[go: up one dir, main page]

MX2014007398A - Derivado de 2,4-diamina-pirimidina como inhibidores de serina/treonina quinasa. - Google Patents

Derivado de 2,4-diamina-pirimidina como inhibidores de serina/treonina quinasa.

Info

Publication number
MX2014007398A
MX2014007398A MX2014007398A MX2014007398A MX2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A MX 2014007398 A MX2014007398 A MX 2014007398A
Authority
MX
Mexico
Prior art keywords
serine
diamine
kinase inhibitors
threonine kinase
pyrimidine derivative
Prior art date
Application number
MX2014007398A
Other languages
English (en)
Inventor
Wendy Lee
Ignacio Aliagas-Martin
Simon Mathieu
Joachim Rudolph
James John Crawford
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority claimed from PCT/EP2012/076531 external-priority patent/WO2013092940A1/en
Publication of MX2014007398A publication Critical patent/MX2014007398A/es

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Compuestos que tienen la fórmula I en donde A, R1a, R1b, R2, R3, R4, R5, R6, R7, R8, Ra, Rb, X1., X2, X3 y n son como se definió aquí, son inhibidores de PAK1. También se describen composiciones y métodos para tratar cáncer y desórdenes hiperproliferativos. (ver Fórmula).
MX2014007398A 2011-12-22 2012-12-21 Derivado de 2,4-diamina-pirimidina como inhibidores de serina/treonina quinasa. MX2014007398A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP61579227 2011-12-22
PCT/EP2012/076531 WO2013092940A1 (en) 2011-12-22 2012-12-21 2, 4-diamine-pyrimidine derivative as serine/threonine kinase inhibitors

Publications (1)

Publication Number Publication Date
MX2014007398A true MX2014007398A (es) 2014-08-08

Family

ID=52130938

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014007398A MX2014007398A (es) 2011-12-22 2012-12-21 Derivado de 2,4-diamina-pirimidina como inhibidores de serina/treonina quinasa.

Country Status (1)

Country Link
MX (1) MX2014007398A (es)

Similar Documents

Publication Publication Date Title
MX2014002208A (es) Inhibidores de serina/treonina quinasa.
MX340756B (es) Compuestos de quinazolina como inhibidores de serina/treonina quinasa.
MX341456B (es) Amino-quinolinas como inhibidores de cinasa.
PH12017502141A1 (en) Compounds and their methods of use
MX339873B (es) Inhibidores de serina/treonina cinasa.
MX2015007097A (es) Nuevas fenil-piridinas/pirazinas bi-anulares para el tratamiento de cancer.
PH12014500883A1 (en) Uracil derivatives as axl and c-met kinase inhibitors
MX358376B (es) Nuevos derivados dihidroquinolina-2-ona.
PH12014501365A1 (en) Compounds
MX2013011329A (es) Combinaciones de compuestos inhibidores de akt y erlotinib y metodos de uso.
MX2015001720A (es) Hetero-azepinonas sustituidas.
MX2014014531A (es) Derivados de aminoquinazolina y piridopirimidina.
PH12014500373A1 (en) Amino quinazolines as kinase inhibitors
HK1210174A1 (en) Serine/threonine kinase inhibitors for the treatment of hyperproliferative|diseases
MX361499B (es) Baricitinib deuterado.
PH12014500814A1 (en) New aryl-quinoline derivatives
PH12016501071B1 (en) Serine/threonine kinase inhibitors
PH12015500363A1 (en) Prodrugs of amino quinazoline kinase inhibitor
PH12015500345A1 (en) Amino-quinolines as kinase inhibitors
PH12015501038A1 (en) Inhibitors of iap
GB201209587D0 (en) Therapeutic compounds
GEP201706687B (en) Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
CR20140495A (es) 5-amino[1,4]thiazines como inhibidores de bace1
MX359399B (es) Inhibidores de 17alfa-hidroxilasa/c17-20-liasa.
IN2015DN02588A (es)