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WO2000061574A3 - Procede de production d'amidines - Google Patents

Procede de production d'amidines Download PDF

Info

Publication number
WO2000061574A3
WO2000061574A3 PCT/EP2000/003018 EP0003018W WO0061574A3 WO 2000061574 A3 WO2000061574 A3 WO 2000061574A3 EP 0003018 W EP0003018 W EP 0003018W WO 0061574 A3 WO0061574 A3 WO 0061574A3
Authority
WO
WIPO (PCT)
Prior art keywords
amidines
producing
thiophenyl
amidoximes
reacted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/EP2000/003018
Other languages
German (de)
English (en)
Other versions
WO2000061574A2 (fr
Inventor
Thomas Zierke
Helmut Mack
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Priority to AU35590/00A priority Critical patent/AU3559000A/en
Priority to JP2000610848A priority patent/JP2002541252A/ja
Priority to CA002369267A priority patent/CA2369267A1/fr
Priority to EP00914182A priority patent/EP1169315A2/fr
Publication of WO2000061574A2 publication Critical patent/WO2000061574A2/fr
Publication of WO2000061574A3 publication Critical patent/WO2000061574A3/fr
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B43/00—Formation or introduction of functional groups containing nitrogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)

Abstract

Procédé permettant de produire des amidines non substituées au niveau de l'atome d'azote et leurs sels d'acides inorganiques ou organiques, qui consiste à faire réagir les amidoximes carboxyliques correspondantes avec du Zn en présence d'acides carboxyliques.
PCT/EP2000/003018 1999-04-09 2000-04-05 Procede de production d'amidines Ceased WO2000061574A2 (fr)

Priority Applications (4)

Application Number Priority Date Filing Date Title
AU35590/00A AU3559000A (en) 1999-04-09 2000-04-05 Method for producing amidines
JP2000610848A JP2002541252A (ja) 1999-04-09 2000-04-05 アミジンの製造
CA002369267A CA2369267A1 (fr) 1999-04-09 2000-04-05 Procede de production d'amidines
EP00914182A EP1169315A2 (fr) 1999-04-09 2000-04-05 Procede de production d'amidines

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19915930.0 1999-04-09
DE19915930 1999-04-09
DE19933873 1999-07-23
DE19933873.6 1999-07-23

Publications (2)

Publication Number Publication Date
WO2000061574A2 WO2000061574A2 (fr) 2000-10-19
WO2000061574A3 true WO2000061574A3 (fr) 2001-04-26

Family

ID=26052817

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2000/003018 Ceased WO2000061574A2 (fr) 1999-04-09 2000-04-05 Procede de production d'amidines

Country Status (5)

Country Link
EP (1) EP1169315A2 (fr)
JP (1) JP2002541252A (fr)
AU (1) AU3559000A (fr)
CA (1) CA2369267A1 (fr)
WO (1) WO2000061574A2 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1489575A (zh) * 2001-01-29 2004-04-14 ������������ʽ���� 苯甲脒衍生物及其制备方法
WO2006101860A1 (fr) * 2005-03-16 2006-09-28 Janssen Pharmaceutica N.V. Nouveaux composes de thiophene sulfoximine destines a traiter des maladies et des etats pathologiques associes au complement

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2375611A (en) * 1941-08-19 1945-05-08 May & Baker Ltd Production of amidines
US2851490A (en) * 1955-04-20 1958-09-09 Monsanto Chemicals Guanyl aliphatic mono-carboxylic acids
WO1998006741A1 (fr) * 1996-08-14 1998-02-19 Basf Aktiengesellschaft Inhibiteurs de la thrombine

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2375611A (en) * 1941-08-19 1945-05-08 May & Baker Ltd Production of amidines
US2851490A (en) * 1955-04-20 1958-09-09 Monsanto Chemicals Guanyl aliphatic mono-carboxylic acids
WO1998006741A1 (fr) * 1996-08-14 1998-02-19 Basf Aktiengesellschaft Inhibiteurs de la thrombine

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
F. ELOY ET AL.: "THE CHEMISTRY OF AMIDOXIMES AND RELATED COMPOUNDS", CHEMICAL REVIEWS., vol. 62, 1962, AMERICAN CHEMICAL SOCIETY. EASTON., US, pages 155 - 183, XP002151891, ISSN: 0009-2665 *

Also Published As

Publication number Publication date
EP1169315A2 (fr) 2002-01-09
JP2002541252A (ja) 2002-12-03
AU3559000A (en) 2000-11-14
CA2369267A1 (fr) 2000-10-19
WO2000061574A2 (fr) 2000-10-19

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