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MX2008000011A - Procesos para preparar derivados de pirazol-o-glucosido y nuevos intermediarios de dichos procesos. - Google Patents

Procesos para preparar derivados de pirazol-o-glucosido y nuevos intermediarios de dichos procesos.

Info

Publication number
MX2008000011A
MX2008000011A MX2008000011A MX2008000011A MX2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A MX 2008000011 A MX2008000011 A MX 2008000011A
Authority
MX
Mexico
Prior art keywords
processes
sup
novel intermediates
glycoside derivatives
preparing
Prior art date
Application number
MX2008000011A
Other languages
English (en)
Inventor
Waldemar Pfrengle
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of MX2008000011A publication Critical patent/MX2008000011A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18One oxygen or sulfur atom
    • C07D231/20One oxygen atom attached in position 3 or 5
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La presente invencion se refiere a procesos para preparar los compuestos de la formula general I, (ver formula I) en donde los grupos R1 a R6 y R7a, R7b, R7c se definen de acuerdo con la reivindiccion 1. Ademas, la presente invencion se refiere a p4rocesos para preparar eductos e intermedios en los procesos anteriores y a los intermediarios como tales.
MX2008000011A 2005-07-22 2006-07-20 Procesos para preparar derivados de pirazol-o-glucosido y nuevos intermediarios de dichos procesos. MX2008000011A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05015935 2005-07-22
PCT/EP2006/064435 WO2007010015A1 (en) 2005-07-22 2006-07-20 Processes for preparing pyrazole-o-glycoside derivatives and novel intermediates of said processes

Publications (1)

Publication Number Publication Date
MX2008000011A true MX2008000011A (es) 2008-03-26

Family

ID=37102155

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2008000011A MX2008000011A (es) 2005-07-22 2006-07-20 Procesos para preparar derivados de pirazol-o-glucosido y nuevos intermediarios de dichos procesos.

Country Status (14)

Country Link
EP (1) EP1910391A1 (es)
JP (2) JP4888840B2 (es)
KR (1) KR20080036112A (es)
CN (1) CN101218244A (es)
AR (1) AR054852A1 (es)
AU (1) AU2006271653A1 (es)
BR (1) BRPI0613690A2 (es)
CA (1) CA2621269A1 (es)
IL (1) IL188898A0 (es)
MX (1) MX2008000011A (es)
RU (1) RU2008106461A (es)
TW (1) TW200728286A (es)
WO (1) WO2007010015A1 (es)
ZA (1) ZA200709951B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2500873C (en) * 2002-10-04 2012-01-17 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, medicinal composition containing the same, medicinal use thereof and intermediate in producing the same
US7375090B2 (en) 2003-08-26 2008-05-20 Boehringer Ingelheim International Gmbh Glucopyranosyloxy-pyrazoles, pharmaceutical compositions containing these compounds, the use thereof and processed for the preparation thereof
UY29694A1 (es) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int Metodos para prevenir y tratar trastornos metabolicos y nuevos derivados de pirazol-o-glucosido
UY30082A1 (es) 2006-01-11 2007-08-31 Boehringer Ingelheim Int Forma cristalina de 1-(1-metiletil)-4`-((2-fluoro-4-metoxifenil)metil)-5`- metil-1h-pirazol-3`-o-b-d-glucopiranosido, un metodo para su preparacion y el uso de la misma para preparar medicamentos
WO2012133783A1 (ja) * 2011-03-31 2012-10-04 キッセイ薬品工業株式会社 ベンジルピラゾール誘導体の製造方法およびその製造中間体

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55157504A (en) * 1979-05-24 1980-12-08 Sankyo Co Ltd Herbicide
WO2002036602A1 (en) * 2000-11-02 2002-05-10 Ajinomoto Co., Inc. Novel pyrazole derivatives and diabetes remedies containing the same
WO2002053573A1 (en) * 2000-12-28 2002-07-11 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivatives and use thereof in medicines
EP1364957B1 (en) * 2001-02-26 2008-12-31 Kissei Pharmaceutical Co., Ltd. Glycopyranosyloxypyrazole derivatives and medicinal use thereof
EP1364958B1 (en) * 2001-02-27 2010-09-08 Kissei Pharmaceutical Co., Ltd. Glycopyranosyloxypyrazole derivatives and medicinal use thereof
CA2672001A1 (en) * 2001-04-27 2002-11-07 Ajinomoto Co., Inc. N-substituted pyrazole-o-glycoside derivatives and therapeutic agent for diabetes containing the same
CA2448741C (en) * 2001-05-30 2010-06-22 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor
US20030087843A1 (en) * 2001-09-05 2003-05-08 Washburn William N. O-pyrazole glucoside SGLT2 inhibitors and method of use
JP4424203B2 (ja) * 2002-04-26 2010-03-03 味の素株式会社 糖尿病予防・治療剤
DE60332743D1 (de) * 2002-08-08 2010-07-08 Kissei Pharmaceutical Pyrazolderivat, dieses enthaltende medizinische zusammensetzung, medizinische verwendung davon, und zwischenprodukt für dessen herstellung
JP2004137245A (ja) * 2002-08-23 2004-05-13 Kissei Pharmaceut Co Ltd ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体
JP4606876B2 (ja) * 2002-08-27 2011-01-05 キッセイ薬品工業株式会社 ピラゾール誘導体、それを含有する医薬組成物及びその医薬用途
CA2500873C (en) * 2002-10-04 2012-01-17 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, medicinal composition containing the same, medicinal use thereof and intermediate in producing the same
WO2004089966A1 (ja) * 2003-04-01 2004-10-21 Taisho Pharmaceutical Co., Ltd. 選択的なヘテロアリール 5-チオ-β-D-アルドヘキソピラノシドの製造法
ES2377741T3 (es) * 2003-06-20 2012-03-30 Kissei Pharmaceutical Co., Ltd. Derivados de pirazol, composición farmacológica que los contiene e intermedios de producción de los mismos
UY29694A1 (es) * 2005-07-28 2007-02-28 Boehringer Ingelheim Int Metodos para prevenir y tratar trastornos metabolicos y nuevos derivados de pirazol-o-glucosido

Also Published As

Publication number Publication date
AU2006271653A1 (en) 2007-01-25
JP2009502763A (ja) 2009-01-29
JP4888840B2 (ja) 2012-02-29
IL188898A0 (en) 2008-04-13
AR054852A1 (es) 2007-07-18
CA2621269A1 (en) 2007-01-25
JP2012006956A (ja) 2012-01-12
WO2007010015A1 (en) 2007-01-25
ZA200709951B (en) 2008-11-26
RU2008106461A (ru) 2009-08-27
EP1910391A1 (en) 2008-04-16
CN101218244A (zh) 2008-07-09
TW200728286A (en) 2007-08-01
KR20080036112A (ko) 2008-04-24
BRPI0613690A2 (pt) 2011-01-25

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Legal Events

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FA Abandonment or withdrawal