MX2009005324A - Process for the synthesis of derivatives of 3-amino-tetrahydrofur an-3-carboxylic acid and use thereof as medicaments. - Google Patents
Process for the synthesis of derivatives of 3-amino-tetrahydrofur an-3-carboxylic acid and use thereof as medicaments.Info
- Publication number
- MX2009005324A MX2009005324A MX2009005324A MX2009005324A MX2009005324A MX 2009005324 A MX2009005324 A MX 2009005324A MX 2009005324 A MX2009005324 A MX 2009005324A MX 2009005324 A MX2009005324 A MX 2009005324A MX 2009005324 A MX2009005324 A MX 2009005324A
- Authority
- MX
- Mexico
- Prior art keywords
- amino
- carboxylic acid
- synthesis
- tetrahydrofur
- medicaments
- Prior art date
Links
- 230000015572 biosynthetic process Effects 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 238000003786 synthesis reaction Methods 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title 1
- 230000003287 optical effect Effects 0.000 abstract 3
- UYZGJJIHZKHDTQ-UHFFFAOYSA-N 3-aminooxolane-3-carboxamide Chemical class NC(=O)C1(N)CCOC1 UYZGJJIHZKHDTQ-UHFFFAOYSA-N 0.000 abstract 2
- 239000002243 precursor Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 150000007522 mineralic acids Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
- 235000005985 organic acids Nutrition 0.000 abstract 1
Landscapes
- Furan Compounds (AREA)
Abstract
The present invention relates to a process for the manufacturing of substituted 3- amino-tetrahydrofuran-3-carboxylic acid amides of general formula (I) and their precursors in high optical purity to the precursors of the synthesis of substituted S-Amino-tetrahydrofuran-S-carboxylic acid amides of general formula (I) in high optical purity, and to the tautomers, enantiomers, diastereomers, mixtures and salts of substituted 3-amino- tetrahydrofuran-3-carboxylic acid amides of general formula (I) in high optical purity, particularly the physiologically acceptable salts thereof with inorganic or organic acids or bases, which have valuable properties.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US89293706P | 2006-12-31 | 2006-12-31 | |
| PCT/EP2007/064406 WO2008080891A2 (en) | 2006-12-31 | 2007-12-21 | Process for the synthesis of derivatives of 3-amino-tetrahydrofuran-3-carboxylic acid and use thereof as medicaments |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2009005324A true MX2009005324A (en) | 2009-06-08 |
Family
ID=41559180
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2009005324A MX2009005324A (en) | 2006-12-31 | 2007-12-21 | Process for the synthesis of derivatives of 3-amino-tetrahydrofur an-3-carboxylic acid and use thereof as medicaments. |
Country Status (1)
| Country | Link |
|---|---|
| MX (1) | MX2009005324A (en) |
-
2007
- 2007-12-21 MX MX2009005324A patent/MX2009005324A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |