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MX2007013263A - Novedosos derivados oxadiazol y su uso medico. - Google Patents

Novedosos derivados oxadiazol y su uso medico.

Info

Publication number
MX2007013263A
MX2007013263A MX2007013263A MX2007013263A MX2007013263A MX 2007013263 A MX2007013263 A MX 2007013263A MX 2007013263 A MX2007013263 A MX 2007013263A MX 2007013263 A MX2007013263 A MX 2007013263A MX 2007013263 A MX2007013263 A MX 2007013263A
Authority
MX
Mexico
Prior art keywords
diseases
disorders
oxadiazole derivatives
medical use
novel oxadiazole
Prior art date
Application number
MX2007013263A
Other languages
English (en)
Inventor
Dan Peters
Gunnar M Olsen
Bjarne H Dahl
Daniel B Timmermann
Sussane J Jorgensen
Original Assignee
Neurosearch As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurosearch As filed Critical Neurosearch As
Publication of MX2007013263A publication Critical patent/MX2007013263A/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)

Abstract

Esta invencion se relaciona con novedosos derivados oxadiazol de la formula (I) que se descubrio son moduladores de receptores nicotinicos de acetilcolina. Debido a su perfil farmacologico, los compuestos de la invencion pueden ser utiles para el tratamiento contra enfermedades o trastornos tan diversos como aquellos relacionados con el sistema colinergico del sistema nervioso central (SNC) al sistema nervioso periferico (SNP), con enfermedades o trastornos relacionados con la contraccion del musculo liso, enfermedades o trastornos endocrinos, enfermedades o trastornos relacionados con neurodegeneracion, enfermedades o trastornos relacionados con inflamacion, dolor y sintomas de abstinencia causador por dejar de abusar de sustancias quimicas.
MX2007013263A 2005-04-26 2006-04-24 Novedosos derivados oxadiazol y su uso medico. MX2007013263A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67471105P 2005-04-26 2005-04-26
DKPA200500612 2005-04-26
PCT/EP2006/061773 WO2006114400A1 (en) 2005-04-26 2006-04-24 Novel oxadiazole derivatives and their medical use

Publications (1)

Publication Number Publication Date
MX2007013263A true MX2007013263A (es) 2008-01-22

Family

ID=36697471

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007013263A MX2007013263A (es) 2005-04-26 2006-04-24 Novedosos derivados oxadiazol y su uso medico.

Country Status (12)

Country Link
US (2) US8017631B2 (es)
EP (1) EP1881979B1 (es)
JP (1) JP2008539195A (es)
KR (1) KR20080000622A (es)
AT (1) ATE477253T1 (es)
AU (1) AU2006239418A1 (es)
CA (1) CA2606087A1 (es)
IL (1) IL186360A0 (es)
MX (1) MX2007013263A (es)
NO (1) NO20076036L (es)
RU (1) RU2007139255A (es)
WO (1) WO2006114400A1 (es)

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