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MX2016006464A - Composicion farmaceutica de una combinacion de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor. - Google Patents

Composicion farmaceutica de una combinacion de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor.

Info

Publication number
MX2016006464A
MX2016006464A MX2016006464A MX2016006464A MX2016006464A MX 2016006464 A MX2016006464 A MX 2016006464A MX 2016006464 A MX2016006464 A MX 2016006464A MX 2016006464 A MX2016006464 A MX 2016006464A MX 2016006464 A MX2016006464 A MX 2016006464A
Authority
MX
Mexico
Prior art keywords
etoricoxib
tramadol
hydrochloride
pain
treatment
Prior art date
Application number
MX2016006464A
Other languages
English (en)
Inventor
Daniel Walls Flores Oliver
Astrid Salto Rivera Reyna
Rodríguez Hernández Ramón
Original Assignee
Laboratorios Liomont S A De C V
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratorios Liomont S A De C V filed Critical Laboratorios Liomont S A De C V
Priority to MX2016006464A priority Critical patent/MX2016006464A/es
Priority to EP17798843.3A priority patent/EP3338771A4/en
Priority to PCT/IB2017/052775 priority patent/WO2017199140A1/es
Priority to CA2997600A priority patent/CA2997600A1/en
Priority to US16/008,277 priority patent/US20190060295A1/en
Publication of MX2016006464A publication Critical patent/MX2016006464A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4833Encapsulating processes; Filling of capsules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

La presente invención consiste en un proceso y composición farmacéutica de una combinación de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor, cuyo proceso de obtención está dado a partir de dos activos la cual consiste en gránulos y/o multiparticulados con clorhidrato de tramadol y gránulos y/o multiparticulados con etoricoxib los cuales pueden estar contenidos en una mezcla de polvos, o comprimidos en una tableta bicapa con o sin recubrimiento o en una capsula como granulados y/o tabletas con o sin recubrimiento.
MX2016006464A 2016-05-18 2016-05-18 Composicion farmaceutica de una combinacion de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor. MX2016006464A (es)

Priority Applications (5)

Application Number Priority Date Filing Date Title
MX2016006464A MX2016006464A (es) 2016-05-18 2016-05-18 Composicion farmaceutica de una combinacion de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor.
EP17798843.3A EP3338771A4 (en) 2016-05-18 2017-05-11 PHARMACEUTICAL COMPOSITION COMPRISING A COMBINATION OF TRAMADOL-ETORICOXIB CHLORHYDRATE FOR THE TREATMENT OF PAIN
PCT/IB2017/052775 WO2017199140A1 (es) 2016-05-18 2017-05-11 Composición farmacéutica de una combinación de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor
CA2997600A CA2997600A1 (en) 2016-05-18 2017-05-11 Pharmaceutical composition of a combination of tramadol-etoricoxib hydrochloride for the treatment of pain
US16/008,277 US20190060295A1 (en) 2016-05-18 2017-05-11 Pharmaceutical composition of a combination of tramadol-etoricoxib hydrochloride for the treatment of pain

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
MX2016006464A MX2016006464A (es) 2016-05-18 2016-05-18 Composicion farmaceutica de una combinacion de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor.

Publications (1)

Publication Number Publication Date
MX2016006464A true MX2016006464A (es) 2017-11-17

Family

ID=60325762

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016006464A MX2016006464A (es) 2016-05-18 2016-05-18 Composicion farmaceutica de una combinacion de clorhidrato de tramadol-etoricoxib para el tratamiento del dolor.

Country Status (5)

Country Link
US (1) US20190060295A1 (es)
EP (1) EP3338771A4 (es)
CA (1) CA2997600A1 (es)
MX (1) MX2016006464A (es)
WO (1) WO2017199140A1 (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4585207A1 (en) 2024-01-12 2025-07-16 Laboratorios Silanes, S.A. de C.V. Synergic and stable pharmaceutical composition of an nsaid and an opioid analgesic for pain and inflammation

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2017009660A (es) * 2017-07-26 2017-11-23 Laboratorios Liomont S A De C V Composicion farmaceutica con un rango de relacion entre el clorhidrato de tramadol y el etoricoxib para su administracion para el tratamiento del dolor.
MX2018013070A (es) 2017-12-29 2019-10-15 Gruenenthal Gmbh Combinación farmacéutica que comprende clorhidrato de tramadol de liberación extendida y etoricoxib de liberación inmediata, y su uso para el tratamiento del dolor.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000051685A1 (en) * 1999-03-01 2000-09-08 Ortho-Mcneil Pharmaceutical, Inc. Composition comprising a tramadol material and a selective cox-2 inhibitor drug
US20080026054A1 (en) * 2007-04-27 2008-01-31 Nectid Inc. Novel anelgesic combination
EP2177215A1 (en) * 2008-10-17 2010-04-21 Laboratorios Del. Dr. Esteve, S.A. Co-crystals of tramadol and NSAIDs
EP2281558A1 (en) * 2009-08-06 2011-02-09 Laboratorios Del. Dr. Esteve, S.A. Pharmaceutical compounds of O-Desmethyl-Tramadol and COX-inhibitors
EP2311446A1 (en) * 2009-10-16 2011-04-20 Laboratorios Del. Dr. Esteve, S.A. Compositions comprising Tramadol and Celecoxib in the treatment of pain
SG178835A1 (en) * 2009-10-16 2012-05-30 Esteve Labor Dr Co-crystals of tramadol and coxibs
HUE033525T2 (en) * 2012-08-27 2017-12-28 Cadila Healthcare Ltd Pharmaceuticals containing Etoricoxib

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4585207A1 (en) 2024-01-12 2025-07-16 Laboratorios Silanes, S.A. de C.V. Synergic and stable pharmaceutical composition of an nsaid and an opioid analgesic for pain and inflammation

Also Published As

Publication number Publication date
US20190060295A1 (en) 2019-02-28
EP3338771A4 (en) 2019-05-08
EP3338771A1 (en) 2018-06-27
CA2997600A1 (en) 2017-11-23
WO2017199140A1 (es) 2017-11-23

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