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MA31785B1 - Nouveaux dérivés d'imidazole - Google Patents

Nouveaux dérivés d'imidazole

Info

Publication number
MA31785B1
MA31785B1 MA32785A MA32785A MA31785B1 MA 31785 B1 MA31785 B1 MA 31785B1 MA 32785 A MA32785 A MA 32785A MA 32785 A MA32785 A MA 32785A MA 31785 B1 MA31785 B1 MA 31785B1
Authority
MA
Morocco
Prior art keywords
halogen
haloalkyl
alkyl
imidazole derivatives
haloalkoxy
Prior art date
Application number
MA32785A
Other languages
Arabic (ar)
English (en)
Inventor
Raphael Dumeunier
Clemens Lamberth
Stephan Trah
Sebastian Wendeborn
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP07020982A external-priority patent/EP2053045A1/fr
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of MA31785B1 publication Critical patent/MA31785B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Cette invention concerne des nouveaux dérivés d'imidaloze représentés par la formule (i) utilisés en tant que principes actifs et présentant une activité microbicide, plus particulièrement, une activité fongicide: dans cette formule, r1 représente, alkyle c1-c4 ou haloalkyle c1-c4; r2 représente un aryle éventuellement substitué ou un hétéroaryle; r3 représente halogène; r4 représente hydrogène, halogène, alkyle c1-c4, haloalkyle c1-c4, alkoxy c1-c4, haloalkoxy c1-c4 ou cyano; r5 représente halogène; x représente n ou c(r); et r représente hydrogène, halogène, alkyle c1-c4, haloalkyle c1-c4, alkoxy c1-c4, haloalkoxy c1-c4ou cyano; ou une forme saline de ceux-ci utilisable au plan agrochimique; sous réserve que lorsque x représente c(r), r2 ne peut être un aryle éventuellement substitué.
MA32785A 2007-10-26 2010-04-22 Nouveaux dérivés d'imidazole MA31785B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07020982A EP2053045A1 (fr) 2007-10-26 2007-10-26 Nouveaux dérivés d'imidazole
EP07024449 2007-12-17
PCT/EP2008/009043 WO2009053102A1 (fr) 2007-10-26 2008-10-24 Nouveaux dérivés d'imidazole

Publications (1)

Publication Number Publication Date
MA31785B1 true MA31785B1 (fr) 2010-10-01

Family

ID=42719243

Family Applications (1)

Application Number Title Priority Date Filing Date
MA32785A MA31785B1 (fr) 2007-10-26 2010-04-22 Nouveaux dérivés d'imidazole

Country Status (16)

Country Link
US (1) US20110224252A1 (fr)
JP (1) JP2011500750A (fr)
KR (1) KR20100101580A (fr)
CN (1) CN101835773A (fr)
AR (1) AR069037A1 (fr)
AT (1) ATE522517T1 (fr)
BR (1) BRPI0818855A2 (fr)
CL (1) CL2008003178A1 (fr)
CO (1) CO6190578A2 (fr)
EA (1) EA201000619A1 (fr)
GT (1) GT200800229A (fr)
IL (1) IL205148A0 (fr)
MA (1) MA31785B1 (fr)
NZ (1) NZ584387A (fr)
TW (1) TW200926981A (fr)
ZA (1) ZA201002439B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2007281911B2 (en) * 2006-08-04 2014-02-06 Beth Israel Deaconess Medical Center Inhibitors of pyruvate kinase and methods of treating disease
AU2010234526B2 (en) 2009-04-06 2016-07-21 Agios Pharmaceuticals, Inc. Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use
WO2010129596A1 (fr) 2009-05-04 2010-11-11 Agios Pharmaceuticals, Inc. Inhibiteurs de la pkm2 destinés à être utilisés dans le traitement du cancer
JP5856052B2 (ja) 2009-06-29 2016-02-09 アジオス ファーマシューティカルズ， インコーポレイテッド 治療化合物および組成物
EP2448581B1 (fr) 2009-06-29 2016-12-07 Agios Pharmaceuticals, Inc. Compositions thérapeutiques et procédés d'utilisation associés
US9221792B2 (en) 2010-12-17 2015-12-29 Agios Pharmaceuticals, Inc N-(4-(azetidine-1-carbonyl) phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase M2 (PMK2) modulators
CA2822432C (fr) 2010-12-21 2019-09-24 Agios Pharmaceuticals, Inc. Activateurs bicycliques de pkm2
TWI549947B (zh) 2010-12-29 2016-09-21 阿吉歐斯製藥公司 治療化合物及組成物
US9181231B2 (en) 2011-05-03 2015-11-10 Agios Pharmaceuticals, Inc Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia
PH12017501176B1 (en) 2011-05-03 2023-03-08 Agios Pharmaceuticals Inc Pyruvate kinase activators for use in therapy
WO2014139144A1 (fr) 2013-03-15 2014-09-18 Agios Pharmaceuticals, Inc. Composés et compositions thérapeutiques
HUE063541T2 (hu) 2015-06-11 2024-01-28 Agios Pharmaceuticals Inc Eljárások piruvát-kináz aktivátorok alkalmazására
CN109810062B (zh) * 2019-01-24 2022-06-17 云南农业大学 一种苯基咪唑衍生物及其合成方法和在农药中的应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL338191A1 (en) * 1997-07-24 2000-10-09 Bayer Ag Nitrophenylsulphonyl imidazoles and their application in fighting against plant and animal pests

Also Published As

Publication number Publication date
CL2008003178A1 (es) 2009-06-05
AR069037A1 (es) 2009-12-23
ATE522517T1 (de) 2011-09-15
IL205148A0 (en) 2010-11-30
ZA201002439B (en) 2011-06-29
CN101835773A (zh) 2010-09-15
TW200926981A (en) 2009-07-01
NZ584387A (en) 2011-10-28
KR20100101580A (ko) 2010-09-17
CO6190578A2 (es) 2010-08-19
GT200800229A (es) 2010-04-20
JP2011500750A (ja) 2011-01-06
BRPI0818855A2 (pt) 2015-04-14
EA201000619A1 (ru) 2010-10-29
US20110224252A1 (en) 2011-09-15

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