MX2017014463A - Cabazitaxel y su uso para tratar cancer. - Google Patents
Cabazitaxel y su uso para tratar cancer.Info
- Publication number
- MX2017014463A MX2017014463A MX2017014463A MX2017014463A MX2017014463A MX 2017014463 A MX2017014463 A MX 2017014463A MX 2017014463 A MX2017014463 A MX 2017014463A MX 2017014463 A MX2017014463 A MX 2017014463A MX 2017014463 A MX2017014463 A MX 2017014463A
- Authority
- MX
- Mexico
- Prior art keywords
- cabazitaxel
- treating cancer
- cancer
- solvate
- hydrate
- Prior art date
Links
- 206010028980 Neoplasm Diseases 0.000 title abstract 2
- 201000011510 cancer Diseases 0.000 title abstract 2
- BMQGVNUXMIRLCK-OAGWZNDDSA-N cabazitaxel Chemical compound O([C@H]1[C@@H]2[C@]3(OC(C)=O)CO[C@@H]3C[C@@H]([C@]2(C(=O)[C@H](OC)C2=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)C=3C=CC=CC=3)C[C@]1(O)C2(C)C)C)OC)C(=O)C1=CC=CC=C1 BMQGVNUXMIRLCK-OAGWZNDDSA-N 0.000 title 1
- 229960001573 cabazitaxel Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 208000019423 liver disease Diseases 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J1/00—Containers specially adapted for medical or pharmaceutical purposes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J2205/00—General identification or selection means
- A61J2205/30—Printed labels
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Urology & Nephrology (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
Abstract
La presente invención se refiere al compuesto que tiene la fórmula (I): (ver Fórmula) que puede estar en forma de base o en la forma de un hidrato o un solvato, para su uso como un medicamento en el tratamiento de cáncer en pacientes con insuficiencia hepática.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15305720.3A EP3093014A1 (en) | 2015-05-13 | 2015-05-13 | Cabazitaxel and its use for treating cancer |
| PCT/EP2016/060759 WO2016180943A1 (en) | 2015-05-13 | 2016-05-12 | Cabazitaxel and its use for treating cancer |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2017014463A true MX2017014463A (es) | 2018-03-21 |
Family
ID=53177311
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2017014463A MX2017014463A (es) | 2015-05-13 | 2016-05-12 | Cabazitaxel y su uso para tratar cancer. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20160331717A1 (es) |
| EP (3) | EP3093014A1 (es) |
| JP (1) | JP2018516890A (es) |
| KR (1) | KR20180006417A (es) |
| CN (1) | CN108135878A (es) |
| AU (1) | AU2016259775A1 (es) |
| CA (1) | CA2985408A1 (es) |
| EA (1) | EA201792502A1 (es) |
| ES (1) | ES2774101T3 (es) |
| IL (1) | IL255541A (es) |
| MX (1) | MX2017014463A (es) |
| PL (1) | PL3294285T3 (es) |
| PT (1) | PT3294285T (es) |
| TW (1) | TW201705950A (es) |
| WO (1) | WO2016180943A1 (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102770131A (zh) | 2009-10-29 | 2012-11-07 | 安万特医药股份有限公司 | 卡巴他赛的新颖抗肿瘤用途 |
| EP3093014A1 (en) | 2015-05-13 | 2016-11-16 | Aventis Pharma S.A. | Cabazitaxel and its use for treating cancer |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA23823A1 (fr) | 1995-03-27 | 1996-10-01 | Aventis Pharma Sa | Nouveaux taxoides, leur preparation et les compositions qui les contiennent |
| US5847170A (en) | 1995-03-27 | 1998-12-08 | Rhone-Poulenc Rorer, S.A. | Taxoids, their preparation and pharmaceutical compositions containing them |
| ES2248684T3 (es) | 2003-07-02 | 2006-03-16 | Scheuten Glasgroep | Procedimiento para la fabricacion de un acristalamiento contra incendios. |
| FR2859996B1 (fr) | 2003-09-19 | 2006-02-03 | Aventis Pharma Sa | Solvat acetonique du dimethoxy docetaxel et son procede de preparation |
| CN102770131A (zh) * | 2009-10-29 | 2012-11-07 | 安万特医药股份有限公司 | 卡巴他赛的新颖抗肿瘤用途 |
| CN102781237A (zh) * | 2009-11-23 | 2012-11-14 | 天蓝制药公司 | 用于传递治疗剂的基于环糊精的聚合物 |
| US20140221389A1 (en) * | 2011-09-15 | 2014-08-07 | Novartis Ag | Use of 4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-quinolin-2-one in the treatment of cancer in moderate hepatic impaired patients |
| EP3093014A1 (en) | 2015-05-13 | 2016-11-16 | Aventis Pharma S.A. | Cabazitaxel and its use for treating cancer |
-
2015
- 2015-05-13 EP EP15305720.3A patent/EP3093014A1/en not_active Ceased
-
2016
- 2016-05-12 EA EA201792502A patent/EA201792502A1/ru unknown
- 2016-05-12 WO PCT/EP2016/060759 patent/WO2016180943A1/en not_active Ceased
- 2016-05-12 KR KR1020177035580A patent/KR20180006417A/ko not_active Withdrawn
- 2016-05-12 EP EP19209255.9A patent/EP3643307A1/en not_active Withdrawn
- 2016-05-12 EP EP16721844.5A patent/EP3294285B1/en not_active Revoked
- 2016-05-12 CA CA2985408A patent/CA2985408A1/en not_active Abandoned
- 2016-05-12 JP JP2017558939A patent/JP2018516890A/ja active Pending
- 2016-05-12 US US15/153,128 patent/US20160331717A1/en not_active Abandoned
- 2016-05-12 PL PL16721844T patent/PL3294285T3/pl unknown
- 2016-05-12 PT PT167218445T patent/PT3294285T/pt unknown
- 2016-05-12 MX MX2017014463A patent/MX2017014463A/es unknown
- 2016-05-12 ES ES16721844T patent/ES2774101T3/es active Active
- 2016-05-12 AU AU2016259775A patent/AU2016259775A1/en not_active Abandoned
- 2016-05-12 CN CN201680040986.2A patent/CN108135878A/zh active Pending
- 2016-05-13 TW TW105114982A patent/TW201705950A/zh unknown
-
2017
- 2017-11-09 IL IL255541A patent/IL255541A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2774101T3 (es) | 2020-07-16 |
| EP3093014A1 (en) | 2016-11-16 |
| CA2985408A1 (en) | 2016-11-17 |
| IL255541A (en) | 2018-01-31 |
| EP3294285A1 (en) | 2018-03-21 |
| US20160331717A1 (en) | 2016-11-17 |
| WO2016180943A1 (en) | 2016-11-17 |
| EP3643307A1 (en) | 2020-04-29 |
| AU2016259775A1 (en) | 2018-01-04 |
| TW201705950A (zh) | 2017-02-16 |
| CN108135878A (zh) | 2018-06-08 |
| PT3294285T (pt) | 2020-03-06 |
| PL3294285T3 (pl) | 2020-05-18 |
| JP2018516890A (ja) | 2018-06-28 |
| EA201792502A1 (ru) | 2018-02-28 |
| EP3294285B1 (en) | 2019-12-18 |
| KR20180006417A (ko) | 2018-01-17 |
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