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MXPA04002067A - Nuevas dihidropteridinonas, procedimientos para su preparacion y su uso como medicamento. - Google Patents

Nuevas dihidropteridinonas, procedimientos para su preparacion y su uso como medicamento.

Info

Publication number
MXPA04002067A
MXPA04002067A MXPA04002067A MXPA04002067A MXPA04002067A MX PA04002067 A MXPA04002067 A MX PA04002067A MX PA04002067 A MXPA04002067 A MX PA04002067A MX PA04002067 A MXPA04002067 A MX PA04002067A MX PA04002067 A MXPA04002067 A MX PA04002067A
Authority
MX
Mexico
Prior art keywords
medicaments
producing
same
dihydropteridinones
novel
Prior art date
Application number
MXPA04002067A
Other languages
English (en)
Inventor
Grauert Matthias
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of MXPA04002067A publication Critical patent/MXPA04002067A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invencion se refiere a nuevas dihidro-pteridinonas de la formula general (I) (ver formula) teniendo los radicales X, R1, R2, R3, R4, R5 y R7 los significados mencionados en las reivindicaciones y en la memoria descriptiva, sus isomeros, procedimientos para la preparacion de estas dihidro-pteridinonas asi como su uso como medicamentos.
MXPA04002067A 2001-09-04 2002-08-30 Nuevas dihidropteridinonas, procedimientos para su preparacion y su uso como medicamento. MXPA04002067A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10143272 2001-09-04
PCT/EP2002/009728 WO2003020722A1 (de) 2001-09-04 2002-08-30 Neue dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
MXPA04002067A true MXPA04002067A (es) 2004-06-07

Family

ID=7697637

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA04002067A MXPA04002067A (es) 2001-09-04 2002-08-30 Nuevas dihidropteridinonas, procedimientos para su preparacion y su uso como medicamento.

Country Status (30)

Country Link
EP (1) EP1427730B1 (es)
JP (1) JP3876254B2 (es)
KR (1) KR100955589B1 (es)
CN (1) CN1551881A (es)
AR (1) AR036586A1 (es)
AT (1) ATE332898T1 (es)
AU (1) AU2002337047B2 (es)
BR (1) BRPI0212137A2 (es)
CA (1) CA2458699C (es)
CO (1) CO5560575A2 (es)
CY (1) CY1105337T1 (es)
DE (1) DE50207522D1 (es)
DK (1) DK1427730T3 (es)
EA (1) EA007062B1 (es)
EC (1) ECSP045003A (es)
ES (1) ES2268093T3 (es)
HR (1) HRP20040213A2 (es)
HU (1) HUP0401293A3 (es)
IL (2) IL160440A0 (es)
MX (1) MXPA04002067A (es)
MY (1) MY129751A (es)
NO (1) NO328804B1 (es)
NZ (1) NZ531928A (es)
PL (1) PL369740A1 (es)
PT (1) PT1427730E (es)
RS (1) RS51012B (es)
UA (1) UA76512C2 (es)
UY (1) UY27427A1 (es)
WO (1) WO2003020722A1 (es)
ZA (1) ZA200401365B (es)

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