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MX2022012833A - (s)-(4,5-dihidro-7h-tieno[2,3-c]piran-7-il)-n-metilmetanamina para tratar trastornos neurologicos y psiquiatricos. - Google Patents

(s)-(4,5-dihidro-7h-tieno[2,3-c]piran-7-il)-n-metilmetanamina para tratar trastornos neurologicos y psiquiatricos.

Info

Publication number
MX2022012833A
MX2022012833A MX2022012833A MX2022012833A MX2022012833A MX 2022012833 A MX2022012833 A MX 2022012833A MX 2022012833 A MX2022012833 A MX 2022012833A MX 2022012833 A MX2022012833 A MX 2022012833A MX 2022012833 A MX2022012833 A MX 2022012833A
Authority
MX
Mexico
Prior art keywords
methylmethanamine
thieno
pyran
dihydro
treating neurological
Prior art date
Application number
MX2022012833A
Other languages
English (en)
Inventor
Carrie A Bowen
Seth Cabot Hopkins
Colleen M Synan
Original Assignee
Sunovion Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sunovion Pharmaceuticals Inc filed Critical Sunovion Pharmaceuticals Inc
Publication of MX2022012833A publication Critical patent/MX2022012833A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Addiction (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

La presente invención se refiere a métodos para tratar enfermedades o trastornos neurológicos o psiquiátricos, tal como la esquizofrenia. El Compuesto 1, o una sal farmacéuticamente aceptable del mismo, es un agente antipsicótico con un mecanismo de acción no D2. Los eventos adversos asociados con los agentes antipsicóticos que se dirigen al receptor de dopamina D2 pueden reducirse tratando los trastornos con el Compuesto 1, o una sal farmacéuticamente aceptable del mismo.
MX2022012833A 2020-04-14 2021-04-13 (s)-(4,5-dihidro-7h-tieno[2,3-c]piran-7-il)-n-metilmetanamina para tratar trastornos neurologicos y psiquiatricos. MX2022012833A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063009595P 2020-04-14 2020-04-14
US202063039722P 2020-06-16 2020-06-16
PCT/US2021/026953 WO2021211489A1 (en) 2020-04-14 2021-04-13 (s)-(4,5-dihydro-7h-thieno[2,3-c]pyran-7-yl)-n-methylmethanamine for treating neurological and psychiatric disorders

Publications (1)

Publication Number Publication Date
MX2022012833A true MX2022012833A (es) 2022-11-07

Family

ID=75787267

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022012833A MX2022012833A (es) 2020-04-14 2021-04-13 (s)-(4,5-dihidro-7h-tieno[2,3-c]piran-7-il)-n-metilmetanamina para tratar trastornos neurologicos y psiquiatricos.

Country Status (11)

Country Link
US (2) US11738002B2 (es)
EP (1) EP4135690A1 (es)
JP (1) JP7781768B2 (es)
KR (1) KR20230003503A (es)
CN (1) CN115734785A (es)
AU (1) AU2021257786A1 (es)
CA (1) CA3180115A1 (es)
IL (1) IL297248A (es)
MX (1) MX2022012833A (es)
WO (1) WO2021211489A1 (es)
ZA (1) ZA202211311B (es)

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CA3091292A1 (en) 2018-02-16 2019-08-22 Sunovion Pharmaceuticals Inc. Salts, crystal forms, and production methods thereof
US11738002B2 (en) 2020-04-14 2023-08-29 Sunovion Pharmaceuticals Inc. Methods of treating neurological and psychiatric disorders
CN114377007A (zh) * 2022-02-23 2022-04-22 江苏海洋大学 一种度洛西汀与sep-363856联用用于制备治疗抑郁症的药物组合物
US12400766B1 (en) 2022-07-22 2025-08-26 Veeva Systems Inc. Systems and methods for electronically collecting and linking standardized case data in a data warehouse
EP4580615A1 (en) * 2022-08-30 2025-07-09 Sumitomo Pharma America, Inc. Ulotaront for the adjuvant treatment of major depressive disorder
EP4601634A1 (en) 2022-10-13 2025-08-20 Sumitomo Pharma America, Inc. Methods of reducing physical dependence to neuropsychiatric treatments
AU2023367071A1 (en) * 2022-10-28 2025-06-12 Sumitomo Pharma America, Inc. Ulotaront for treating anxiety and associated conditions
WO2025179091A2 (en) * 2024-02-23 2025-08-28 Sumitomo Pharma America, Inc. Ulotaront hydrochloride manufacturing process
WO2025252814A1 (en) 2024-06-04 2025-12-11 Duc Duy Vo Methods for treating trace amine-associated receptor 1 (taar1)-associated diseases or disorders comprising administration of novel taar1 agonists or pharmaceutical compositions thereof

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US20210315859A1 (en) 2021-10-14
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