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MX2017008808A - Nuevas imidazo[1,2-a]quinoxalinas y derivados de las mismas para el tratamiento contra cancer. - Google Patents

Nuevas imidazo[1,2-a]quinoxalinas y derivados de las mismas para el tratamiento contra cancer.

Info

Publication number
MX2017008808A
MX2017008808A MX2017008808A MX2017008808A MX2017008808A MX 2017008808 A MX2017008808 A MX 2017008808A MX 2017008808 A MX2017008808 A MX 2017008808A MX 2017008808 A MX2017008808 A MX 2017008808A MX 2017008808 A MX2017008808 A MX 2017008808A
Authority
MX
Mexico
Prior art keywords
quinoxalinas
derivatives
same
against cancer
treatment against
Prior art date
Application number
MX2017008808A
Other languages
English (en)
Other versions
MX375551B (es
Inventor
Deleuze-Masquefa Carine
Cuq Pierre
Patinote Cindy
Antoine Bonnet Pierre-
Original Assignee
Univ Montpellier
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Montpellier filed Critical Univ Montpellier
Publication of MX2017008808A publication Critical patent/MX2017008808A/es
Publication of MX375551B publication Critical patent/MX375551B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención se relaciona con compuestos de imidazo[1,2-a]quinoxalinas para el tratamiento contra el cáncer, composiciones farmacéuticas que comprenden los compuestos, y usos terapéuticos de los mismos. La invención también se relaciona con el uso de compuestos derivados de imidazo[1,2-a]quinoxalinas para la preparación de productos medicinales para tratar el cáncer y en particular para el tratamiento de melanomas y linfomas de linfocitos T.
MX2017008808A 2014-12-31 2015-12-30 Nuevas imidazo[1,2-a]quinoxalinas y derivados de las mismas para el tratamiento contra cancer. MX375551B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR1463480A FR3031105B1 (fr) 2014-12-31 2014-12-31 Nouveaux imidazo[1,2-a]quinoxalines et derives pour le traitement des cancers
PCT/EP2015/081397 WO2016107895A1 (fr) 2014-12-31 2015-12-30 Nouveaux imidazo[1,2-a]quinoxalines et dérivés pour le traitement des cancers

Publications (2)

Publication Number Publication Date
MX2017008808A true MX2017008808A (es) 2018-03-15
MX375551B MX375551B (es) 2025-03-06

Family

ID=52692888

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017008808A MX375551B (es) 2014-12-31 2015-12-30 Nuevas imidazo[1,2-a]quinoxalinas y derivados de las mismas para el tratamiento contra cancer.

Country Status (11)

Country Link
US (1) US10689384B2 (es)
EP (1) EP3240789B1 (es)
JP (1) JP6703006B2 (es)
CN (1) CN107454900B (es)
AU (1) AU2015373422B2 (es)
BR (1) BR112017014162A2 (es)
CA (1) CA2972511A1 (es)
FR (1) FR3031105B1 (es)
MX (1) MX375551B (es)
WO (1) WO2016107895A1 (es)
ZA (1) ZA201704727B (es)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL73534A (en) 1983-11-18 1990-12-23 Riker Laboratories Inc 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
US5182386A (en) 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands
CN1046518C (zh) * 1994-09-30 1999-11-17 巴斯福股份公司 新型的带杂环取代基的咪唑并喹喔啉酮及其制备方法和应用
US6869956B2 (en) 2000-10-03 2005-03-22 Bristol-Myers Squibb Company Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
GB0211649D0 (en) * 2002-05-21 2002-07-03 Novartis Ag Organic compounds
US20060025419A1 (en) * 2004-06-25 2006-02-02 Ann Richmond Imidazoquinoxaline compound for the treatment of melanoma
CN101048404A (zh) 2004-12-27 2007-10-03 Usv有限公司 制备4-氨基-1-异丁基-1H-咪唑[4,5-c]-喹啉(咪喹莫特)的方法
MX2008009475A (es) 2006-01-23 2008-10-20 Amira Pharmaceuticals Inc Inhibidores triciclicos de 5-lipoxigenasa.
ES2376492T3 (es) 2006-03-23 2012-03-14 Novartis Ag Compuestos de imidazoquinoxalina como inmunomoduladores.
EP1972629A1 (en) * 2007-03-23 2008-09-24 Mutabilis SA New imidazolo-heteroaryl derivatives with antibacterial properties
FR2921927B1 (fr) * 2007-10-03 2012-10-12 Univ De Montpellier 1 Imidazo°1,2-a!quinoxalines et derives pour le traitement des cancers
US20100120762A1 (en) * 2008-11-07 2010-05-13 Wyeth Triazine derivatives as inhibitors of phosphodiesterases
WO2010124826A1 (en) * 2009-04-29 2010-11-04 Bayer Schering Pharma Aktiengesellschaft Substituted imidazoquinoxalines

Also Published As

Publication number Publication date
CN107454900A (zh) 2017-12-08
AU2015373422A8 (en) 2017-08-24
JP6703006B2 (ja) 2020-06-03
AU2015373422B2 (en) 2020-07-09
JP2018502914A (ja) 2018-02-01
CA2972511A1 (fr) 2016-07-07
AU2015373422A1 (en) 2017-08-17
MX375551B (es) 2025-03-06
FR3031105A1 (fr) 2016-07-01
US20180016278A1 (en) 2018-01-18
CN107454900B (zh) 2020-08-07
EP3240789A1 (fr) 2017-11-08
EP3240789B1 (fr) 2020-07-29
US10689384B2 (en) 2020-06-23
BR112017014162A2 (pt) 2018-01-02
FR3031105B1 (fr) 2018-04-06
ZA201704727B (en) 2021-05-26
WO2016107895A1 (fr) 2016-07-07

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