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MY127144A - New anticholinergics which may be used as medicaments as well as processes for preparing them - Google Patents

New anticholinergics which may be used as medicaments as well as processes for preparing them

Info

Publication number
MY127144A
MY127144A MYPI20014765A MYPI20014765A MY127144A MY 127144 A MY127144 A MY 127144A MY PI20014765 A MYPI20014765 A MY PI20014765A MY PI20014765 A MYPI20014765 A MY PI20014765A MY 127144 A MY127144 A MY 127144A
Authority
MY
Malaysia
Prior art keywords
preparing
processes
medicaments
well
anticholinergics
Prior art date
Application number
MYPI20014765A
Inventor
Georg Speck Dr
Rolf Banholzer Dr
Richard Reichl Dr
Meissner Helmut
Morschhauser Gerd
Gerald Pohl Dr
Michael-Paul Pieper Dr
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of MY127144A publication Critical patent/MY127144A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • C07D451/10Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

THE PRESENT INVENTION RELATES TO NEW ANTICHOLINERGICS OF GENERAL FORMULA 1: WHEREIN A, X- AND THE GROUPS R1, R2, R3, R4, R5, R6 AND R7 MAY HAVE THE MEANINGS GIVEN IN THE CLAIMS AND IN THE SPECIFICATION, PROCESSES FOR PREPARING THEM AND THEIR USE AS PHARAMACEUTICAL COMPOSITIONS.
MYPI20014765A 2000-10-14 2001-10-12 New anticholinergics which may be used as medicaments as well as processes for preparing them MY127144A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050994A DE10050994A1 (en) 2000-10-14 2000-10-14 New diphenylalkanoic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease

Publications (1)

Publication Number Publication Date
MY127144A true MY127144A (en) 2006-11-30

Family

ID=7659808

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI20014765A MY127144A (en) 2000-10-14 2001-10-12 New anticholinergics which may be used as medicaments as well as processes for preparing them

Country Status (37)

Country Link
EP (2) EP1382606A3 (en)
JP (2) JP4109106B2 (en)
KR (1) KR100830359B1 (en)
CN (1) CN1275962C (en)
AR (1) AR035589A1 (en)
AT (1) ATE259805T1 (en)
AU (2) AU1397502A (en)
BG (1) BG66225B1 (en)
BR (1) BR0114635A (en)
CA (1) CA2425557C (en)
DE (2) DE10050994A1 (en)
DK (1) DK1325001T3 (en)
EA (1) EA005816B1 (en)
EC (1) ECSP034542A (en)
EE (1) EE05179B1 (en)
ES (1) ES2215147T3 (en)
HR (1) HRP20030278B1 (en)
HU (1) HUP0301203A3 (en)
IL (2) IL155334A0 (en)
ME (1) MEP39908A (en)
MX (1) MXPA03003160A (en)
MY (1) MY127144A (en)
NO (1) NO328207B1 (en)
NZ (1) NZ525836A (en)
PE (1) PE20020433A1 (en)
PL (1) PL207311B1 (en)
PT (1) PT1325001E (en)
RS (1) RS50464B (en)
SA (1) SA01220414B1 (en)
SI (1) SI1325001T1 (en)
SK (1) SK287138B6 (en)
TR (1) TR200400376T4 (en)
TW (1) TWI306098B (en)
UA (1) UA73804C2 (en)
UY (1) UY26958A1 (en)
WO (1) WO2002032899A1 (en)
ZA (1) ZA200302914B (en)

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Also Published As

Publication number Publication date
BG107688A (en) 2003-09-30
EA005816B1 (en) 2005-06-30
IL155334A (en) 2009-02-11
SA01220414B1 (en) 2007-01-20
EE200300151A (en) 2003-06-16
CA2425557A1 (en) 2003-04-11
CA2425557C (en) 2007-11-13
CN1468236A (en) 2004-01-14
TR200400376T4 (en) 2004-03-22
EP1325001A1 (en) 2003-07-09
DE50101524D1 (en) 2004-03-25
SK287138B6 (en) 2010-01-07
AR035589A1 (en) 2004-06-16
NZ525836A (en) 2004-09-24
DE10050994A1 (en) 2002-04-18
WO2002032899A1 (en) 2002-04-25
SI1325001T1 (en) 2004-08-31
HRP20030278A2 (en) 2005-02-28
AU1397502A (en) 2002-04-29
CN1275962C (en) 2006-09-20
ZA200302914B (en) 2003-11-14
BR0114635A (en) 2004-02-10
MEP39908A (en) 2011-02-10
TWI306098B (en) 2009-02-11
UY26958A1 (en) 2002-06-20
ATE259805T1 (en) 2004-03-15
EE05179B1 (en) 2009-06-15
ES2215147T3 (en) 2004-10-01
BG66225B1 (en) 2012-06-29
HUP0301203A3 (en) 2006-05-29
HK1060566A1 (en) 2004-08-13
EP1382606A2 (en) 2004-01-21
EP1325001B1 (en) 2004-02-18
PL207311B1 (en) 2010-11-30
AU2002213975B2 (en) 2006-11-09
JP4109106B2 (en) 2008-07-02
UA73804C2 (en) 2005-09-15
KR100830359B1 (en) 2008-05-20
RS50464B (en) 2010-03-02
YU29503A (en) 2006-03-03
PE20020433A1 (en) 2002-06-28
NO20031693D0 (en) 2003-04-11
JP2008120834A (en) 2008-05-29
KR20030041165A (en) 2003-05-23
NO20031693L (en) 2003-05-28
HRP20030278B1 (en) 2006-02-28
MXPA03003160A (en) 2005-09-09
DK1325001T3 (en) 2004-06-21
NO328207B1 (en) 2010-01-11
EA200300459A1 (en) 2003-10-30
SK4352003A3 (en) 2003-08-05
EP1382606A3 (en) 2004-10-13
JP2004511557A (en) 2004-04-15
ECSP034542A (en) 2003-06-25
PL360673A1 (en) 2004-09-20
HUP0301203A2 (en) 2003-10-28
IL155334A0 (en) 2003-11-23
PT1325001E (en) 2004-07-30

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