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MA32385B1 - Forme posologique pharmaceutique en capsule comprenant une formulation en suspension d'un derive d'indolinone - Google Patents

Forme posologique pharmaceutique en capsule comprenant une formulation en suspension d'un derive d'indolinone

Info

Publication number
MA32385B1
MA32385B1 MA33402A MA33402A MA32385B1 MA 32385 B1 MA32385 B1 MA 32385B1 MA 33402 A MA33402 A MA 33402A MA 33402 A MA33402 A MA 33402A MA 32385 B1 MA32385 B1 MA 32385B1
Authority
MA
Morocco
Prior art keywords
capsule
dosage form
pharmaceutical dosage
suspension formulation
indolinone derivative
Prior art date
Application number
MA33402A
Other languages
Arabic (ar)
English (en)
Inventor
Thomas Bock
Werner Brox
Roman Messerschmid
Rudolf Binder
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40911908&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA32385(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of MA32385B1 publication Critical patent/MA32385B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816Wall or shell material
    • A61K9/4825Proteins, e.g. gelatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61JCONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
    • A61J1/00Containers specially adapted for medical or pharmaceutical purposes
    • A61J1/03Containers specially adapted for medical or pharmaceutical purposes for pills or tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4808Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816Wall or shell material
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5052Proteins, e.g. albumin
    • A61K9/5057Gelatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La présente invention concerne une formulation en suspension dont le principe actif est le 3-z-[1-(4- (n-((4-méthyl-pipérazin-1-yl)-méthylcarbonyl)-n-méthyl-amino)-anilino)-1-phényl-méthylène]-6- méthoxycarbonyl-2- indolinone-monoéthane-sulphonate. L'invention concerne également, d'une part une forme posologique pharmaceutique en capsule contenant ladite formulation en suspension, d'autre part un procédé d'élaboration de ladite formulation en suspension, mais aussi un procédé d'élaboration de ladite capsule comprenant ladite formulation en suspension, et également le matériau d'enveloppe de la capsule.
MA33402A 2008-06-06 2010-12-06 Forme posologique pharmaceutique en capsule comprenant une formulation en suspension d'un derive d'indolinone MA32385B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08157748 2008-06-06
PCT/EP2009/056878 WO2009147212A1 (fr) 2008-06-06 2009-06-04 Forme posologique pharmaceutique en capsule comprenant une formulation en suspension d'un dérivé d'indolinone

Publications (1)

Publication Number Publication Date
MA32385B1 true MA32385B1 (fr) 2011-06-01

Family

ID=40911908

Family Applications (1)

Application Number Title Priority Date Filing Date
MA33402A MA32385B1 (fr) 2008-06-06 2010-12-06 Forme posologique pharmaceutique en capsule comprenant une formulation en suspension d'un derive d'indolinone

Country Status (35)

Country Link
US (4) US20110301177A1 (fr)
EP (1) EP2299987B1 (fr)
JP (2) JP5661031B2 (fr)
KR (2) KR20170020557A (fr)
CN (2) CN105193720B (fr)
AR (1) AR072059A1 (fr)
AU (1) AU2009254548B2 (fr)
BR (1) BRPI0913434B8 (fr)
CA (1) CA2726267C (fr)
CL (1) CL2010001279A1 (fr)
CO (1) CO6280467A2 (fr)
CY (1) CY1120533T1 (fr)
DK (1) DK2299987T3 (fr)
EA (1) EA029996B1 (fr)
EC (1) ECSP10010660A (fr)
ES (1) ES2669469T3 (fr)
HR (1) HRP20180709T1 (fr)
HU (1) HUE039187T2 (fr)
IL (1) IL208954A (fr)
LT (1) LT2299987T (fr)
MA (1) MA32385B1 (fr)
MX (2) MX359229B (fr)
MY (1) MY158930A (fr)
NO (1) NO2299987T3 (fr)
NZ (1) NZ603162A (fr)
PE (1) PE20100254A1 (fr)
PL (1) PL2299987T3 (fr)
PT (1) PT2299987T (fr)
RS (1) RS57142B1 (fr)
SI (1) SI2299987T1 (fr)
TW (1) TW201002691A (fr)
UA (1) UA104590C2 (fr)
UY (1) UY31879A (fr)
WO (1) WO2009147212A1 (fr)
ZA (1) ZA201007636B (fr)

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EP4125890A1 (fr) 2020-04-01 2023-02-08 Boehringer Ingelheim International GmbH Utilisation de biomarqueurs dans le traitement d'états fibrotiques
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Also Published As

Publication number Publication date
AU2009254548A1 (en) 2009-12-10
LT2299987T (lt) 2018-05-25
JP2011522812A (ja) 2011-08-04
PL2299987T3 (pl) 2018-08-31
HUE039187T2 (hu) 2018-12-28
IL208954A0 (en) 2011-01-31
CN105193720B (zh) 2018-07-31
DK2299987T3 (en) 2018-05-22
US20160324791A1 (en) 2016-11-10
NO2299987T3 (fr) 2018-07-21
KR101725469B1 (ko) 2017-04-11
PE20100254A1 (es) 2010-04-21
NZ603162A (en) 2014-05-30
EA029996B1 (ru) 2018-06-29
JP5661031B2 (ja) 2015-01-28
ZA201007636B (en) 2011-08-31
US20110301177A1 (en) 2011-12-08
CO6280467A2 (es) 2011-05-20
TW201002691A (en) 2010-01-16
CN102056598B (zh) 2017-09-19
HRP20180709T1 (hr) 2018-06-15
ES2669469T3 (es) 2018-05-25
MX2010013203A (es) 2011-02-25
JP5905542B2 (ja) 2016-04-20
RS57142B1 (sr) 2018-07-31
CA2726267A1 (fr) 2009-12-10
CN105193720A (zh) 2015-12-30
SI2299987T1 (en) 2018-06-29
US20160022672A1 (en) 2016-01-28
UY31879A (es) 2010-01-29
MX359229B (es) 2018-09-20
BRPI0913434A2 (pt) 2015-12-01
EP2299987B1 (fr) 2018-02-21
UA104590C2 (ru) 2014-02-25
CY1120533T1 (el) 2019-07-10
IL208954A (en) 2017-11-30
US9907756B2 (en) 2018-03-06
ECSP10010660A (es) 2011-02-28
US20140004187A1 (en) 2014-01-02
MY158930A (en) 2016-11-30
EA201001856A1 (ru) 2011-06-30
WO2009147212A1 (fr) 2009-12-10
JP2014208712A (ja) 2014-11-06
PT2299987T (pt) 2018-05-21
EP2299987A1 (fr) 2011-03-30
BRPI0913434B1 (pt) 2020-10-13
KR20110017872A (ko) 2011-02-22
AU2009254548B2 (en) 2015-10-01
BRPI0913434B8 (pt) 2021-05-25
CA2726267C (fr) 2017-10-31
AR072059A1 (es) 2010-08-04
CL2010001279A1 (es) 2011-05-13
CN102056598A (zh) 2011-05-11
KR20170020557A (ko) 2017-02-22

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