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MXPA02012563A - Compuestos ciclicos fusionados como moduladores de la funcion del receptor de la hormona nuclear. - Google Patents

Compuestos ciclicos fusionados como moduladores de la funcion del receptor de la hormona nuclear.

Info

Publication number
MXPA02012563A
MXPA02012563A MXPA02012563A MXPA02012563A MXPA02012563A MX PA02012563 A MXPA02012563 A MX PA02012563A MX PA02012563 A MXPA02012563 A MX PA02012563A MX PA02012563 A MXPA02012563 A MX PA02012563A MX PA02012563 A MXPA02012563 A MX PA02012563A
Authority
MX
Mexico
Prior art keywords
substituted
alkyl
dazo
heterocycle
methane
Prior art date
Application number
MXPA02012563A
Other languages
English (en)
Spanish (es)
Inventor
Mark E Salvati
Original Assignee
Squibb Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb Bristol Myers Co filed Critical Squibb Bristol Myers Co
Publication of MXPA02012563A publication Critical patent/MXPA02012563A/es

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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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MXPA02012563A 2000-06-28 2001-06-20 Compuestos ciclicos fusionados como moduladores de la funcion del receptor de la hormona nuclear. MXPA02012563A (es)

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US28461701P 2001-04-18 2001-04-18
PCT/US2001/019663 WO2002000653A2 (fr) 2000-06-28 2001-06-20 Modulateurs cycliques condenses de la fonction du recepteur hormonal nucleaire

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US7405234B2 (en) 2002-05-17 2008-07-29 Bristol-Myers Squibb Company Bicyclic modulators of androgen receptor function
EP1553074B1 (fr) 2002-08-12 2014-06-18 Takeda Pharmaceutical Company Limited Derive de benzene a cycles accoles et son utilisation
EP1567487A4 (fr) 2002-11-15 2005-11-16 Bristol Myers Squibb Co Modulateurs lies a prolyl uree a chaine ouverte de la fonction du recepteur d'androgene
US7199125B2 (en) 2003-10-02 2007-04-03 Bristol-Myers Squibb Company Spiro-cyclic compounds useful as anti-inflammatory agents
US7820702B2 (en) 2004-02-04 2010-10-26 Bristol-Myers Squibb Company Sulfonylpyrrolidine modulators of androgen receptor function and method
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CA2642205C (fr) * 2006-02-10 2015-01-27 Janssen Pharmaceutica N.V. Imidazole ou thiadiazole bicyclique servant de modulateur selectif de recepteur d'androgene
EP2039695A4 (fr) 2006-07-11 2010-09-15 Takeda Pharmaceutical Composé hétérocyclique bicycique et son utilisation
EP2334683B1 (fr) 2008-08-29 2017-03-22 MSD Italia S.r.l. Dérivés hétérocycliques bicycliques saturés en tant qu antagonistes de smo
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US9427418B2 (en) 2009-02-23 2016-08-30 Gtx, Inc. Estrogen receptor ligands and methods of use thereof

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WO2002000653A2 (fr) 2002-01-03
JP2004515462A (ja) 2004-05-27
HUP0303165A2 (hu) 2003-12-29
EP1299385A2 (fr) 2003-04-09
NZ523802A (en) 2005-11-25
BR0111869A (pt) 2003-09-23
WO2002000653A3 (fr) 2002-07-25
NO20026167L (no) 2002-12-20
CA2413683A1 (fr) 2002-01-03
NO20026167D0 (no) 2002-12-20
HUP0303165A3 (en) 2006-05-29
AU2002215609A1 (en) 2002-01-08

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