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MX2008000011A - Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes. - Google Patents

Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes.

Info

Publication number
MX2008000011A
MX2008000011A MX2008000011A MX2008000011A MX2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A
Authority
MX
Mexico
Prior art keywords
processes
sup
novel intermediates
glycoside derivatives
preparing
Prior art date
Application number
MX2008000011A
Other languages
Spanish (es)
Inventor
Waldemar Pfrengle
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of MX2008000011A publication Critical patent/MX2008000011A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

The present invention relates to processes for preparing the compounds of general formula I, wherein the groups R<sup>1</sup> to R<sup>6</sup> and R<sup>7a</sup>, R<sup>7b</sup>, R<sup>7c</sup> are defined according to claim 1. Furthermore the present invention relates to processes for preparing educts and intermediates in the above processes and to intermediates as such.
MX2008000011A 2005-07-22 2006-07-20 Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes. MX2008000011A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05015935 2005-07-22
PCT/EP2006/064435 WO2007010015A1 (en) 2005-07-22 2006-07-20 Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes

Publications (1)

Publication Number Publication Date
MX2008000011A true MX2008000011A (en) 2008-03-26

Family

ID=37102155

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2008000011A MX2008000011A (en) 2005-07-22 2006-07-20 Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes.

Country Status (14)

Country Link
EP (1) EP1910391A1 (en)
JP (2) JP4888840B2 (en)
KR (1) KR20080036112A (en)
CN (1) CN101218244A (en)
AR (1) AR054852A1 (en)
AU (1) AU2006271653A1 (en)
BR (1) BRPI0613690A2 (en)
CA (1) CA2621269A1 (en)
IL (1) IL188898A0 (en)
MX (1) MX2008000011A (en)
RU (1) RU2008106461A (en)
TW (1) TW200728286A (en)
WO (1) WO2007010015A1 (en)
ZA (1) ZA200709951B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2500873C (en) * 2002-10-04 2012-01-17 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, medicinal composition containing the same, medicinal use thereof and intermediate in producing the same
US7375090B2 (en) 2003-08-26 2008-05-20 Boehringer Ingelheim International Gmbh Glucopyranosyloxy-pyrazoles, pharmaceutical compositions containing these compounds, the use thereof and processed for the preparation thereof
UY29694A1 (en) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int METHODS TO PREVENT AND TREAT METABOLIC AND NEW DISORDERS DERIVED FROM PIRAZOL-O-GLUCOSIDO
UY30082A1 (en) 2006-01-11 2007-08-31 Boehringer Ingelheim Int CRYSTAL FORM OF 1- (1-METHYLETHYL) -4` - ((2-FLUORO-4-METOXIFENIL) METHYL) -5`- METHYL-1H-PIRAZOL-3`-OBD-GLUCOPYRANOSIDE, A METHOD FOR PREPARATION AND USE OF THE SAME TO PREPARE MEDICATIONS
WO2012133783A1 (en) * 2011-03-31 2012-10-04 キッセイ薬品工業株式会社 Method for producing benzylpyrazole derivative and production intermediate thereof

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55157504A (en) * 1979-05-24 1980-12-08 Sankyo Co Ltd Herbicide
WO2002036602A1 (en) * 2000-11-02 2002-05-10 Ajinomoto Co., Inc. Novel pyrazole derivatives and diabetes remedies containing the same
WO2002053573A1 (en) * 2000-12-28 2002-07-11 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivatives and use thereof in medicines
EP1364957B1 (en) * 2001-02-26 2008-12-31 Kissei Pharmaceutical Co., Ltd. Glycopyranosyloxypyrazole derivatives and medicinal use thereof
EP1364958B1 (en) * 2001-02-27 2010-09-08 Kissei Pharmaceutical Co., Ltd. Glycopyranosyloxypyrazole derivatives and medicinal use thereof
CA2672001A1 (en) * 2001-04-27 2002-11-07 Ajinomoto Co., Inc. N-substituted pyrazole-o-glycoside derivatives and therapeutic agent for diabetes containing the same
CA2448741C (en) * 2001-05-30 2010-06-22 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor
US20030087843A1 (en) * 2001-09-05 2003-05-08 Washburn William N. O-pyrazole glucoside SGLT2 inhibitors and method of use
JP4424203B2 (en) * 2002-04-26 2010-03-03 味の素株式会社 Diabetes prevention and treatment
DE60332743D1 (en) * 2002-08-08 2010-07-08 Kissei Pharmaceutical PYRAZOL DERIVATIVE, MEDICAL COMPOSITION, MEDICAL USE THEREOF, AND INTERMEDIATE PRODUCT FOR THE PRODUCTION THEREOF
JP2004137245A (en) * 2002-08-23 2004-05-13 Kissei Pharmaceut Co Ltd Pyrazole derivative, pharmaceutical composition containing the same, its pharmaceutical use and production intermediate
JP4606876B2 (en) * 2002-08-27 2011-01-05 キッセイ薬品工業株式会社 Pyrazole derivative, pharmaceutical composition containing the same, and pharmaceutical use thereof
CA2500873C (en) * 2002-10-04 2012-01-17 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, medicinal composition containing the same, medicinal use thereof and intermediate in producing the same
WO2004089966A1 (en) * 2003-04-01 2004-10-21 Taisho Pharmaceutical Co., Ltd. METHOD FOR SELECTIVE PREPARATION OF HETEROARYL 5-THIO- β-D-ALDOHEXOPYRANOSIDE
ES2377741T3 (en) * 2003-06-20 2012-03-30 Kissei Pharmaceutical Co., Ltd. Pyrazole derivatives, pharmacological composition that contains them and production intermediates thereof
UY29694A1 (en) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int METHODS TO PREVENT AND TREAT METABOLIC AND NEW DISORDERS DERIVED FROM PIRAZOL-O-GLUCOSIDO

Also Published As

Publication number Publication date
AU2006271653A1 (en) 2007-01-25
JP2009502763A (en) 2009-01-29
JP4888840B2 (en) 2012-02-29
IL188898A0 (en) 2008-04-13
AR054852A1 (en) 2007-07-18
CA2621269A1 (en) 2007-01-25
JP2012006956A (en) 2012-01-12
WO2007010015A1 (en) 2007-01-25
ZA200709951B (en) 2008-11-26
RU2008106461A (en) 2009-08-27
EP1910391A1 (en) 2008-04-16
CN101218244A (en) 2008-07-09
TW200728286A (en) 2007-08-01
KR20080036112A (en) 2008-04-24
BRPI0613690A2 (en) 2011-01-25

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal