MX3308E - Procedimiento para la preparacion de derivados de la tieno-piridina - Google Patents
Procedimiento para la preparacion de derivados de la tieno-piridinaInfo
- Publication number
- MX3308E MX3308E MX000231U MX23176U MX3308E MX 3308 E MX3308 E MX 3308E MX 000231 U MX000231 U MX 000231U MX 23176 U MX23176 U MX 23176U MX 3308 E MX3308 E MX 3308E
- Authority
- MX
- Mexico
- Prior art keywords
- formula
- derivatives
- preparation
- alcoholic
- radical
- Prior art date
Links
- 230000001476 alcoholic effect Effects 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000012948 isocyanate Substances 0.000 abstract 1
- 150000002513 isocyanates Chemical class 0.000 abstract 1
- 150000003242 quaternary ammonium salts Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- DBDCNCCRPKTRSD-UHFFFAOYSA-N thieno[3,2-b]pyridine Chemical class C1=CC=C2SC=CC2=N1 DBDCNCCRPKTRSD-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a procedimiento para la preparación de derivados de la tieno-piridina de fórmula: (VER FIGURA) sus sales de adición con ácidos y sus sales de amonio cuaternario caracterizado porque se hace reccionar un compuesto de fórmulas (VER FIGURA) obteniendo así los derivados de fórmula (I) o (II), en las cuales R2 es hidrógeno, que se puede hacer reaccionar con un agente acilante de fórmula C1COR4 ó (R4 CO2)O, en las cuales R4 es un radical alcohilo, aralcohilo ó arilo para obtener un derivado de fórmula (I) ó (II), en la cual R2 es un grupo acilo; o con un isocianato de fórmula R5NCO, en la cual R5 es un radical alcohilo, para obtener un derivado de fórmula (I) ó (II) en las cuales R2 es un radical alcohilaminocarbonilo.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7517007A FR2312247A1 (fr) | 1975-05-30 | 1975-05-30 | Derives de la thieno-pyridine, leur procede de preparation et leurs applications |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX3308E true MX3308E (es) | 1980-09-09 |
Family
ID=9155902
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX000231U MX3308E (es) | 1975-05-30 | 1976-05-13 | Procedimiento para la preparacion de derivados de la tieno-piridina |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4076819A (es) |
| JP (1) | JPS51149297A (es) |
| AR (1) | AR211339A1 (es) |
| AT (1) | AT349471B (es) |
| AU (1) | AU498517B2 (es) |
| BE (1) | BE842310A (es) |
| CA (1) | CA1071633A (es) |
| CH (1) | CH613969A5 (es) |
| DD (1) | DD125214A5 (es) |
| DE (1) | DE2623567C2 (es) |
| DK (1) | DK235876A (es) |
| ES (1) | ES447570A1 (es) |
| FR (1) | FR2312247A1 (es) |
| GB (1) | GB1501797A (es) |
| GR (1) | GR59797B (es) |
| HU (1) | HU172176B (es) |
| IE (1) | IE43224B1 (es) |
| IL (1) | IL49405A (es) |
| LU (1) | LU74617A1 (es) |
| MX (1) | MX3308E (es) |
| NL (1) | NL7604944A (es) |
| PL (1) | PL100792B1 (es) |
| RO (1) | RO68891A (es) |
| SE (1) | SE421623B (es) |
| SU (1) | SU667138A3 (es) |
| YU (1) | YU39479B (es) |
| ZA (1) | ZA762263B (es) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2376860A1 (fr) * | 1977-01-07 | 1978-08-04 | Parcor | Tetrahydro-4,5,6,7 thieno (2,3-c) et (3,2-c) pyridines, leur procede de preparation et leur application therapeutique |
| FR2395271A1 (fr) * | 1977-06-21 | 1979-01-19 | Parcor | Procede de preparation de thieno (2,3-c) et thieno (3,2-c) pyridines |
| FR2397417A1 (fr) * | 1977-07-12 | 1979-02-09 | Parcor | Procede de preparation de derives de la thienopyridine |
| US4321266A (en) * | 1980-10-06 | 1982-03-23 | Sanofi | 5-o-Cyanobenzyl-4,5,6,7-tetrahydrothieno [3,2-C] pyridine |
| FR2597102B1 (fr) * | 1986-04-14 | 1988-08-26 | Sanofi Sa | Derives de l'acide a-(hydroxy-7 tetrahydro-4,5,6,7 thieno (3,2-c) pyridyl-5) phenyl acetique, leur procede de preparation, leur application comme medicament et les compositions les renfermant |
| AU5154699A (en) * | 1998-09-02 | 2000-03-27 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno(2,3-c)pyridine derivatives |
| US6090797A (en) * | 1998-09-02 | 2000-07-18 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno(2,3-C)pyridine derivatives |
| PT1350511E (pt) | 2000-12-25 | 2008-10-28 | Ube Industries | Composições medicinais contendo aspirina |
| US7838026B2 (en) | 2001-09-28 | 2010-11-23 | Mcneil-Ppc, Inc. | Burst-release polymer composition and dosage forms comprising the same |
| US7122143B2 (en) * | 2001-09-28 | 2006-10-17 | Mcneil-Ppc, Inc. | Methods for manufacturing dosage forms |
| CA2461653A1 (en) * | 2001-09-28 | 2003-04-03 | Mcneil-Ppc, Inc. | Edible composition and dosage form comprising an edible shell |
| US7323192B2 (en) * | 2001-09-28 | 2008-01-29 | Mcneil-Ppc, Inc. | Immediate release tablet |
| US7064211B2 (en) * | 2002-03-22 | 2006-06-20 | Eisai Co., Ltd. | Hemiasterlin derivatives and uses thereof |
| TWI350168B (en) | 2004-05-07 | 2011-10-11 | Incyte Corp | Amido compounds and their use as pharmaceuticals |
| US20060009471A1 (en) * | 2004-06-24 | 2006-01-12 | Wenqing Yao | Amido compounds and their use as pharmaceuticals |
| WO2006012226A2 (en) | 2004-06-24 | 2006-02-02 | Incyte Corporation | N-substituted piperidines and their use as pharmaceuticals |
| WO2006002350A1 (en) * | 2004-06-24 | 2006-01-05 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
| JP2008504280A (ja) * | 2004-06-24 | 2008-02-14 | インサイト・コーポレイション | ２−メチルプロパンアミドおよびその医薬としての使用 |
| CN101080226A (zh) * | 2004-08-10 | 2007-11-28 | 因塞特公司 | 酰氨基化合物及它们作为药物的用途 |
| KR20070097441A (ko) * | 2004-11-18 | 2007-10-04 | 인사이트 산 디에고 인코포레이티드 | 11-β 하이드록실 스테로이드 데하이드로게나제 유형 1의억제제 및 이를 사용하는 방법 |
| US8673352B2 (en) * | 2005-04-15 | 2014-03-18 | Mcneil-Ppc, Inc. | Modified release dosage form |
| WO2007038138A2 (en) * | 2005-09-21 | 2007-04-05 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
| EP1957494A2 (en) * | 2005-12-05 | 2008-08-20 | Incyte Corporation | Lactam compounds and methods of using the same |
| US7998959B2 (en) * | 2006-01-12 | 2011-08-16 | Incyte Corporation | Modulators of 11-β hydroxyl steroid dehydrogenase type 1, pharmaceutical compositions thereof, and methods of using the same |
| KR20080091503A (ko) * | 2006-01-31 | 2008-10-13 | 인사이트 코포레이션 | 아미도 화합물 및 약제로서의 이의 용도 |
| TW200808807A (en) * | 2006-03-02 | 2008-02-16 | Incyte Corp | Modulators of 11-β hydroxyl steroid dehydrogenase type 1, pharmaceutical compositions thereof, and methods of using the same |
| US20070208001A1 (en) * | 2006-03-03 | 2007-09-06 | Jincong Zhuo | Modulators of 11- beta hydroxyl steroid dehydrogenase type 1, pharmaceutical compositions thereof, and methods of using the same |
| WO2007130898A1 (en) * | 2006-05-01 | 2007-11-15 | Incyte Corporation | TETRASUBSTITUTED UREAS AS MODULATORS OF 11-β HYDROXYL STEROID DEHYDROGENASE TYPE 1 |
| WO2007137066A2 (en) * | 2006-05-17 | 2007-11-29 | Incyte Corporation | HETEROCYCLIC INHIBITORS OF 11-β HYDROXYL STEROID DEHYDROGENASE TYPE I AND METHODS OF USING THE SAME |
| MX2009010559A (es) * | 2007-03-30 | 2009-10-22 | Nippon Shinyaku Co Ltd | Derivados de heteroarilo. |
| CN102241690B (zh) | 2010-05-13 | 2015-08-12 | 天津药物研究院 | 一类含腈基的噻吩并吡啶酯类衍生物、其制备方法和用途 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2215948B1 (es) * | 1973-02-01 | 1976-05-14 | Centre Etd Ind Pharma | |
| AR205040A1 (es) * | 1974-07-16 | 1976-03-31 | Parcor | Procedimiento de preparacion de derivados de la tetrahidro-4,5,6,7,-tieno(3,2-c)o(2,3-c)piridina |
-
1975
- 1975-05-30 FR FR7517007A patent/FR2312247A1/fr active Granted
-
1976
- 1976-03-19 CH CH345676A patent/CH613969A5/xx not_active IP Right Cessation
- 1976-03-22 LU LU74617A patent/LU74617A1/xx unknown
- 1976-03-23 GR GR50384A patent/GR59797B/el unknown
- 1976-04-05 YU YU856/76A patent/YU39479B/xx unknown
- 1976-04-12 IE IE763/76A patent/IE43224B1/en unknown
- 1976-04-13 IL IL49405A patent/IL49405A/xx unknown
- 1976-04-14 CA CA250,739A patent/CA1071633A/en not_active Expired
- 1976-04-14 ZA ZA762263A patent/ZA762263B/xx unknown
- 1976-04-14 US US05/676,796 patent/US4076819A/en not_active Expired - Lifetime
- 1976-05-04 ES ES447570A patent/ES447570A1/es not_active Expired
- 1976-05-05 AR AR263208A patent/AR211339A1/es active
- 1976-05-07 NL NL7604944A patent/NL7604944A/xx not_active Application Discontinuation
- 1976-05-13 MX MX000231U patent/MX3308E/es unknown
- 1976-05-17 SU SU762356004A patent/SU667138A3/ru active
- 1976-05-22 RO RO7686177A patent/RO68891A/ro unknown
- 1976-05-26 DE DE2623567A patent/DE2623567C2/de not_active Expired
- 1976-05-26 AT AT386576A patent/AT349471B/de not_active IP Right Cessation
- 1976-05-28 BE BE167404A patent/BE842310A/xx not_active IP Right Cessation
- 1976-05-28 HU HU76PA00001248A patent/HU172176B/hu not_active IP Right Cessation
- 1976-05-28 DD DD193073A patent/DD125214A5/xx unknown
- 1976-05-28 DK DK235876A patent/DK235876A/da unknown
- 1976-05-28 GB GB22400/76A patent/GB1501797A/en not_active Expired
- 1976-05-28 AU AU14417/76A patent/AU498517B2/en not_active Expired
- 1976-05-28 SE SE7606062A patent/SE421623B/xx not_active IP Right Cessation
- 1976-05-29 PL PL1976189958A patent/PL100792B1/xx unknown
- 1976-05-29 JP JP51062884A patent/JPS51149297A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| CA1071633A (en) | 1980-02-12 |
| AT349471B (de) | 1979-04-10 |
| ES447570A1 (es) | 1977-07-01 |
| PL100792B1 (pl) | 1978-11-30 |
| CH613969A5 (es) | 1979-10-31 |
| HU172176B (hu) | 1978-06-28 |
| IE43224L (en) | 1976-11-30 |
| IE43224B1 (en) | 1981-01-14 |
| SE7606062L (sv) | 1976-12-01 |
| DE2623567A1 (de) | 1976-12-09 |
| DD125214A5 (es) | 1977-04-06 |
| RO68891A (ro) | 1982-09-09 |
| GR59797B (en) | 1978-02-28 |
| AR211339A1 (es) | 1977-11-30 |
| YU85676A (en) | 1982-06-30 |
| YU39479B (en) | 1984-12-31 |
| JPS51149297A (en) | 1976-12-22 |
| SU667138A3 (ru) | 1979-06-05 |
| LU74617A1 (es) | 1976-09-01 |
| ZA762263B (en) | 1977-04-27 |
| NL7604944A (nl) | 1976-12-02 |
| GB1501797A (en) | 1978-02-22 |
| IL49405A (en) | 1979-09-30 |
| ATA386576A (de) | 1978-09-15 |
| SE421623B (sv) | 1982-01-18 |
| FR2312247A1 (fr) | 1976-12-24 |
| DE2623567C2 (de) | 1984-03-01 |
| AU498517B2 (en) | 1979-03-15 |
| DK235876A (da) | 1976-12-01 |
| FR2312247B1 (es) | 1978-08-18 |
| US4076819A (en) | 1978-02-28 |
| AU1441776A (en) | 1977-12-01 |
| BE842310A (fr) | 1976-11-29 |
| IL49405A0 (en) | 1976-06-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MX3308E (es) | Procedimiento para la preparacion de derivados de la tieno-piridina | |
| ES478228A1 (es) | Procedimiento para la preparacion de derivados de acidos fe-noxi-alcohilcarboxilicos. | |
| ES473818A1 (es) | Procedimiento para preparar derivados de piperazina. | |
| ES464463A1 (es) | Un procedimiento para preparar derivados de acilo sustituidode aminoacidos. | |
| BR7606378A (pt) | Processo para producao de gas de sintese | |
| ES2058292T3 (es) | Derivados de indol. | |
| ES456694A1 (es) | Procedimiento para preparar colorantes que contienen un sis-tema cromoforico. | |
| ES387016A1 (es) | Un procedimiento para la preparacion de derivado de isoqui-nolina. | |
| ES485096A1 (es) | Un procedimiento para preparar aminoglicosidos | |
| ES8307718A1 (es) | "procedimiento de preparar amidoaminoacidos y similares". | |
| ES8403127A1 (es) | Procedimiento para la preparacion de derivados de eburnamonina. | |
| ES453861A1 (es) | Un procedimiento para la preparacion de nuevos derivados de indazol. | |
| ES461796A1 (es) | Un procedimiento para la preparacion de nuevos derivados de tiofeno. | |
| IT1050008B (it) | Processo per la preparazione di coloranti ossazinici basici | |
| IT1062521B (it) | Processo per la preparazione di derivati nitrilici | |
| ES465322A1 (es) | Un procedimiento para preparar compuestos e imericos de 4"- amino. | |
| MX3034E (es) | Procedimiento para preparar esteres de acido alquil iden amino oxi alquil carboxilico | |
| MX3388E (es) | Procedimiento para la preparacion de homoftalimidas | |
| ES308785A1 (es) | Procedimiento para la preparacion de derivados de benzimidazolona. | |
| ES172075A1 (es) | UN PROCEDIMIENTO DE PRODUCIR N - PENToSIDAS AMiNICAS AROMáTICAS. | |
| ES481314A1 (es) | Procedimiento para la preparacion de halogenobenzoin-o-metil-eter-oximas. | |
| MX2978E (es) | Procedimiento para la preparacion de derivados sustituidos de piperazina 5 - metil o 5 - metil tio pirimidina | |
| ES455532A1 (es) | Procedimiento para la preparacion de triazapentadienos. | |
| SE387343B (sv) | Sett att framstella tienyl-imidazolyl-fettsyraderivat avsedda att anvendas som antimykotika | |
| AR217037A1 (es) | Nuevos derivados de aminas policiclicas policlorados con puente metilenico,composiciones insecticidas que los contienen,y metodo para producirlos |