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NI201200025A - Heterociclos microbicidas - Google Patents

Heterociclos microbicidas

Info

Publication number
NI201200025A
NI201200025A NI201200025A NI201200025A NI201200025A NI 201200025 A NI201200025 A NI 201200025A NI 201200025 A NI201200025 A NI 201200025A NI 201200025 A NI201200025 A NI 201200025A NI 201200025 A NI201200025 A NI 201200025A
Authority
NI
Nicaragua
Prior art keywords
phenyl
alkyl
pyrazolyl
imidazolyl
haloalkyl
Prior art date
Application number
NI201200025A
Other languages
English (en)
Inventor
Sulzer-Mosse Sarah
Lamberth Clemens
Stephan Respondek Mathias
Quaranta Laura
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of NI201200025A publication Critical patent/NI201200025A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención trata acerca de compuestos heterocíclicos de fórmula I los cuales tienen actividad microbicida, en particular actividad fungicida así como acerca de métodos de utilización de los compuestos de fórmula I para controlar microbios: en donde A es X - C ( R10 R11 ) - C ( =O ) - , x - C ( R12 R13 ) - C ( =S ) - , x - O - C (=O) - , x - O - C ( = S) - , x - N ( R14 ) - C ( =O ) - , x - N ( R15 ) - C ( =S ) - , x - C ( R16R17 ) - SO2 - o x - N = C (R30) - , en cada caso x representa en enlace que está conectado a R1; T es CR18 o N; Y1, Y2, Y3, y Y4 son independientemente CR19 o N; Q es O o S; n es 1 o 2; p es 1 o 2, con la condición de que cuando n es 2, p es 1. R1 es fenilo, piridilo, imidazolilo, o pirazolilo; en donde cada uno de fenilo, piridilo, imidazolilo y pirazolilo están sustituidos opcionalmente con entre 1 y 3 sustituyentes escogidos independientemente entre alquilo C1 - C4, haloalquilo C1 - C4, halógeno, ciano, hidroxi y amino; R2, R3, R4, R5, R6, R7, R10, R11, R12, R13, R16, R17, R18, R19 y R30 son, cada uno independientemente, hidrógeno, halógeno, ciano, alquilo C1 - C4, o haloalquilo C1 - C4; R8, R14 y R15 son, cada uno independientemente, hidrógeno o alquilo C1 - C4; y R9 es fenilo, bencilo o el grupo (a).
NI201200025A 2009-08-12 2012-02-08 Heterociclos microbicidas NI201200025A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09167741 2009-08-12

Publications (1)

Publication Number Publication Date
NI201200025A true NI201200025A (es) 2012-10-29

Family

ID=42683487

Family Applications (1)

Application Number Title Priority Date Filing Date
NI201200025A NI201200025A (es) 2009-08-12 2012-02-08 Heterociclos microbicidas

Country Status (33)

Country Link
US (2) US8367844B2 (es)
EP (1) EP2464630B1 (es)
JP (1) JP5778674B2 (es)
KR (1) KR101750027B1 (es)
CN (1) CN102471277B (es)
AP (1) AP3383A (es)
AR (1) AR077835A1 (es)
AU (1) AU2010283767B2 (es)
BR (1) BR112012003124A2 (es)
CA (1) CA2768636C (es)
CL (1) CL2012000339A1 (es)
CO (1) CO6612179A2 (es)
CR (1) CR20120064A (es)
EA (1) EA021137B1 (es)
ES (1) ES2588330T3 (es)
GE (1) GEP20146113B (es)
HN (1) HN2012000308A (es)
HR (1) HRP20160951T1 (es)
HU (1) HUE029097T2 (es)
IL (1) IL217645A (es)
JO (1) JO3140B1 (es)
MX (1) MX2012001689A (es)
MY (1) MY157410A (es)
NI (1) NI201200025A (es)
NZ (1) NZ597503A (es)
PL (1) PL2464630T3 (es)
PT (1) PT2464630T (es)
SA (1) SA110310646B1 (es)
TW (1) TWI488849B (es)
UA (1) UA107938C2 (es)
UY (1) UY32840A (es)
WO (1) WO2011018415A2 (es)
ZA (1) ZA201200368B (es)

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US20120122928A1 (en) 2010-08-11 2012-05-17 Bayer Cropscience Ag Heteroarylpiperidine and -Piperazine Derivatives as Fungicides
US8759527B2 (en) 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
JP5918773B2 (ja) 2010-10-27 2016-05-18 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺菌剤としてのヘテロアリールピペリジンおよびヘテロアリールピペラジン誘導体
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NZ629795A (en) 2012-02-02 2016-06-24 Actelion Pharmaceuticals Ltd 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives
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EP2801575A1 (en) 2013-05-07 2014-11-12 Bayer CropScience AG Heteroaryldihydropyridine derivatives as fungicides
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AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
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KR102605762B1 (ko) 2016-02-08 2023-11-27 고완 크롭 프로텍션 리미티드 살균성 조성물
CN108602765B (zh) 2016-02-08 2022-05-03 高文有限公司 1,2-苯二甲醇化合物的制造方法
WO2017197240A1 (en) * 2016-05-12 2017-11-16 The Regents Of The University Of Michigan Ash1l inhibitors and methods of treatment therewith
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CN114380802B (zh) * 2022-01-07 2023-11-17 贵州大学 一类含咔唑基咪唑盐类化合物及其制备方法和应用

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Also Published As

Publication number Publication date
CR20120064A (es) 2012-03-22
CN102471277A (zh) 2012-05-23
AU2010283767A1 (en) 2012-02-23
JP2013501745A (ja) 2013-01-17
TWI488849B (zh) 2015-06-21
GEP20146113B (en) 2014-06-25
HN2012000308A (es) 2015-01-05
CO6612179A2 (es) 2013-02-01
WO2011018415A2 (en) 2011-02-17
EP2464630A2 (en) 2012-06-20
US8367844B2 (en) 2013-02-05
KR20120048010A (ko) 2012-05-14
JP5778674B2 (ja) 2015-09-16
UA107938C2 (en) 2015-03-10
MX2012001689A (es) 2012-02-22
CN102471277B (zh) 2015-05-06
AP2012006152A0 (en) 2012-04-30
ZA201200368B (en) 2012-09-26
US20120142698A1 (en) 2012-06-07
WO2011018415A3 (en) 2011-08-18
TW201114755A (en) 2011-05-01
JO3140B1 (ar) 2017-09-20
SA110310646B1 (ar) 2013-10-03
AU2010283767B2 (en) 2015-04-09
EP2464630B1 (en) 2016-05-25
ES2588330T3 (es) 2016-11-02
AR077835A1 (es) 2011-09-28
CA2768636A1 (en) 2011-02-17
IL217645A (en) 2015-03-31
AP3383A (en) 2015-07-31
US20130144064A1 (en) 2013-06-06
UY32840A (es) 2011-03-31
EA021137B1 (ru) 2015-04-30
CA2768636C (en) 2017-06-13
BR112012003124A2 (pt) 2020-08-25
CL2012000339A1 (es) 2012-10-12
NZ597503A (en) 2013-11-29
PT2464630T (pt) 2016-07-14
EA201200259A1 (ru) 2012-09-28
MY157410A (en) 2016-06-15
HRP20160951T1 (hr) 2016-10-07
KR101750027B1 (ko) 2017-06-22
HUE029097T2 (en) 2017-02-28
PL2464630T3 (pl) 2016-12-30

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