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ZA9410040B - Non-peptide tachykinin receptor antagonists - Google Patents

Non-peptide tachykinin receptor antagonists

Info

Publication number
ZA9410040B
ZA9410040B ZA9410040A ZA9410040A ZA9410040B ZA 9410040 B ZA9410040 B ZA 9410040B ZA 9410040 A ZA9410040 A ZA 9410040A ZA 9410040 A ZA9410040 A ZA 9410040A ZA 9410040 B ZA9410040 B ZA 9410040B
Authority
ZA
South Africa
Prior art keywords
receptor antagonists
tachykinin receptor
peptide tachykinin
peptide
antagonists
Prior art date
Application number
ZA9410040A
Other languages
English (en)
Inventor
Thomas Alan Crowell
Charles David Jones
Bruce Donald Gitter
William Henry Walker Lunn
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of ZA9410040B publication Critical patent/ZA9410040B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/80—Radicals substituted by oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Furan Compounds (AREA)
ZA9410040A 1993-12-21 1994-12-15 Non-peptide tachykinin receptor antagonists ZA9410040B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17113493A 1993-12-21 1993-12-21

Publications (1)

Publication Number Publication Date
ZA9410040B true ZA9410040B (en) 1996-06-18

Family

ID=22622667

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9410040A ZA9410040B (en) 1993-12-21 1994-12-15 Non-peptide tachykinin receptor antagonists

Country Status (7)

Country Link
EP (1) EP0736007A4 (es)
JP (1) JPH09506898A (es)
AU (1) AU1339795A (es)
CA (1) CA2176130A1 (es)
MX (1) MXPA99001870A (es)
WO (1) WO1995017382A1 (es)
ZA (1) ZA9410040B (es)

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DE69824410T2 (de) 1997-04-30 2005-06-02 Eli Lilly And Co., Indianapolis Antithrombosemittel
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EP1027051B1 (en) 1997-04-30 2005-01-05 Eli Lilly And Company Antithrombotic agents
US6284756B1 (en) 1998-04-30 2001-09-04 Eli Lilly And Company Antithrombotic agents
DE69904427T2 (de) * 1998-10-28 2003-07-17 Eli Lilly And Co., Indianapolis Benzothiophenderivate als antithrombotische Mitteln und Zwischenprodukte
WO2001032625A1 (en) 1999-11-03 2001-05-10 Du Pont Pharmaceuticals Company Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine and serotonin
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KR102196882B1 (ko) 2012-12-20 2020-12-30 머크 샤프 앤드 돔 코포레이션 Hdm2 억제제로서의 치환된 이미다조피리딘
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Also Published As

Publication number Publication date
WO1995017382A1 (en) 1995-06-29
JPH09506898A (ja) 1997-07-08
AU1339795A (en) 1995-07-10
EP0736007A4 (en) 1997-03-19
CA2176130A1 (en) 1995-06-29
MXPA99001870A (es) 2004-09-06
EP0736007A1 (en) 1996-10-09

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