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MX2014001885A - Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona. - Google Patents

Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona.

Info

Publication number
MX2014001885A
MX2014001885A MX2014001885A MX2014001885A MX2014001885A MX 2014001885 A MX2014001885 A MX 2014001885A MX 2014001885 A MX2014001885 A MX 2014001885A MX 2014001885 A MX2014001885 A MX 2014001885A MX 2014001885 A MX2014001885 A MX 2014001885A
Authority
MX
Mexico
Prior art keywords
dihydropyrimidin
imino
fluoro
derivatives
substituted
Prior art date
Application number
MX2014001885A
Other languages
English (en)
Other versions
MX354021B (es
Inventor
Timothy A Boebel
Beth Lorsbach
John W Owen
Michael T Sullenberger
Jeffery D Webster
Chenglin Yao
Chris V Galliford
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47713076&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2014001885(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of MX2014001885A publication Critical patent/MX2014001885A/es
Publication of MX354021B publication Critical patent/MX354021B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)

Abstract

La presente descripción se refiere al campo de las 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidina-2(1H)onas y sus derivados y al uso de estos compuestos como fungicidas.
MX2014001885A 2011-08-17 2012-08-15 Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona. MX354021B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161524506P 2011-08-17 2011-08-17
PCT/US2012/050930 WO2013025795A1 (en) 2011-08-17 2012-08-15 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives

Publications (2)

Publication Number Publication Date
MX2014001885A true MX2014001885A (es) 2014-05-30
MX354021B MX354021B (es) 2018-02-08

Family

ID=47713076

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014001885A MX354021B (es) 2011-08-17 2012-08-15 Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona.

Country Status (30)

Country Link
US (1) US8658660B2 (es)
EP (1) EP2775842B1 (es)
JP (3) JP6128658B2 (es)
KR (1) KR102012992B1 (es)
CN (2) CN106977462B (es)
AR (1) AR087549A1 (es)
BR (1) BR112014003587B1 (es)
CA (1) CA2844497C (es)
CL (1) CL2014000352A1 (es)
CO (1) CO6910204A2 (es)
CR (1) CR20140058A (es)
DK (1) DK2775842T3 (es)
EC (1) ECSP14013251A (es)
ES (1) ES2646725T3 (es)
GT (1) GT201400023A (es)
HR (1) HRP20171776T1 (es)
HU (1) HUE035248T2 (es)
IL (1) IL230981A (es)
LT (1) LT2775842T (es)
ME (1) ME02924B (es)
MX (1) MX354021B (es)
NO (1) NO2874589T3 (es)
PL (1) PL2775842T3 (es)
PT (1) PT2775842T (es)
RS (1) RS56609B1 (es)
RU (1) RU2613451C2 (es)
SI (1) SI2775842T1 (es)
UA (1) UA113062C2 (es)
WO (1) WO2013025795A1 (es)
ZA (1) ZA201400875B (es)

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JP6128658B2 (ja) * 2011-08-17 2017-05-17 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−（置換）−３，４−ジヒドロピリミジン−２−（１ｈ）−オン誘導体
JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体
DK2938194T3 (da) 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
CN103819412B (zh) * 2013-12-11 2016-02-03 浙江先锋科技股份有限公司 一种5-氟胞嘧啶的制备方法
WO2015103144A1 (en) * 2013-12-31 2015-07-09 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
KR102805798B1 (ko) 2014-12-30 2025-05-15 코르테바 애그리사이언스 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
TWI774762B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺作為一種殺真菌劑以防治蔬菜中植物病原性真菌的用途
TWI801380B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 一種非環狀吡啶醯胺化合物作為殺真菌劑以防治在果園、葡萄藤園及農園作物中的植物病原性真菌之用途
TWI774761B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TWI801381B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺化合物作為殺真菌劑以防治行栽作物中具植物病原性的真菌之用途
TWI774760B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於蔬菜中的真菌防治之協同性混合物
TW201842851A (zh) * 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CN118515619A (zh) 2017-07-17 2024-08-20 阿达玛克西姆股份有限公司 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物
CN109053553A (zh) * 2018-10-16 2018-12-21 山东省农药科学研究院 杀虫剂氟啶虫胺腈中间体3-[1-(甲硫基)乙基]-6(三氟甲基)吡啶的合成方法
KR20210136961A (ko) 2018-11-05 2021-11-17 아다마 마켓심 리미티드 5-플루오로-4-이미노-3-메틸-1-토실-3,4-디하이드로피리미딘-2-온을 포함하는 혼합물들과 조성물들 및 이들을 사용하는 방법들
JP7353012B2 (ja) 2019-08-22 2023-09-29 フジアン ヨンジン テクノロジー カンパニー リミテッド 直接フッ素化によるフルオロベンゼンの製造プロセス
CN114599639A (zh) 2019-09-23 2022-06-07 阿达玛马克西姆有限公司 用于制备5-(氟-4-亚氨基-3-甲基)-1-甲苯磺酰基-3,4-二氢嘧啶-(1h)-酮的方法
US12281076B2 (en) 2019-10-18 2025-04-22 Corteva Agriscience Llc Process for synthesis of picolinamides
WO2021181274A1 (en) * 2020-03-09 2021-09-16 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
IL311455A (en) * 2021-09-15 2024-05-01 Adama Makhteshim Ltd Method for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-H1-pyrimidin-2-one
WO2025248515A1 (en) 2024-05-26 2025-12-04 Adama Makhteshim Ltd. Fungicidal mixtures and composition comprising thereof

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Also Published As

Publication number Publication date
ES2646725T3 (es) 2017-12-15
HUE035248T2 (en) 2018-05-02
DK2775842T3 (en) 2017-12-18
AU2012296629A8 (en) 2016-06-16
CA2844497C (en) 2021-03-02
ZA201400875B (en) 2015-04-29
BR112014003587B1 (pt) 2021-04-13
US20130045984A1 (en) 2013-02-21
RU2613451C2 (ru) 2017-03-16
JP2017125060A (ja) 2017-07-20
BR112014003587A2 (pt) 2017-03-14
SI2775842T1 (en) 2018-01-31
CN103874413B (zh) 2017-03-08
IL230981A (en) 2017-10-31
CN106977462B (zh) 2020-04-28
EP2775842A4 (en) 2015-04-15
JP6901462B2 (ja) 2021-07-14
AU2012296629B2 (en) 2016-02-11
AU2012296629A1 (en) 2014-02-20
NO2874589T3 (es) 2018-02-03
JP2019088283A (ja) 2019-06-13
RU2014110049A (ru) 2015-09-27
GT201400023A (es) 2015-02-27
CO6910204A2 (es) 2014-03-31
JP2014524440A (ja) 2014-09-22
PL2775842T3 (pl) 2018-02-28
IL230981A0 (en) 2014-03-31
ME02924B (me) 2018-04-20
HK1199177A1 (en) 2015-06-26
ECSP14013251A (es) 2014-04-30
HRP20171776T1 (hr) 2018-01-26
NZ620537A (en) 2016-11-25
CL2014000352A1 (es) 2014-07-25
RS56609B1 (sr) 2018-02-28
BR112014003587A8 (pt) 2017-07-11
PT2775842T (pt) 2017-11-15
MX354021B (es) 2018-02-08
CN106977462A (zh) 2017-07-25
WO2013025795A1 (en) 2013-02-21
EP2775842A1 (en) 2014-09-17
US8658660B2 (en) 2014-02-25
UA113062C2 (xx) 2016-12-12
KR102012992B1 (ko) 2019-08-21
JP6128658B2 (ja) 2017-05-17
KR20140057605A (ko) 2014-05-13
CA2844497A1 (en) 2013-02-21
CR20140058A (es) 2014-03-20
LT2775842T (lt) 2017-12-11
EP2775842B1 (en) 2017-10-04
AR087549A1 (es) 2014-04-03
CN103874413A (zh) 2014-06-18

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