[go: up one dir, main page]

MX2010010017A - Derivados de guanidina lineales y ciclicos, metodo de preparacion y sus usos. - Google Patents

Derivados de guanidina lineales y ciclicos, metodo de preparacion y sus usos.

Info

Publication number
MX2010010017A
MX2010010017A MX2010010017A MX2010010017A MX2010010017A MX 2010010017 A MX2010010017 A MX 2010010017A MX 2010010017 A MX2010010017 A MX 2010010017A MX 2010010017 A MX2010010017 A MX 2010010017A MX 2010010017 A MX2010010017 A MX 2010010017A
Authority
MX
Mexico
Prior art keywords
linear
preparation
guanidine derivatives
cyclic guanidine
cyclic
Prior art date
Application number
MX2010010017A
Other languages
English (en)
Inventor
Maurizio Botta
Francesco Raffi
Paolo Visca
Original Assignee
Univ Siena
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Siena filed Critical Univ Siena
Publication of MX2010010017A publication Critical patent/MX2010010017A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D255/00—Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D249/00 - C07D253/00
    • C07D255/02—Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D249/00 - C07D253/00 not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/04—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
    • C07C279/12—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D259/00—Heterocyclic compounds containing rings having more than four nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

La presente invención se refiere a derivados de guanidina lineales y cíclicos, método de preparación y su uso, a composiciones farmacéuticas que serán utilizadas como agentes antifúngicos, particularmente contra especies Candida.
MX2010010017A 2008-03-13 2009-03-12 Derivados de guanidina lineales y ciclicos, metodo de preparacion y sus usos. MX2010010017A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3616508P 2008-03-13 2008-03-13
PCT/IB2009/051032 WO2009113033A2 (en) 2008-03-13 2009-03-12 Linear and cyclic guanidine derivatives, method of preparation and uses thereof

Publications (1)

Publication Number Publication Date
MX2010010017A true MX2010010017A (es) 2010-10-07

Family

ID=40622063

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010010017A MX2010010017A (es) 2008-03-13 2009-03-12 Derivados de guanidina lineales y ciclicos, metodo de preparacion y sus usos.

Country Status (13)

Country Link
US (1) US8685953B2 (es)
EP (1) EP2274290B1 (es)
JP (1) JP5733988B2 (es)
CN (1) CN101977901B (es)
AU (1) AU2009223204B2 (es)
BR (1) BRPI0908953A2 (es)
DK (1) DK2274290T3 (es)
EA (1) EA018926B1 (es)
ES (1) ES2396288T3 (es)
MX (1) MX2010010017A (es)
PL (1) PL2274290T3 (es)
PT (1) PT2274290E (es)
WO (1) WO2009113033A2 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105612147B (zh) * 2013-06-18 2018-06-05 小天鹅生物科学有限公司 大环脒基脲衍生物，其制备方法及其作为几丁质酶抑制剂的应用
JP6378179B2 (ja) 2013-07-03 2018-08-22 株式会社新日本科学 新規化合物，有機カチオントランスポーター３の検出剤及び活性阻害剤
WO2016055644A1 (en) 2014-10-10 2016-04-14 Lead Discovery Siena S.R.L. Linear guanidine derivatives, methods of preparation and uses thereof
EP3854789A1 (en) * 2020-01-22 2021-07-28 Cygnet Biosciences B.V. Macrocyclic compounds useful as chitinase inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1114155A (en) * 1964-08-24 1968-05-15 Evans Medical Ltd Guanidino derivatives
US3988370A (en) * 1970-10-08 1976-10-26 Sterling Drug Inc. Amidinoureas

Also Published As

Publication number Publication date
ES2396288T3 (es) 2013-02-20
AU2009223204B2 (en) 2014-07-24
JP2011513477A (ja) 2011-04-28
US20110039854A1 (en) 2011-02-17
WO2009113033A3 (en) 2009-12-30
AU2009223204A1 (en) 2009-09-17
DK2274290T3 (da) 2013-01-14
JP5733988B2 (ja) 2015-06-10
EP2274290B1 (en) 2012-09-26
CN101977901B (zh) 2015-04-01
BRPI0908953A2 (pt) 2016-06-07
EP2274290A2 (en) 2011-01-19
EA201071072A1 (ru) 2011-04-29
EA018926B1 (ru) 2013-11-29
CN101977901A (zh) 2011-02-16
US8685953B2 (en) 2014-04-01
PL2274290T3 (pl) 2013-03-29
WO2009113033A2 (en) 2009-09-17
PT2274290E (pt) 2013-01-14

Similar Documents

Publication Publication Date Title
MX2010007677A (es) Derivados de hidroximoil-tetrazol como fungicidas.
MX2010010135A (es) Derivados de hidroximoil-tetrazol fungicidas.
MX2010003258A (es) Utilizacion de un nuevo agente natural en composiciones cosmeticas.
WO2008036932A3 (en) Compositions and methods comprising boswellia species
EA033311B1 (ru) Производные бензоксаборола в качестве антибактериальных средств
MX2009013515A (es) Derivados de 7-alquinil-1,8-naftiridonas, su preparacion y su aplicacion en terapeutica.
MX2010014041A (es) Una forma cristalina de posaconazol.
GEP20125652B (en) cMET INHIBITORS
MX2009009948A (es) Derivados de piridazinona utiles como inhibidores de glucano sintasa.
WO2008132229A3 (en) Highly concentrated insulin solutions and compositions
BRPI0914343A2 (pt) composição, produto, uso da composição e método
MA32776B1 (fr) Inhibiteurs de l'akt et de la p70 s6 kinase
EA201101214A1 (ru) Полиеновые противогрибковые композиции
MA32544B1 (fr) Derives de pyridino-pyridinones, leur preparation et leur application en therapeutique
WO2009130616A3 (en) Improved tlr3 agonist compositions
MX342947B (es) Tratamiento de diabetes tipo 2.
MX2012010127A (es) Derivados de aminoindanos, su preparacion y su aplicacion en terapeuticos.
MY161601A (en) Films and compositions comprising the same
MX352553B (es) Composicion para el cuidado oral comprendiendo un compuesto de amadori.
NZ701463A (en) Anti-phytopathogenic composition
MX336392B (es) Derivados de hidroximoil-heterociclos fungicidas.
CL2012001757A1 (es) Compuestos derivados de 8-hidroxiquinolina-7-carboxamida; composicion farmaceutica; y su uso en el tratamiento de infecciones micoticas.
ATE545640T1 (de) Als geruchsstoffe geeignete isolongifolanylderivate
MX2010010017A (es) Derivados de guanidina lineales y ciclicos, metodo de preparacion y sus usos.
MX2013004878A (es) N-hetarilmetil pirazolilcarboxamidas.

Legal Events

Date Code Title Description
FG Grant or registration