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MX2018011992A - Compuestos de aminopurina sustituida, composiciones de estos y metodos de tratamiento con estos. - Google Patents

Compuestos de aminopurina sustituida, composiciones de estos y metodos de tratamiento con estos.

Info

Publication number
MX2018011992A
MX2018011992A MX2018011992A MX2018011992A MX2018011992A MX 2018011992 A MX2018011992 A MX 2018011992A MX 2018011992 A MX2018011992 A MX 2018011992A MX 2018011992 A MX2018011992 A MX 2018011992A MX 2018011992 A MX2018011992 A MX 2018011992A
Authority
MX
Mexico
Prior art keywords
compositions
methods
aminopurine compounds
treatment therewith
substituted aminopurine
Prior art date
Application number
MX2018011992A
Other languages
English (en)
Other versions
MX379513B (es
Inventor
F Boylan John
L Bray Gordon
Filvaroff Ellen
Hubbard Robert
Mikolon David
Raymon Heather
Shi Tao
M Tran Tam
L Wong Lilly
Xu Suichan
Zhu Dan
Tsuji Toshiya
Original Assignee
Signal Pharm Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Signal Pharm Llc filed Critical Signal Pharm Llc
Publication of MX2018011992A publication Critical patent/MX2018011992A/es
Publication of MX379513B publication Critical patent/MX379513B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se proporcionan en la presente métodos para el tratamiento o prevención de un cáncer, que incluyen sólidos y canceres hematológicos, que comprenden administrar una cantidad eficaz de compuestos de Aminopurina de formula (I) y composiciones que comprenden una cantidad eficaz de dichos compuestos.
MX2018011992A 2016-04-01 2017-03-31 Compuestos de aminopurina sustituida, composiciones de estos y métodos de tratamiento con estos. MX379513B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662317412P 2016-04-01 2016-04-01
PCT/US2017/025252 WO2017173206A1 (en) 2016-04-01 2017-03-31 Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith

Publications (2)

Publication Number Publication Date
MX2018011992A true MX2018011992A (es) 2019-01-24
MX379513B MX379513B (es) 2025-03-11

Family

ID=59959573

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018011992A MX379513B (es) 2016-04-01 2017-03-31 Compuestos de aminopurina sustituida, composiciones de estos y métodos de tratamiento con estos.

Country Status (15)

Country Link
US (1) US10576085B2 (es)
EP (1) EP3436018A4 (es)
JP (1) JP7014731B2 (es)
KR (1) KR102356433B1 (es)
CN (1) CN109069512B (es)
AU (1) AU2017241837B2 (es)
BR (1) BR112018070163A2 (es)
CA (1) CA3018986A1 (es)
CL (1) CL2018002787A1 (es)
EA (1) EA039392B1 (es)
IL (1) IL262007B2 (es)
MX (1) MX379513B (es)
NZ (1) NZ746554A (es)
SG (2) SG10202009589UA (es)
WO (1) WO2017173206A1 (es)

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JOP20180026A1 (ar) 2017-03-31 2019-01-30 Univ Leuven Kath مشتقات اندولين مستبدلة بصفتها مانعات للتكاثر الفيروسي لحمى الفنك
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JP7287955B2 (ja) 2017-10-04 2023-06-06 セルジーン コーポレイション シス-4-[2-{[(3s,4r)-3-フルオロオキサン-4-イル]アミノ}-8-(2,4,6-トリクロロアニリノ)-9h-プリン-9-イル]-1-メチルシクロヘキサン-1-カルボキサミドの組成物及び使用方法
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Also Published As

Publication number Publication date
BR112018070163A2 (pt) 2019-01-29
AU2017241837B2 (en) 2021-07-22
JP7014731B2 (ja) 2022-02-01
SG11201808388QA (en) 2018-10-30
US20170281633A1 (en) 2017-10-05
IL262007B2 (en) 2023-04-01
WO2017173206A1 (en) 2017-10-05
CN109069512A (zh) 2018-12-21
IL262007B (en) 2022-12-01
EA039392B1 (ru) 2022-01-21
EP3436018A1 (en) 2019-02-06
NZ746554A (en) 2023-03-31
SG10202009589UA (en) 2020-10-29
JP2019510066A (ja) 2019-04-11
IL262007A (en) 2018-10-31
EA201892229A1 (ru) 2019-03-29
KR20180126497A (ko) 2018-11-27
EP3436018A4 (en) 2019-11-13
AU2017241837A1 (en) 2018-10-25
CL2018002787A1 (es) 2019-01-18
CA3018986A1 (en) 2017-10-05
US10576085B2 (en) 2020-03-03
CN109069512B (zh) 2022-06-14
KR102356433B1 (ko) 2022-01-27
MX379513B (es) 2025-03-11

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