en)	2002-01-22
SK13552001A3 (sk)	2002-03-05
KR100370981B1 (ko)	2003-02-06
CA2368108C (en)	2009-12-22
JP3240293B2 (ja)	2001-12-17
KR20010015920A (ko)	2001-02-26
NO20014603L (no)	2001-11-26
BR0009297A (pt)	2001-12-18
IL145549A (en)	2005-11-20
WO2000056739A1 (en)	2000-09-28
ES2212992T3 (es)	2004-08-16
CA2368108A1 (en)	2000-09-28
PL351202A1 (en)	2003-03-24
AU3326200A (en)	2000-10-09
EP1163244A1 (en)	2001-12-19
ID30393A (id)	2001-11-29
DK1163244T3 (da)	2004-07-12
IL145549A0 (en)	2002-06-30
JP2001278884A (ja)	2001-10-10
NZ514737A (en)	2003-10-31
TWI225863B (en)	2005-01-01
DE60008862D1 (de)	2004-04-15
ATE261449T1 (de)	2004-03-15
DE60008862T2 (de)	2005-01-27
OA11920A (en)	2006-04-12
HUP0200550A3 (en)	2004-07-28
CN1349536A (zh)	2002-05-15
KR20010090430A (ko)	2001-10-18
EP1163244B1 (en)	2004-03-10
KR100533483B1 (ko)	2005-12-05
HUP0200550A2 (en)	2002-06-29
HK1042495B (en)	2004-10-08
AR023152A1 (es)	2002-09-04
PT1163244E (pt)	2004-07-30
AU764019B2 (en)	2003-08-07

Publication	Publication Date	Title
NO20015156L (no)	2001-12-18	5-pyridyl-1,3-azolforbindelser, deres fremstilling og anvendelse
NO20014603L (no)	2001-11-26	Tienopyrimidinforbindelser, deres fremstilling og anvendelse
NO20021449L (no)	2002-05-07	Substituerte 2-tio-3,5-dicyano-4-aryl-6-aminopyridiner og deres anvendelse
NO20024742D0 (no)	2002-10-02	Heterocykliske forbindelser, deres fremstilling og anvendelse
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DK1161434T3 (da)	2003-05-26	Pyridopyranoazepinderivater, deres fremstilling og terapeutiske anvendelse
NO20031838D0 (no)	2003-04-24	Benzokazinonderivater, deres fremstilling og anvendelse
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NO20024107L (no)	2002-09-27	Tienopyridin derivater, deres fremstilling og anvendelse
NO20006479D0 (no)	2000-12-19	Tienopyridinforbindelser, deres fremstilling og anvendelse
NO20025209L (no)	2002-10-30	Cyklipostiner, deres fremstilling og anvendelse
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NO996156L (no)	2000-06-15	Substituerte cykloheptener, deres fremstilling og anvendelse
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NO20011921L (no)	2001-10-29	Sulfidoamidokarboksylsyre, deres fremstilling og anvendelse
DK1177196T3 (da)	2004-06-21	Heteroaryldiazabicycloalkaner, deres fremstilling og anvendelse