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MXPA06000416A - Amidas azaheterociclicas novedosas utiles para tratar el dolor. - Google Patents

Amidas azaheterociclicas novedosas utiles para tratar el dolor.

Info

Publication number
MXPA06000416A
MXPA06000416A MXPA06000416A MXPA06000416A MXPA06000416A MX PA06000416 A MXPA06000416 A MX PA06000416A MX PA06000416 A MXPA06000416 A MX PA06000416A MX PA06000416 A MXPA06000416 A MX PA06000416A MX PA06000416 A MXPA06000416 A MX PA06000416A
Authority
MX
Mexico
Prior art keywords
treating pain
amides useful
azaheterocyclic
novel
compounds
Prior art date
Application number
MXPA06000416A
Other languages
English (en)
Inventor
Robert G Schmidt
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of MXPA06000416A publication Critical patent/MXPA06000416A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

La presente invencion se refiere a compuestos de la formula (I-VII) (I), o una sal farmaceutica aceptable o profarmaco del mismo, en la cual A, L, R6, R7 y R8 se definen en la presente. La presente invencion tambien se refiere a metodos para tratar dolor usando aquellos compuestos y composiciones farmaceuticas que incluye estos compuestos.
MXPA06000416A 2003-07-11 2004-07-09 Amidas azaheterociclicas novedosas utiles para tratar el dolor. MXPA06000416A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/618,016 US20050009841A1 (en) 2003-07-11 2003-07-11 Novel amides useful for treating pain
PCT/US2004/021836 WO2005007642A2 (en) 2003-07-11 2004-07-09 Novel azaheterocyclic amides useful for treating pain

Publications (1)

Publication Number Publication Date
MXPA06000416A true MXPA06000416A (es) 2006-04-05

Family

ID=33565052

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA06000416A MXPA06000416A (es) 2003-07-11 2004-07-09 Amidas azaheterociclicas novedosas utiles para tratar el dolor.

Country Status (13)

Country Link
US (1) US20050009841A1 (es)
EP (1) EP1646621A2 (es)
JP (1) JP2007523865A (es)
KR (1) KR20060034282A (es)
CN (2) CN101434596A (es)
AU (1) AU2004257220A1 (es)
BR (1) BRPI0412438A (es)
CA (1) CA2532057A1 (es)
IL (1) IL172985A0 (es)
MX (1) MXPA06000416A (es)
TW (1) TW200510372A (es)
WO (1) WO2005007642A2 (es)
ZA (1) ZA200600228B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2281823A3 (en) * 2003-05-20 2011-09-07 Ajinomoto Co., Inc. Anti-inflammatory and analgesic piperidine derivatives
MY142655A (en) 2003-06-12 2010-12-15 Euro Celtique Sa Therapeutic agents useful for treating pain
ATE431822T1 (de) * 2003-07-24 2009-06-15 Euro Celtique Sa Zur behandlung oder vorbeugung von schmerzen geeignete heteroaryl-tetrahydropiperidyl- verbindungen
DE602004020994D1 (de) * 2003-07-24 2009-06-18 Euro Celtique Sa Piperidinverbindungen und pharmazeutische zusammensetzungen, die diese enthalten
PL1942106T3 (pl) 2003-08-01 2012-02-29 Euro Celtique Sa Środki lecznicze użyteczne do leczenia bólu
KR20100005725A (ko) 2007-04-27 2010-01-15 퍼듀 퍼머 엘피 Ｔｒｐｖ１ 길항제 및 그의 용도
AU2008246202B2 (en) 2007-04-27 2011-12-01 Purdue Pharma L.P. Therapeutic agents useful for treating pain
RU2621708C2 (ru) 2011-06-22 2017-06-07 ПУРДЬЮ ФАРМА Эл. Пи. Антагонисты trpv1, включающие дигидроксигруппу в качестве заместителя, и их применение
WO2013146970A1 (ja) * 2012-03-29 2013-10-03 第一三共株式会社 新規キノリン誘導体
TWI652264B (zh) * 2013-09-26 2019-03-01 東麗股份有限公司 Cyclic amine derivatives and their medical uses
DE102022104759A1 (de) 2022-02-28 2023-08-31 SCi Kontor GmbH Co-Kristall-Screening Verfahren, insbesondere zur Herstellung von Co-Kristallen

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2579596B1 (fr) * 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique
WO1999064394A1 (en) * 1998-06-08 1999-12-16 Schering Corporation Neuropeptide y5 receptor antagonists
KR20030024799A (ko) * 2000-07-20 2003-03-26 뉴로젠 코포레이션 캡사이신 수용체 리간드
WO2003029199A1 (en) * 2001-09-28 2003-04-10 Takeda Chemical Industries, Ltd. Benzene derivatives, process for preparing the same and use thereof
JP2003192673A (ja) * 2001-12-27 2003-07-09 Bayer Ag ピペラジンカルボキシアミド誘導体
US7071335B2 (en) * 2002-02-01 2006-07-04 Euro-Celtique S.A. 2-pyridinyl-1-piperazine therapeutic agents useful for treating pain
US6974818B2 (en) * 2002-03-01 2005-12-13 Euro-Celtique S.A. 1,2,5-thiadiazol-3-YL-piperazine therapeutic agents useful for treating pain
US7262194B2 (en) * 2002-07-26 2007-08-28 Euro-Celtique S.A. Therapeutic agents useful for treating pain
EP2281823A3 (en) * 2003-05-20 2011-09-07 Ajinomoto Co., Inc. Anti-inflammatory and analgesic piperidine derivatives
MY142655A (en) * 2003-06-12 2010-12-15 Euro Celtique Sa Therapeutic agents useful for treating pain

Also Published As

Publication number Publication date
WO2005007642A3 (en) 2005-05-26
IL172985A0 (en) 2006-06-11
KR20060034282A (ko) 2006-04-21
TW200510372A (en) 2005-03-16
ZA200600228B (en) 2007-04-25
CN1849315A (zh) 2006-10-18
JP2007523865A (ja) 2007-08-23
BRPI0412438A (pt) 2006-09-05
CN101434596A (zh) 2009-05-20
AU2004257220A1 (en) 2005-01-27
US20050009841A1 (en) 2005-01-13
EP1646621A2 (en) 2006-04-19
WO2005007642A2 (en) 2005-01-27
CA2532057A1 (en) 2005-01-27

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