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MX2011008634A - Derivados de aminotetralina composiciones farmaceuticas que los contienen y su uso en terapia. - Google Patents

Derivados de aminotetralina composiciones farmaceuticas que los contienen y su uso en terapia.

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Publication number
MX2011008634A
MX2011008634A MX2011008634A MX2011008634A MX2011008634A MX 2011008634 A MX2011008634 A MX 2011008634A MX 2011008634 A MX2011008634 A MX 2011008634A MX 2011008634 A MX2011008634 A MX 2011008634A MX 2011008634 A MX2011008634 A MX 2011008634A
Authority
MX
Mexico
Prior art keywords
pharmaceutical compositions
aminotetraline derivatives
therapy
compositions containing
aminotetraline
Prior art date
Application number
MX2011008634A
Other languages
English (en)
Inventor
Wilfried Hornberger
Wilhelm Amberg
Udo Lange
Michael Ochse
Mario Mezler
Andreas Kling
Berthold Behl
Charles Hutchins
Original Assignee
Abbott Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co Kg filed Critical Abbott Gmbh & Co Kg
Publication of MX2011008634A publication Critical patent/MX2011008634A/es

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    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/05—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by nitrogen atoms, not being part of nitro or nitroso groups
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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    • C07C233/19—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a saturated carbon skeleton containing rings
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Abstract

La presente invención se refiere a derivados de aminotetralina de fórmula (I) o una sal fisiológicamente aceptable de lo mismo. La invención se refiere a composiciones farmacéuticas que comprenden tales derivados de aminotetralina, y el uso de tales derivados de aminotetralina con propósitos terapéuticos. Los derivados de aminotetralina son inhibidores de GlyT1.
MX2011008634A 2009-02-16 2010-02-16 Derivados de aminotetralina composiciones farmaceuticas que los contienen y su uso en terapia. MX2011008634A (es)

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