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MX2016014119A - Proceso para preparar cicloserinas sustituidas. - Google Patents

Proceso para preparar cicloserinas sustituidas.

Info

Publication number
MX2016014119A
MX2016014119A MX2016014119A MX2016014119A MX2016014119A MX 2016014119 A MX2016014119 A MX 2016014119A MX 2016014119 A MX2016014119 A MX 2016014119A MX 2016014119 A MX2016014119 A MX 2016014119A MX 2016014119 A MX2016014119 A MX 2016014119A
Authority
MX
Mexico
Prior art keywords
substituted
aryl
preparation
compounds
c4alkylene
Prior art date
Application number
MX2016014119A
Other languages
English (en)
Other versions
MX388328B (es
Inventor
Smits Helmars
Smejkal Tomas
LOTHSCHUETZ Christian
Terinek Miroslav
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of MX2016014119A publication Critical patent/MX2016014119A/es
Publication of MX388328B publication Critical patent/MX388328B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/04—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
    • C07C259/06—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/12—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La presente invención se refiere a procesos para preparar compuestos de tipo cicloserina sustituida de fórmula (I) (ver Fórmula) donde R1 es alquilo C1-C8, haloalquilo C1-C8, cicloalquilo C3-C6, arilo o arilo sustituido con de uno a cinco R11, o aril-(alquileno C1-C4) o aril- (alquileno C1-C4) sustituido con de uno a cinco R11; y cada R11 es independientemente alquilo C1-C4, haloalquilo C1-C4, alcoxi C1-C4, haloalcoxi C1-C4, ciano o halógeno. La invención también se refiere a intermedios producidos mediante los procesos. Los compuestos de fórmula (I) son intermedios útiles para producir compuestos en los campos agrícola y farmacéutico.
MX2016014119A 2014-04-30 2015-04-30 Proceso para preparar cicloserinas sustituidas. MX388328B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14166654 2014-04-30
PCT/EP2015/059612 WO2015166094A1 (en) 2014-04-30 2015-04-30 Process for the preparation of substituted cycloserines

Publications (2)

Publication Number Publication Date
MX2016014119A true MX2016014119A (es) 2017-02-09
MX388328B MX388328B (es) 2025-03-19

Family

ID=50693448

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2016014119A MX388328B (es) 2014-04-30 2015-04-30 Proceso para preparar cicloserinas sustituidas.
MX2021011971A MX2021011971A (es) 2014-04-30 2016-10-27 Proceso para preparar cicloserinas sustituidas.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2021011971A MX2021011971A (es) 2014-04-30 2016-10-27 Proceso para preparar cicloserinas sustituidas.

Country Status (13)

Country Link
US (2) US9643938B2 (es)
EP (1) EP3137449B1 (es)
JP (1) JP6523334B2 (es)
CN (3) CN114031572B (es)
BR (2) BR122021004312B1 (es)
DK (1) DK3137449T3 (es)
ES (1) ES2774363T3 (es)
HU (1) HUE049170T2 (es)
IL (1) IL248267B (es)
MX (2) MX388328B (es)
PL (1) PL3137449T3 (es)
SI (1) SI3137449T1 (es)
WO (1) WO2015166094A1 (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3137449T3 (pl) * 2014-04-30 2020-07-27 Syngenta Participations Ag Sposób wytwarzania podstawionych cykloseryn
MX2022007455A (es) 2019-12-18 2022-08-15 Elanco Tiergesundheit Ag Derivados de isoxazolina como plaguicidas.
CN114014776B (zh) * 2021-12-09 2024-03-12 西安鸿钧睿泽新材料科技有限公司 一种具有低全球变暖潜值的化合物、制备方法及其应用
CA3253813A1 (en) 2022-05-30 2023-12-07 Syngenta Crop Protection Ag PROCESS FOR PREPARATION OF 2-OXAZOLIDINONES SUBSTITUTED AT POSITION 4
WO2024033374A1 (en) 2022-08-11 2024-02-15 Syngenta Crop Protection Ag Novel arylcarboxamide or arylthioamide compounds
WO2024089216A1 (en) 2022-10-27 2024-05-02 Syngenta Crop Protection Ag Novel sulfur-containing heteroaryl carboxamide compounds
JP2026500298A (ja) 2022-12-15 2026-01-06 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト 殺有害生物剤として有用である新規な二環式カルボキサミド化合物
IL322407A (en) 2023-02-24 2025-09-01 Syngenta Crop Protection Ag Process for preparing isoxazoline derivatives
WO2026021962A1 (en) 2024-07-26 2026-01-29 Basf Se Process for the preparation of an aqueous solution comprising n-alkylhydroxylamine

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB799066A (en) * 1955-11-17 1958-07-30 Hoffmann La Roche Process for the manufacture of isoxazolidone compounds
CH488719A (de) * 1967-06-26 1970-04-15 Eprova Ag Verfahren zur Herstellung von Cycloserin (D-4-Amino-3-isoxazolidinon)
JPS5714337B2 (es) 1973-02-23 1982-03-24
WO1996030381A1 (en) 1995-03-28 1996-10-03 Novo Nordisk A/S Immunosuppressive agents
WO2008153942A1 (en) * 2007-06-06 2008-12-18 Xcovery, Inc. Kinase inhibitor compounds
EP2172462A4 (en) * 2007-06-27 2010-12-15 Nissan Chemical Ind Ltd METHOD FOR PRODUCING A 3-HYDROXYPROPAN-1-ON COMPOUND, METHOD FOR PRODUCING A 2-PROPENE-1-ON COMPOUND, AND METHOD FOR PRODUCING AN ISOXAZOLINE COMPOUND
TWI487486B (zh) * 2009-12-01 2015-06-11 Syngenta Participations Ag 以異唑啉衍生物為主之殺蟲化合物
KR20120131646A (ko) 2011-05-26 2012-12-05 주식회사 참조아 이속사졸리디논 유도체인 ｄ-시클로세린의 제조방법
AR086587A1 (es) * 2011-05-31 2014-01-08 Syngenta Participations Ag Compuestos insecticidas
PL3137449T3 (pl) * 2014-04-30 2020-07-27 Syngenta Participations Ag Sposób wytwarzania podstawionych cykloseryn

Also Published As

Publication number Publication date
PL3137449T3 (pl) 2020-07-27
EP3137449A1 (en) 2017-03-08
IL248267A0 (en) 2016-11-30
US9815803B2 (en) 2017-11-14
DK3137449T3 (da) 2020-03-02
HUE049170T2 (hu) 2020-09-28
IL248267B (en) 2019-07-31
CN114031572A (zh) 2022-02-11
CN114031572B (zh) 2025-07-08
BR112016025076B1 (pt) 2022-03-03
ES2774363T3 (es) 2020-07-20
JP2017518272A (ja) 2017-07-06
EP3137449B1 (en) 2019-12-18
CN108822053A (zh) 2018-11-16
CN106255681B (zh) 2019-11-22
SI3137449T1 (sl) 2020-04-30
BR122021004312B1 (pt) 2022-02-08
US20170044116A1 (en) 2017-02-16
US9643938B2 (en) 2017-05-09
WO2015166094A1 (en) 2015-11-05
JP6523334B2 (ja) 2019-05-29
BR112016025076A2 (pt) 2018-07-10
MX2021011971A (es) 2021-11-03
CN106255681A (zh) 2016-12-21
MX388328B (es) 2025-03-19
US20170204072A1 (en) 2017-07-20

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