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MX2018003875A - Alquilacion de picolinamidas con cloroacilales sustituidos con el uso de un catalizador de eter de corona. - Google Patents

Alquilacion de picolinamidas con cloroacilales sustituidos con el uso de un catalizador de eter de corona.

Info

Publication number
MX2018003875A
MX2018003875A MX2018003875A MX2018003875A MX2018003875A MX 2018003875 A MX2018003875 A MX 2018003875A MX 2018003875 A MX2018003875 A MX 2018003875A MX 2018003875 A MX2018003875 A MX 2018003875A MX 2018003875 A MX2018003875 A MX 2018003875A
Authority
MX
Mexico
Prior art keywords
chloroacylals
picolinamides
alkylation
substituted
utilizing
Prior art date
Application number
MX2018003875A
Other languages
English (en)
Inventor
Jansma Matthew
Adaway Timothy
Trippeer Michael
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of MX2018003875A publication Critical patent/MX2018003875A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J27/00Catalysts comprising the elements or compounds of halogens, sulfur, selenium, tellurium, phosphorus or nitrogen; Catalysts comprising carbon compounds
    • B01J27/06Halogens; Compounds thereof
    • B01J27/08Halides
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J31/00Catalysts comprising hydrides, coordination complexes or organic compounds
    • B01J31/02Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides
    • B01J31/0201Oxygen-containing compounds
    • B01J31/0204Ethers
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J31/00Catalysts comprising hydrides, coordination complexes or organic compounds
    • B01J31/16Catalysts comprising hydrides, coordination complexes or organic compounds containing coordination complexes
    • B01J31/22Organic complexes
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J31/00Catalysts comprising hydrides, coordination complexes or organic compounds
    • B01J31/26Catalysts comprising hydrides, coordination complexes or organic compounds containing in addition, inorganic metal compounds not provided for in groups B01J31/02 - B01J31/24
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2231/00Catalytic reactions performed with catalysts classified in B01J31/00
    • B01J2231/40Substitution reactions at carbon centres, e.g. C-C or C-X, i.e. carbon-hetero atom, cross-coupling, C-H activation or ring-opening reactions
    • B01J2231/44Allylic alkylation, amination, alkoxylation or analogues
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2531/00Additional information regarding catalytic systems classified in B01J31/00
    • B01J2531/001General concepts, e.g. reviews, relating to catalyst systems and methods of making them, the concept being defined by a common material or method/theory
    • B01J2531/002Materials
    • B01J2531/007Promoter-type Additives
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2531/00Additional information regarding catalytic systems classified in B01J31/00
    • B01J2531/90Catalytic systems characterized by the solvent or solvent system used
    • B01J2531/98Phase-transfer catalysis in a mixed solvent system containing at least 2 immiscible solvents or solvent phases

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Materials Engineering (AREA)
  • Inorganic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Plant Pathology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Un proceso para la alquilación de picolinamidas con cloroacilales sustituidos para producir una estructura de la Fórmula (III), en donde la reacción se realiza en la presencia de un catalizador de transferencia de fase y un cocatalizador de haluro inorgánico.
MX2018003875A 2015-10-06 2016-10-04 Alquilacion de picolinamidas con cloroacilales sustituidos con el uso de un catalizador de eter de corona. MX2018003875A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562237844P 2015-10-06 2015-10-06
PCT/US2016/055331 WO2017062362A1 (en) 2015-10-06 2016-10-04 Alkylation of picolinamides with substituted chloroacylals utilizing a crown ether catalyst

Publications (1)

Publication Number Publication Date
MX2018003875A true MX2018003875A (es) 2018-08-16

Family

ID=58447241

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018003875A MX2018003875A (es) 2015-10-06 2016-10-04 Alquilacion de picolinamidas con cloroacilales sustituidos con el uso de un catalizador de eter de corona.

Country Status (19)

Country Link
US (1) US10144728B2 (es)
EP (1) EP3359153B1 (es)
JP (2) JP6975142B2 (es)
KR (1) KR102687147B1 (es)
CN (1) CN108135890B (es)
AR (1) AR106262A1 (es)
BR (1) BR102016023198B8 (es)
CA (1) CA3000198C (es)
CO (1) CO2018003474A2 (es)
DK (1) DK3359153T3 (es)
ES (1) ES2858364T3 (es)
HU (1) HUE052841T2 (es)
IL (1) IL258386B (es)
LT (1) LT3359153T (es)
MX (1) MX2018003875A (es)
PL (1) PL3359153T3 (es)
TW (1) TWI718187B (es)
WO (1) WO2017062362A1 (es)
ZA (1) ZA201802085B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202146007A (zh) * 2020-02-27 2021-12-16 法商賽諾菲公司 包含阿培利司(alpelisib)與6-(2,4-二氯苯基)-5-[4-[(3s)-1-(3-氟丙基)吡咯啶-3-基]氧苯基]-8,9-二氫-7h-苯并[7]輪烯-2-羧酸之組合

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5480762A (en) * 1990-11-28 1996-01-02 Fuji Photo Film Co., Ltd. Method for preparing lithographic printing plate
AR037328A1 (es) * 2001-10-23 2004-11-03 Dow Agrosciences Llc Compuesto de [7-bencil-2,6-dioxo-1,5-dioxonan-3-il]-4-metoxipiridin-2-carboxamida, composicion que lo comprende y metodo que lo utiliza
US6861930B2 (en) 2001-11-15 2005-03-01 Eaton Corporation Transfer switch including a circuit breaker housing
US7091270B2 (en) * 2002-01-31 2006-08-15 Bromine Compounds Ltd. Pentabromobenzyl alkyl ethers and their use as fire retardants
US20130060023A1 (en) 2011-09-07 2013-03-07 Satori Pharmaceuticals, Inc. Compounds useful for treating neurodegenerative disorders
EP2847187A4 (en) * 2012-05-07 2015-10-28 Dow Agrosciences Llc MACROCYCLIC PICOLINAMIDE AS FUNGICIDES
EP2875024A4 (en) * 2012-07-20 2015-12-23 Merck Sharp & Dohme HIV TREATMENT WITH AMIDOSUBSTITUTED PYRIMIDINONE DERIVATIVES

Also Published As

Publication number Publication date
TWI718187B (zh) 2021-02-11
CO2018003474A2 (es) 2018-06-12
LT3359153T (lt) 2021-03-25
JP2021185157A (ja) 2021-12-09
WO2017062362A9 (en) 2017-12-28
EP3359153A4 (en) 2019-05-08
TW201718560A (zh) 2017-06-01
BR102016023198B8 (pt) 2022-09-06
ES2858364T3 (es) 2021-09-30
CN108135890B (zh) 2024-07-09
WO2017062362A1 (en) 2017-04-13
EP3359153A1 (en) 2018-08-15
KR20180066101A (ko) 2018-06-18
CA3000198C (en) 2024-02-27
US20170096414A1 (en) 2017-04-06
ZA201802085B (en) 2019-06-26
AR106262A1 (es) 2017-12-27
EP3359153B1 (en) 2020-12-16
JP2018537407A (ja) 2018-12-20
BR102016023198B1 (pt) 2021-06-22
BR102016023198A2 (pt) 2017-04-18
HUE052841T2 (hu) 2021-05-28
CA3000198A1 (en) 2017-04-13
KR102687147B1 (ko) 2024-07-24
IL258386B (en) 2021-02-28
IL258386A (en) 2018-05-31
DK3359153T3 (da) 2021-03-08
US10144728B2 (en) 2018-12-04
PL3359153T3 (pl) 2021-07-05
JP6975142B2 (ja) 2021-12-01
CN108135890A (zh) 2018-06-08

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