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MX2016013245A - Regimen de dosificacion de liberacion inmediata de moduladores s1p. - Google Patents

Regimen de dosificacion de liberacion inmediata de moduladores s1p.

Info

Publication number
MX2016013245A
MX2016013245A MX2016013245A MX2016013245A MX2016013245A MX 2016013245 A MX2016013245 A MX 2016013245A MX 2016013245 A MX2016013245 A MX 2016013245A MX 2016013245 A MX2016013245 A MX 2016013245A MX 2016013245 A MX2016013245 A MX 2016013245A
Authority
MX
Mexico
Prior art keywords
immediate release
release dosage
modulator
dosage regimen
siponimod
Prior art date
Application number
MX2016013245A
Other languages
English (en)
Inventor
Wallstroem Erik
Legangneux Eric
Michel Rene Bouillot Philippe
Reynaud Emeric
Dehlke Frank
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52988364&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2016013245(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2016013245A publication Critical patent/MX2016013245A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere al siponimod (BAF312) para uso en el tratamiento de una enfermedad autoinmune, donde una forma de dosificación de liberación inmediata se administra una vez al día a un paciente como régimen de mantenimiento y donde el paciente ha sido sometido previamente a un régimen de ajuste de dosis específico con siponimod.
MX2016013245A 2014-04-10 2015-04-08 Regimen de dosificacion de liberacion inmediata de moduladores s1p. MX2016013245A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201461977816P 2014-04-10 2014-04-10
PCT/IB2015/052550 WO2015155709A1 (en) 2014-04-10 2015-04-08 S1p modulator immediate release dosage regimen

Publications (1)

Publication Number Publication Date
MX2016013245A true MX2016013245A (es) 2017-01-16

Family

ID=52988364

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016013245A MX2016013245A (es) 2014-04-10 2015-04-08 Regimen de dosificacion de liberacion inmediata de moduladores s1p.

Country Status (16)

Country Link
US (4) US20170027907A1 (es)
EP (3) EP4074312A1 (es)
JP (1) JP6674903B2 (es)
KR (2) KR20220156981A (es)
CN (2) CN106456552A (es)
AU (2) AU2015246036A1 (es)
CA (1) CA2943598C (es)
CL (1) CL2016002562A1 (es)
IL (2) IL305337A (es)
MX (1) MX2016013245A (es)
PH (1) PH12016501965A1 (es)
RU (2) RU2715734C2 (es)
SG (1) SG11201607894RA (es)
TW (1) TW201622721A (es)
WO (1) WO2015155709A1 (es)
ZA (1) ZA201606519B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO2699580T3 (es) 2014-01-24 2018-02-24
SG11201607894RA (en) * 2014-04-10 2016-10-28 Novartis Ag S1p modulator immediate release dosage regimen
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
US11434200B2 (en) 2017-03-09 2022-09-06 Novartis Ag Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
AU2018341154A1 (en) * 2017-09-29 2020-03-12 Novartis Ag Dosing regimen of siponimod
AU2018343239A1 (en) * 2017-09-29 2020-03-12 Novartis Ag Dosing regimen of siponimod
MA52424B1 (fr) 2018-03-01 2025-04-30 Astrazeneca Ab Compositions pharmaceutiques comprenant du (2s)--((1s)-1-cyano-2-[4-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)phenyl]ethyl)-1,4-oxazepane-2-carboxamide
CA3106269A1 (en) 2018-07-17 2020-01-23 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis
CN109908095A (zh) * 2019-04-08 2019-06-21 肇庆学院 一种西尼莫德片剂及制备方法
KR20220093330A (ko) 2019-10-31 2022-07-05 이도르시아 파마슈티컬스 리미티드 Cxcr7 안타고니스트와 s1p1 수용체 조절인자의 조합
US11135197B2 (en) 2020-02-07 2021-10-05 Argentum Pharmaceuticals Llc Dosage regimen of an S1P receptor modulator
AU2024206233A1 (en) 2023-01-06 2025-08-21 Insmed Incorporated Novel, reversible dpp1 inhibitors and uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2747437C (en) * 2008-12-18 2018-08-21 Novartis Ag Hemifumarate salt of 1-[4-[1-(4-cyclohexyl-3-trifluoromethyl-benzyloxyimino)-ethyl]-2-ethyl-benzyl]-a zetidine-3-carboxylic acid
SI2379067T1 (sl) * 2008-12-22 2016-01-29 Novartis Ag Režim odmerjanja fingolimoda za zdravljenje multiple skleroze
KR101660555B1 (ko) * 2008-12-22 2016-09-27 노파르티스 아게 Ｓ１ｐ 수용체 효능제의 투여 요법
WO2011041146A2 (en) * 2009-09-29 2011-04-07 Novartis Ag Dosage regimen of an s1p receptor modulator
HRP20191842T1 (hr) * 2011-01-07 2019-12-27 Novartis Ag Formulacije imunosupresiva
WO2012095853A1 (en) * 2011-01-10 2012-07-19 Novartis Pharma Ag Modified release formulations comprising sip receptor modulators
SG11201401065RA (en) * 2011-10-21 2014-09-26 Novartis Ag Dosage regimen for an s1p receptor modulator or agonist
SG11201607894RA (en) * 2014-04-10 2016-10-28 Novartis Ag S1p modulator immediate release dosage regimen

Also Published As

Publication number Publication date
ZA201606519B (en) 2017-11-29
CN106456552A (zh) 2017-02-22
US20250041266A1 (en) 2025-02-06
IL247986A0 (en) 2016-11-30
KR20220156981A (ko) 2022-11-28
TW201622721A (zh) 2016-07-01
RU2016143979A (ru) 2018-05-14
KR20160141841A (ko) 2016-12-09
AU2020203107A1 (en) 2020-05-28
SG11201607894RA (en) 2016-10-28
IL305337A (en) 2023-10-01
WO2015155709A1 (en) 2015-10-15
CN116650467A (zh) 2023-08-29
EP4074312A1 (en) 2022-10-19
JP6674903B2 (ja) 2020-04-01
CA2943598A1 (en) 2015-10-15
US20220016076A1 (en) 2022-01-20
CA2943598C (en) 2023-03-07
RU2020107732A (ru) 2020-03-30
RU2715734C2 (ru) 2020-03-03
RU2016143979A3 (es) 2018-11-12
EP3129020A1 (en) 2017-02-15
PH12016501965A1 (en) 2017-01-09
US20170027907A1 (en) 2017-02-02
EP3831378A1 (en) 2021-06-09
AU2015246036A1 (en) 2016-10-13
US20190054065A1 (en) 2019-02-21
CL2016002562A1 (es) 2017-07-28
JP2017510607A (ja) 2017-04-13
AU2020203107B2 (en) 2021-10-21

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